IL64506A - 7beta-(2-(2-amino-4-thiazolyl)-2-(syn)-methoxyiminoacetamido)-3-cephem-4-carboxylic acid esters,their production and pharmaceutical compositions containing them - Google Patents

7beta-(2-(2-amino-4-thiazolyl)-2-(syn)-methoxyiminoacetamido)-3-cephem-4-carboxylic acid esters,their production and pharmaceutical compositions containing them

Info

Publication number
IL64506A
IL64506A IL64506A IL6450681A IL64506A IL 64506 A IL64506 A IL 64506A IL 64506 A IL64506 A IL 64506A IL 6450681 A IL6450681 A IL 6450681A IL 64506 A IL64506 A IL 64506A
Authority
IL
Israel
Prior art keywords
7beta
methoxyiminoacetamido
cephem
syn
thiazolyl
Prior art date
Application number
IL64506A
Other languages
English (en)
Other versions
IL64506A0 (en
Original Assignee
Ciba Geigy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy filed Critical Ciba Geigy
Publication of IL64506A0 publication Critical patent/IL64506A0/xx
Publication of IL64506A publication Critical patent/IL64506A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL64506A 1980-12-12 1981-12-10 7beta-(2-(2-amino-4-thiazolyl)-2-(syn)-methoxyiminoacetamido)-3-cephem-4-carboxylic acid esters,their production and pharmaceutical compositions containing them IL64506A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH919680 1980-12-12

Publications (2)

Publication Number Publication Date
IL64506A0 IL64506A0 (en) 1982-03-31
IL64506A true IL64506A (en) 1985-05-31

Family

ID=4349398

Family Applications (1)

Application Number Title Priority Date Filing Date
IL64506A IL64506A (en) 1980-12-12 1981-12-10 7beta-(2-(2-amino-4-thiazolyl)-2-(syn)-methoxyiminoacetamido)-3-cephem-4-carboxylic acid esters,their production and pharmaceutical compositions containing them

Country Status (18)

Country Link
EP (1) EP0054512A3 (xx)
JP (1) JPS57123190A (xx)
KR (1) KR830007683A (xx)
AR (1) AR231984A1 (xx)
AU (1) AU7846681A (xx)
DD (1) DD208155A5 (xx)
DK (1) DK550081A (xx)
ES (6) ES8303424A1 (xx)
FI (1) FI813946L (xx)
GB (1) GB2111043B (xx)
GR (1) GR76967B (xx)
HU (1) HU185985B (xx)
IE (1) IE52008B1 (xx)
IL (1) IL64506A (xx)
NO (1) NO814232L (xx)
NZ (1) NZ199255A (xx)
PT (1) PT74119B (xx)
ZA (1) ZA818622B (xx)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES507942A0 (es) * 1980-12-15 1983-02-01 Fujisawa Pharmaceutical Co Un procedimiento para preparar derivados del acido 7-acilaminocefalosporanico .
JPS57156495A (en) * 1981-03-23 1982-09-27 Kyoto Yakuhin Kogyo Kk Cephalosporin derivative and remedy for microbism used in oral administration
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
JPS59116291A (ja) * 1982-12-06 1984-07-05 Fujisawa Pharmaceut Co Ltd ７−置換−３−セフエム−４−カルボン酸エステルおよびその製法
US5202454A (en) * 1986-07-11 1993-04-13 Societe Nationale Des Poudres Et Explosifs Process for the manufacture of 1-bromoalkyl hydrocarbyl carbonates
EP0497978B1 (en) * 1989-10-28 1997-04-16 Kyoto Pharmaceutical Industries, Ltd. Cephalosporin compounds and production thereof
ES2198003T3 (es) * 1996-07-26 2004-01-16 Gilead Sciences, Inc. Analogos de nucleotidos.
US20040224917A1 (en) 2003-01-14 2004-11-11 Gilead Sciences, Inc. Compositions and methods for combination antiviral therapy
TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
TWI375560B (en) 2005-06-13 2012-11-01 Gilead Sciences Inc Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3965099A (en) * 1974-06-26 1976-06-22 Smithkline Corporation Cephalosporin esters with antibacterial activity
JPS5321192A (en) * 1976-08-10 1978-02-27 Takeda Chem Ind Ltd Cephalosporin derivatives and their preparation
US4370326A (en) * 1977-09-13 1983-01-25 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds and composition
ZA793391B (en) * 1978-07-07 1980-06-25 Ciba Geigy Ag Aminothiazole compounds
MA18686A1 (fr) * 1978-07-07 1980-10-01 Ciba Geigy Ag Composes aminothiazoliques
JPS5543011A (en) * 1978-09-20 1980-03-26 Shionogi & Co Ltd 7-halothiazolylalkoxyiminoacetamido-3-cephem compound
GR78221B (xx) * 1980-02-01 1984-09-26 Ciba Geigy Ag

Also Published As

Publication number Publication date
NZ199255A (en) 1985-08-30
IE812915L (en) 1982-06-12
ES516590A0 (es) 1983-11-16
ES8307820A1 (es) 1983-08-01
AR231984A1 (es) 1985-04-30
PT74119A (de) 1982-01-01
ES516592A0 (es) 1983-08-01
ES516594A0 (es) 1983-11-16
ES8401079A1 (es) 1983-11-16
IL64506A0 (en) 1982-03-31
AU7846681A (en) 1982-06-17
KR830007683A (ko) 1983-11-04
ES8401080A1 (es) 1983-11-16
EP0054512A3 (de) 1983-08-03
EP0054512A2 (de) 1982-06-23
GR76967B (xx) 1984-09-04
HU185985B (en) 1985-04-28
PT74119B (de) 1983-12-19
GB2111043B (en) 1985-02-06
ES507907A0 (es) 1983-02-01
ES8401077A1 (es) 1983-11-16
JPH0314038B2 (xx) 1991-02-25
NO814232L (no) 1982-06-14
ES516593A0 (es) 1983-11-16
IE52008B1 (en) 1987-05-13
FI813946L (fi) 1982-06-13
ES8303424A1 (es) 1983-02-01
ES516591A0 (es) 1983-11-16
JPS57123190A (en) 1982-07-31
ZA818622B (en) 1982-10-27
DD208155A5 (de) 1984-03-28
DK550081A (da) 1982-06-13
GB2111043A (en) 1983-06-29
ES8401078A1 (es) 1983-11-16

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