IL59803A0 - Oxazoline and thiazoline derivatives,their preparation and pharmaceutical compositions containing them - Google Patents
Oxazoline and thiazoline derivatives,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL59803A0 IL59803A0 IL59803A IL5980380A IL59803A0 IL 59803 A0 IL59803 A0 IL 59803A0 IL 59803 A IL59803 A IL 59803A IL 5980380 A IL5980380 A IL 5980380A IL 59803 A0 IL59803 A0 IL 59803A0
- Authority
- IL
- Israel
- Prior art keywords
- alkyl
- halogen
- optionally substituted
- alkoxy
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/48—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Developing Agents For Electrophotography (AREA)
- Peptides Or Proteins (AREA)
- Luminescent Compositions (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7913864 | 1979-04-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
IL59803A0 true IL59803A0 (en) | 1980-06-30 |
Family
ID=10504680
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL59803A IL59803A0 (en) | 1979-04-20 | 1980-04-10 | Oxazoline and thiazoline derivatives,their preparation and pharmaceutical compositions containing them |
Country Status (14)
Country | Link |
---|---|
US (1) | US4409216A (xx) |
EP (1) | EP0018107B1 (xx) |
JP (1) | JPS55141474A (xx) |
AT (1) | ATE2075T1 (xx) |
AU (1) | AU5758880A (xx) |
DE (1) | DE3061396D1 (xx) |
DK (1) | DK167580A (xx) |
ES (2) | ES490675A0 (xx) |
FI (1) | FI801253A (xx) |
GR (1) | GR67301B (xx) |
IE (1) | IE49697B1 (xx) |
IL (1) | IL59803A0 (xx) |
NO (1) | NO801131L (xx) |
ZA (1) | ZA801970B (xx) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2075805B1 (es) * | 1993-12-30 | 1996-10-16 | Univ Murcia | Procedimiento para la obtencion de iminooxazolinas n-n'-sustituidas. |
DE102004008141A1 (de) | 2004-02-19 | 2005-09-01 | Abbott Gmbh & Co. Kg | Guanidinverbindungen und ihre Verwendung als Bindungspartner für 5-HT5-Rezeptoren |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3023103A (en) * | 1960-08-02 | 1962-02-27 | Gen Aniline & Film Corp | Antifoggants and stabilizers for photographic silver halide emulsions |
DE2205744A1 (de) | 1972-02-08 | 1973-08-09 | Thomae Gmbh Dr K | Neue durch einen guanidinylidenrest substituierte heterocyclen und verfahren zu ihrer herstellung |
CS225804B2 (cs) | 1976-03-19 | 1984-02-13 | Mcneilab Inc | Způsob výroby heterocyklických derivátů guanidinu |
NZ183570A (en) * | 1976-03-19 | 1979-06-08 | Mcneilab Inc | Heterocyclic guanidine derivatives, having anti-secretory and hypogliycaemic activity |
US4089965A (en) * | 1976-03-26 | 1978-05-16 | American Cyanamid Company | Thiazolylphenylguanidines as antirhinovirus agents |
CA1201119A (en) * | 1978-09-18 | 1986-02-25 | Mcneilab, Inc. | Diaza-cyclic derivatives of guanidine |
AU5263779A (en) * | 1978-11-29 | 1980-05-29 | Beecham Group Limited | Derivatives of thiazolidin-2-ylidene and oxazolidin-2-ylidene with hypoglycaemic acitivity |
-
1980
- 1980-03-27 AT AT80300949T patent/ATE2075T1/de active
- 1980-03-27 DE DE8080300949T patent/DE3061396D1/de not_active Expired
- 1980-03-27 EP EP80300949A patent/EP0018107B1/en not_active Expired
- 1980-04-02 ZA ZA00801970A patent/ZA801970B/xx unknown
- 1980-04-10 IL IL59803A patent/IL59803A0/xx unknown
- 1980-04-11 US US06/139,284 patent/US4409216A/en not_active Expired - Lifetime
- 1980-04-15 GR GR61687A patent/GR67301B/el unknown
- 1980-04-17 ES ES490675A patent/ES490675A0/es active Granted
- 1980-04-18 FI FI801253A patent/FI801253A/fi not_active Application Discontinuation
- 1980-04-18 DK DK167580A patent/DK167580A/da active IP Right Grant
- 1980-04-18 AU AU57588/80A patent/AU5758880A/en not_active Abandoned
- 1980-04-18 NO NO801131A patent/NO801131L/no unknown
- 1980-04-18 JP JP5155880A patent/JPS55141474A/ja active Pending
- 1980-04-18 IE IE787/80A patent/IE49697B1/en unknown
- 1980-12-09 ES ES497560A patent/ES8200668A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
DE3061396D1 (en) | 1983-01-27 |
ES497560A0 (es) | 1981-11-16 |
US4409216A (en) | 1983-10-11 |
ES8200668A1 (es) | 1981-11-16 |
GR67301B (xx) | 1981-06-29 |
IE49697B1 (en) | 1985-11-27 |
ATE2075T1 (de) | 1983-01-15 |
FI801253A (fi) | 1980-10-21 |
AU5758880A (en) | 1980-10-23 |
JPS55141474A (en) | 1980-11-05 |
IE800787L (en) | 1980-10-20 |
ZA801970B (en) | 1981-04-29 |
DK167580A (da) | 1980-10-21 |
ES8105306A1 (es) | 1981-05-16 |
ES490675A0 (es) | 1981-05-16 |
EP0018107A1 (en) | 1980-10-29 |
NO801131L (no) | 1980-10-21 |
EP0018107B1 (en) | 1982-12-22 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE9793T1 (de) | 5-oxo- und 5-thioxoproline, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen. | |
FI892787A0 (fi) | Analogiamenetelmä terapeuttisesti käyttökelpoisten 1-indolyylialkyyli-4-(substituoitu pyridinyyli)piperatsiinien valmistamiseksi | |
ES8600288A1 (es) | Un procedimiento para la preparacion de derivados de quinolina. | |
ES482134A1 (es) | Un procedimiento para preparar derivados de 1-(3-mercapto- 2-metilpropanoil)-prolil-aminoacido. | |
DK159148C (da) | Analogifremgangsmaade til fremstilling af tranexamsyrederivater | |
SE7714592L (sv) | Cyklopentan-1-aminer, forfarande for framstellning derav och medel innehallande dessa foreningar | |
FI853717L (fi) | 3-amino-2-benzoyl- akrylsyraderivat och foerfarande foer deras framstaellning. | |
AU560286B2 (en) | Imidazobenzodiazepines | |
ES8101589A1 (es) | Un procedimiento para la preparacion de nuevos compuestos iminicos heterociclicos. | |
DE3061396D1 (en) | Oxazoline and thiazoline derivatives, processes for their preparation and pharmaceutical compositions containing them | |
DE3174132D1 (en) | New ethenylimidazole derivatives, processes for their preparation and pharmaceutical compositions containing them; intermediates, useful in their preparation and a process for the preparation thereof | |
ES8305359A1 (es) | Un procedimiento para la preparacion de benzamitas sustituidas. | |
ES8200661A1 (es) | Un procedimiento para la preparacion de nuevos derivados de dihidropiridina | |
ATE52509T1 (de) | Thiazolidinderivate und verfahren zu ihrer herstellung. | |
ES8503655A1 (es) | Un procedimiento para preparar nuevas dihidropiridinas. | |
BE879727A (fr) | Derives de 1,2,4-triazole, leur preparation et leur utilisation | |
AU579416B2 (en) | 3-Amino-2,3-dihydro-1-benzoxepine-compounds and methods for their preparation and pharmaceutical preparations containing these compounds | |
ES483889A1 (es) | Un procedimiento para la preparacion de un derivado de aci- doclavulanico. | |
DE2963724D1 (en) | Clavulanic acid derivatives, their preparation and pharmaceutical compositions containing them | |
GB1042199A (en) | Certain substituted ª-alkyl and ª-cycloalkylamino-propionamides |