IL59803A0 - Oxazoline and thiazoline derivatives,their preparation and pharmaceutical compositions containing them - Google Patents
Oxazoline and thiazoline derivatives,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL59803A0 IL59803A0 IL59803A IL5980380A IL59803A0 IL 59803 A0 IL59803 A0 IL 59803A0 IL 59803 A IL59803 A IL 59803A IL 5980380 A IL5980380 A IL 5980380A IL 59803 A0 IL59803 A0 IL 59803A0
- Authority
- IL
- Israel
- Prior art keywords
- alkyl
- halogen
- optionally substituted
- alkoxy
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/48—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Developing Agents For Electrophotography (AREA)
- Peptides Or Proteins (AREA)
- Luminescent Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7913864 | 1979-04-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
IL59803A0 true IL59803A0 (en) | 1980-06-30 |
Family
ID=10504680
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL59803A IL59803A0 (en) | 1979-04-20 | 1980-04-10 | Oxazoline and thiazoline derivatives,their preparation and pharmaceutical compositions containing them |
Country Status (14)
Country | Link |
---|---|
US (1) | US4409216A (da) |
EP (1) | EP0018107B1 (da) |
JP (1) | JPS55141474A (da) |
AT (1) | ATE2075T1 (da) |
AU (1) | AU5758880A (da) |
DE (1) | DE3061396D1 (da) |
DK (1) | DK167580A (da) |
ES (2) | ES490675A0 (da) |
FI (1) | FI801253A (da) |
GR (1) | GR67301B (da) |
IE (1) | IE49697B1 (da) |
IL (1) | IL59803A0 (da) |
NO (1) | NO801131L (da) |
ZA (1) | ZA801970B (da) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2075805B1 (es) * | 1993-12-30 | 1996-10-16 | Univ Murcia | Procedimiento para la obtencion de iminooxazolinas n-n'-sustituidas. |
DE102004008141A1 (de) | 2004-02-19 | 2005-09-01 | Abbott Gmbh & Co. Kg | Guanidinverbindungen und ihre Verwendung als Bindungspartner für 5-HT5-Rezeptoren |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3023103A (en) * | 1960-08-02 | 1962-02-27 | Gen Aniline & Film Corp | Antifoggants and stabilizers for photographic silver halide emulsions |
DE2205744A1 (de) | 1972-02-08 | 1973-08-09 | Thomae Gmbh Dr K | Neue durch einen guanidinylidenrest substituierte heterocyclen und verfahren zu ihrer herstellung |
NZ183570A (en) * | 1976-03-19 | 1979-06-08 | Mcneilab Inc | Heterocyclic guanidine derivatives, having anti-secretory and hypogliycaemic activity |
CS225804B2 (cs) | 1976-03-19 | 1984-02-13 | Mcneilab Inc | Způsob výroby heterocyklických derivátů guanidinu |
US4089965A (en) * | 1976-03-26 | 1978-05-16 | American Cyanamid Company | Thiazolylphenylguanidines as antirhinovirus agents |
CA1201119A (en) * | 1978-09-18 | 1986-02-25 | Mcneilab, Inc. | Diaza-cyclic derivatives of guanidine |
AU5263779A (en) * | 1978-11-29 | 1980-05-29 | Beecham Group Limited | Derivatives of thiazolidin-2-ylidene and oxazolidin-2-ylidene with hypoglycaemic acitivity |
-
1980
- 1980-03-27 DE DE8080300949T patent/DE3061396D1/de not_active Expired
- 1980-03-27 EP EP80300949A patent/EP0018107B1/en not_active Expired
- 1980-03-27 AT AT80300949T patent/ATE2075T1/de active
- 1980-04-02 ZA ZA00801970A patent/ZA801970B/xx unknown
- 1980-04-10 IL IL59803A patent/IL59803A0/xx unknown
- 1980-04-11 US US06/139,284 patent/US4409216A/en not_active Expired - Lifetime
- 1980-04-15 GR GR61687A patent/GR67301B/el unknown
- 1980-04-17 ES ES490675A patent/ES490675A0/es active Granted
- 1980-04-18 IE IE787/80A patent/IE49697B1/en unknown
- 1980-04-18 FI FI801253A patent/FI801253A/fi not_active Application Discontinuation
- 1980-04-18 JP JP5155880A patent/JPS55141474A/ja active Pending
- 1980-04-18 NO NO801131A patent/NO801131L/no unknown
- 1980-04-18 AU AU57588/80A patent/AU5758880A/en not_active Abandoned
- 1980-04-18 DK DK167580A patent/DK167580A/da active IP Right Grant
- 1980-12-09 ES ES497560A patent/ES497560A0/es active Granted
Also Published As
Publication number | Publication date |
---|---|
ES8105306A1 (es) | 1981-05-16 |
AU5758880A (en) | 1980-10-23 |
NO801131L (no) | 1980-10-21 |
DE3061396D1 (en) | 1983-01-27 |
DK167580A (da) | 1980-10-21 |
GR67301B (da) | 1981-06-29 |
ATE2075T1 (de) | 1983-01-15 |
US4409216A (en) | 1983-10-11 |
ES8200668A1 (es) | 1981-11-16 |
IE49697B1 (en) | 1985-11-27 |
JPS55141474A (en) | 1980-11-05 |
IE800787L (en) | 1980-10-20 |
ZA801970B (en) | 1981-04-29 |
EP0018107A1 (en) | 1980-10-29 |
ES490675A0 (es) | 1981-05-16 |
FI801253A (fi) | 1980-10-21 |
EP0018107B1 (en) | 1982-12-22 |
ES497560A0 (es) | 1981-11-16 |
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