IL221007A - Pharmaceutical combinations for antiviral therapy - Google Patents

Pharmaceutical combinations for antiviral therapy Download PDF

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Publication number
IL221007A
IL221007A IL221007A IL22100712A IL221007A IL 221007 A IL221007 A IL 221007A IL 221007 A IL221007 A IL 221007A IL 22100712 A IL22100712 A IL 22100712A IL 221007 A IL221007 A IL 221007A
Authority
IL
Israel
Prior art keywords
antiviral therapy
pharmaceutical combinations
pharmaceutical
combinations
antiviral
Prior art date
Application number
IL221007A
Other languages
English (en)
Hebrew (he)
Other versions
IL221007A0 (en
Original Assignee
Viiv Healthcare Co
Glaxosmithkline Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44319704&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL221007(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Viiv Healthcare Co, Glaxosmithkline Llc filed Critical Viiv Healthcare Co
Publication of IL221007A0 publication Critical patent/IL221007A0/en
Publication of IL221007A publication Critical patent/IL221007A/en

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/536Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5365Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL221007A 2010-01-27 2012-07-18 Pharmaceutical combinations for antiviral therapy IL221007A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29858910P 2010-01-27 2010-01-27
PCT/US2011/022219 WO2011094150A1 (en) 2010-01-27 2011-01-24 Antiviral therapy

Publications (2)

Publication Number Publication Date
IL221007A0 IL221007A0 (en) 2012-09-24
IL221007A true IL221007A (en) 2016-06-30

Family

ID=44319704

Family Applications (5)

Application Number Title Priority Date Filing Date
IL221007A IL221007A (en) 2010-01-27 2012-07-18 Pharmaceutical combinations for antiviral therapy
IL245182A IL245182B (en) 2010-01-27 2016-04-18 A combination of compounds for antiviral treatment
IL257267A IL257267B (en) 2010-01-27 2018-01-31 A combination of compounds for antiviral treatment
IL267658A IL267658B (en) 2010-01-27 2019-06-26 A combination of compounds for antiviral treatment
IL281959A IL281959B (en) 2010-01-27 2021-04-01 Combining compounds for antiviral therapy

Family Applications After (4)

Application Number Title Priority Date Filing Date
IL245182A IL245182B (en) 2010-01-27 2016-04-18 A combination of compounds for antiviral treatment
IL257267A IL257267B (en) 2010-01-27 2018-01-31 A combination of compounds for antiviral treatment
IL267658A IL267658B (en) 2010-01-27 2019-06-26 A combination of compounds for antiviral treatment
IL281959A IL281959B (en) 2010-01-27 2021-04-01 Combining compounds for antiviral therapy

Country Status (45)

Country Link
US (12) US20120295898A1 (US07585860-20090908-C00112.png)
EP (6) EP3351249A1 (US07585860-20090908-C00112.png)
JP (8) JP2013518107A (US07585860-20090908-C00112.png)
KR (4) KR101883750B1 (US07585860-20090908-C00112.png)
CN (2) CN102791129B (US07585860-20090908-C00112.png)
AP (1) AP3551A (US07585860-20090908-C00112.png)
AU (1) AU2011209788C1 (US07585860-20090908-C00112.png)
BR (1) BR112012018670A2 (US07585860-20090908-C00112.png)
CA (4) CA3003988C (US07585860-20090908-C00112.png)
CL (1) CL2012002080A1 (US07585860-20090908-C00112.png)
CO (1) CO6602152A2 (US07585860-20090908-C00112.png)
CR (1) CR20120423A (US07585860-20090908-C00112.png)
CY (4) CY1116509T1 (US07585860-20090908-C00112.png)
DK (4) DK3127542T3 (US07585860-20090908-C00112.png)
DO (2) DOP2012000205A (US07585860-20090908-C00112.png)
EA (4) EA032868B1 (US07585860-20090908-C00112.png)
EC (1) ECSP12012106A (US07585860-20090908-C00112.png)
ES (4) ES2688925T3 (US07585860-20090908-C00112.png)
FI (2) FI3494972T3 (US07585860-20090908-C00112.png)
FR (1) FR18C1043I2 (US07585860-20090908-C00112.png)
HK (3) HK1209629A1 (US07585860-20090908-C00112.png)
HR (4) HRP20240168T1 (US07585860-20090908-C00112.png)
HU (4) HUE037812T2 (US07585860-20090908-C00112.png)
IL (5) IL221007A (US07585860-20090908-C00112.png)
LT (4) LT2932970T (US07585860-20090908-C00112.png)
LU (1) LUC00090I2 (US07585860-20090908-C00112.png)
MA (1) MA34002B1 (US07585860-20090908-C00112.png)
ME (2) ME03058B (US07585860-20090908-C00112.png)
MX (4) MX367937B (US07585860-20090908-C00112.png)
MY (1) MY188334A (US07585860-20090908-C00112.png)
NO (2) NO2932970T3 (US07585860-20090908-C00112.png)
NZ (4) NZ601319A (US07585860-20090908-C00112.png)
PE (2) PE20160180A1 (US07585860-20090908-C00112.png)
PH (2) PH12016500195B1 (US07585860-20090908-C00112.png)
PL (4) PL3494972T3 (US07585860-20090908-C00112.png)
PT (4) PT3494972T (US07585860-20090908-C00112.png)
RS (4) RS65183B1 (US07585860-20090908-C00112.png)
SG (3) SG10201509476RA (US07585860-20090908-C00112.png)
SI (4) SI2932970T1 (US07585860-20090908-C00112.png)
SM (1) SMT201500177B (US07585860-20090908-C00112.png)
TN (1) TN2012000376A1 (US07585860-20090908-C00112.png)
TR (1) TR201807704T4 (US07585860-20090908-C00112.png)
UA (1) UA105556C2 (US07585860-20090908-C00112.png)
WO (1) WO2011094150A1 (US07585860-20090908-C00112.png)
ZA (1) ZA201205586B (US07585860-20090908-C00112.png)

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