IL217952A - Derivatives of n1- acyl-5-fluoropyrimidinone - Google Patents

Derivatives of n1- acyl-5-fluoropyrimidinone

Info

Publication number
IL217952A
IL217952A IL217952A IL21795212A IL217952A IL 217952 A IL217952 A IL 217952A IL 217952 A IL217952 A IL 217952A IL 21795212 A IL21795212 A IL 21795212A IL 217952 A IL217952 A IL 217952A
Authority
IL
Israel
Prior art keywords
acyl
fluoropyrimidinone
derivatives
fluoropyrimidinone derivatives
Prior art date
Application number
IL217952A
Other languages
English (en)
Hebrew (he)
Other versions
IL217952A0 (en
Inventor
Bryan Kristy
A Boebel Timothy
Lorsbach Beth
p martin Timothy
john owen W
Pobanz Mark
Thornburgh Scott
D Webster Jeffery
Yao Chenglin
Original Assignee
Bryan Kristy
A Boebel Timothy
Lorsbach Beth
p martin Timothy
john owen W
Pobanz Mark
Thornburgh Scott
D Webster Jeffery
Yao Chenglin
Adama Makhteshim Ltd
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL217952(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bryan Kristy, A Boebel Timothy, Lorsbach Beth, p martin Timothy, john owen W, Pobanz Mark, Thornburgh Scott, D Webster Jeffery, Yao Chenglin, Adama Makhteshim Ltd, Dow Agrosciences Llc filed Critical Bryan Kristy
Publication of IL217952A0 publication Critical patent/IL217952A0/en
Publication of IL217952A publication Critical patent/IL217952A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL217952A 2009-08-07 2012-02-05 Derivatives of n1- acyl-5-fluoropyrimidinone IL217952A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (2)

Publication Number Publication Date
IL217952A0 IL217952A0 (en) 2012-03-29
IL217952A true IL217952A (en) 2017-11-30

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
IL217952A IL217952A (en) 2009-08-07 2012-02-05 Derivatives of n1- acyl-5-fluoropyrimidinone

Country Status (33)

Country Link
US (1) US8470839B2 (OSRAM)
EP (1) EP2519512B1 (OSRAM)
JP (1) JP5748754B2 (OSRAM)
KR (1) KR101792285B1 (OSRAM)
CN (1) CN102548981B (OSRAM)
AU (1) AU2010279402B2 (OSRAM)
BR (1) BR112012002810B1 (OSRAM)
CA (1) CA2768510C (OSRAM)
CL (1) CL2012000316A1 (OSRAM)
CO (1) CO6491117A2 (OSRAM)
CR (1) CR20120030A (OSRAM)
CY (1) CY1122115T1 (OSRAM)
DK (1) DK2519512T3 (OSRAM)
EA (1) EA023411B1 (OSRAM)
EC (1) ECSP12011653A (OSRAM)
ES (1) ES2728966T3 (OSRAM)
HN (1) HN2012000269A (OSRAM)
HR (1) HRP20190919T1 (OSRAM)
HU (1) HUE045290T2 (OSRAM)
IL (1) IL217952A (OSRAM)
IN (1) IN2012DN00539A (OSRAM)
LT (1) LT2519512T (OSRAM)
MX (1) MX2012001620A (OSRAM)
NI (1) NI201200022A (OSRAM)
NZ (1) NZ597570A (OSRAM)
PE (1) PE20120688A1 (OSRAM)
PL (1) PL2519512T3 (OSRAM)
PT (1) PT2519512T (OSRAM)
SI (1) SI2519512T1 (OSRAM)
TR (1) TR201908180T4 (OSRAM)
UA (1) UA106889C2 (OSRAM)
WO (1) WO2011017538A1 (OSRAM)
ZA (1) ZA201200819B (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体
EP2775842B1 (en) 2011-08-17 2017-10-04 Adama Makhteshim Ltd. 1-substituted-5-fluoro-3,6-dihydro-6-imino-2(1H)-pyrimidinone derivatives as fungicidal agents for use in plant protection
CN104884062B (zh) 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
AU2013370493B2 (en) 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
EP3689142A1 (en) * 2012-12-28 2020-08-05 Adama Makhteshim Ltd. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
NZ749557A (en) 2012-12-31 2020-01-31 Adama Makhteshim Ltd 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CN111362881A (zh) 2013-12-31 2020-07-03 阿达玛马克西姆股份有限公司 一种化合物及其制备方法
PT3096619T (pt) 2013-12-31 2025-09-11 Adama Makhteshim Ltd Misturas fungicidas sinérgicas para controlo de fungos em cereais
EP3197903B1 (en) 2014-09-26 2019-11-27 The Chemours Company FC, LLC Isocyanate derived organosilanes
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
BR112021008755A2 (pt) 2018-11-05 2021-08-10 Adama Makhteshim Ltd. misturas e composições contendo 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidina-2-ona, e métodos de uso.
AR120035A1 (es) 2019-09-23 2022-01-26 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (OSRAM) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
MX9800136A (es) * 1995-07-05 1998-03-29 Du Pont Pirimidinonas fungicidas.
JP2000506171A (ja) 1996-03-11 2000-05-23 ノバルティス アクチェンゲゼルシャフト 農薬としてのピリミジン−４−オン誘導体
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) * 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
WO2005095419A1 (ja) * 2004-04-01 2005-10-13 Takeda Pharmaceutial Company Limited チアゾロピリミジン誘導体
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
EP2562161A1 (en) 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
EP2647287A1 (en) 2008-08-01 2013-10-09 Dow AgroSciences LLC Use of 5-fluorocytosine and its derivatives as fungicides
HUE025349T2 (en) 2009-01-23 2016-02-29 Euro Celtique Sa Hydroxamic acid derivatives
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体

Also Published As

Publication number Publication date
IN2012DN00539A (OSRAM) 2015-06-12
BR112012002810A2 (pt) 2015-09-15
AU2010279402A1 (en) 2012-02-02
AU2010279402B2 (en) 2015-04-16
PT2519512T (pt) 2019-06-04
BR112012002810B1 (pt) 2018-12-11
HUE045290T2 (hu) 2019-12-30
NI201200022A (es) 2012-05-22
CN102548981A (zh) 2012-07-04
IL217952A0 (en) 2012-03-29
HN2012000269A (es) 2015-04-27
KR20120041786A (ko) 2012-05-02
CA2768510A1 (en) 2011-02-10
HRP20190919T1 (hr) 2019-09-20
EP2519512A1 (en) 2012-11-07
JP5748754B2 (ja) 2015-07-15
EP2519512B1 (en) 2019-03-20
CL2012000316A1 (es) 2014-06-27
US8470839B2 (en) 2013-06-25
ES2728966T3 (es) 2019-10-29
EA201270253A1 (ru) 2012-07-30
LT2519512T (lt) 2019-07-25
WO2011017538A1 (en) 2011-02-10
CY1122115T1 (el) 2020-11-25
DK2519512T3 (da) 2019-05-27
JP2013501723A (ja) 2013-01-17
NZ597570A (en) 2014-04-30
SI2519512T1 (sl) 2019-09-30
EP2519512A4 (en) 2013-01-16
EA023411B1 (ru) 2016-06-30
ECSP12011653A (es) 2012-03-30
PE20120688A1 (es) 2012-06-06
TR201908180T4 (tr) 2019-06-21
CA2768510C (en) 2018-05-15
CN102548981B (zh) 2015-05-13
CR20120030A (es) 2012-03-28
MX2012001620A (es) 2012-04-11
CO6491117A2 (es) 2012-07-31
HK1172894A1 (en) 2013-05-03
UA106889C2 (uk) 2014-10-27
PL2519512T3 (pl) 2019-09-30
KR101792285B1 (ko) 2017-10-31
US20110034490A1 (en) 2011-02-10
ZA201200819B (en) 2013-05-29

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