UA106889C2 - Похідні n1-ацил-5-фторпіримідинону - Google Patents

Похідні n1-ацил-5-фторпіримідинону

Info

Publication number
UA106889C2
UA106889C2 UAA201202731A UAA201202731A UA106889C2 UA 106889 C2 UA106889 C2 UA 106889C2 UA A201202731 A UAA201202731 A UA A201202731A UA A201202731 A UAA201202731 A UA A201202731A UA 106889 C2 UA106889 C2 UA 106889C2
Authority
UA
Ukraine
Prior art keywords
acyl
derivatives
florpyrimidinone
fluoropyrimidinones
fungicides
Prior art date
Application number
UAA201202731A
Other languages
English (en)
Ukrainian (uk)
Inventor
Тімоті Бебель
Крісті Брайан
Бет Лорсбах
Тімоті Мартін
В. Оуен
Марк Побанс
Скотт Торнберг
Джеффрі Вебстер
Ченьлінь Яо
Original Assignee
ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA106889(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі filed Critical ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі
Publication of UA106889C2 publication Critical patent/UA106889C2/uk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
UAA201202731A 2009-08-07 2010-05-08 Похідні n1-ацил-5-фторпіримідинону UA106889C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
UA106889C2 true UA106889C2 (uk) 2014-10-27

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201202731A UA106889C2 (uk) 2009-08-07 2010-05-08 Похідні n1-ацил-5-фторпіримідинону

Country Status (33)

Country Link
US (1) US8470839B2 (OSRAM)
EP (1) EP2519512B1 (OSRAM)
JP (1) JP5748754B2 (OSRAM)
KR (1) KR101792285B1 (OSRAM)
CN (1) CN102548981B (OSRAM)
AU (1) AU2010279402B2 (OSRAM)
BR (1) BR112012002810B1 (OSRAM)
CA (1) CA2768510C (OSRAM)
CL (1) CL2012000316A1 (OSRAM)
CO (1) CO6491117A2 (OSRAM)
CR (1) CR20120030A (OSRAM)
CY (1) CY1122115T1 (OSRAM)
DK (1) DK2519512T3 (OSRAM)
EA (1) EA023411B1 (OSRAM)
EC (1) ECSP12011653A (OSRAM)
ES (1) ES2728966T3 (OSRAM)
HN (1) HN2012000269A (OSRAM)
HR (1) HRP20190919T1 (OSRAM)
HU (1) HUE045290T2 (OSRAM)
IL (1) IL217952A (OSRAM)
IN (1) IN2012DN00539A (OSRAM)
LT (1) LT2519512T (OSRAM)
MX (1) MX2012001620A (OSRAM)
NI (1) NI201200022A (OSRAM)
NZ (1) NZ597570A (OSRAM)
PE (1) PE20120688A1 (OSRAM)
PL (1) PL2519512T3 (OSRAM)
PT (1) PT2519512T (OSRAM)
SI (1) SI2519512T1 (OSRAM)
TR (1) TR201908180T4 (OSRAM)
UA (1) UA106889C2 (OSRAM)
WO (1) WO2011017538A1 (OSRAM)
ZA (1) ZA201200819B (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA022289B1 (ru) * 2009-08-07 2015-12-30 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Производные n1-сульфонил-5-фторпиримидинона
KR102012992B1 (ko) * 2011-08-17 2019-08-21 아다마 마켓심 리미티드 5-플루오로-4-이미노-3-(치환된)-3,4-디히드로피리미딘-2-(1ｈ)-온 유도체
KR20150103095A (ko) * 2012-12-28 2015-09-09 다우 아그로사이언시즈 엘엘씨 1-(치환된-벤조일)-5-플루오로-4-이미노-3-메틸-3,4-디히드로피리미딘-2(1h)-온 유도체
CN104884062B (zh) 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
AU2013370493B2 (en) 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
US9642368B2 (en) * 2012-12-31 2017-05-09 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
CR20210172A (es) 2013-12-31 2021-05-11 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2 (1h)-ona y los procesos para su preparación
BR112016015158A2 (pt) 2013-12-31 2017-08-08 Adama Makhteshim Ltd Misturas fungicidas sinergísticas para controle de fungos em cereais
KR102430183B1 (ko) 2014-09-26 2022-08-08 더 케무어스 컴퍼니 에프씨, 엘엘씨 아이소시아네이트 유도된 유기실란
US11632954B2 (en) 2017-07-17 2023-04-25 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1 -tosyl-3,4-dihydropyrimidin-2-one
IL282939B2 (en) 2018-11-05 2024-10-01 Adama Makhteshim Ltd Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and methods of use thereof
UY38890A (es) 2019-09-23 2021-04-30 Adama Makhteshim Ltd Procedimiento para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

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Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (OSRAM) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
AU6478396A (en) * 1995-07-05 1997-02-05 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
ES2176697T3 (es) * 1996-03-11 2002-12-01 Syngenta Participations Ag Derivados pirimidin-4-ona como pesticidas.
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
WO2005095419A1 (ja) * 2004-04-01 2005-10-13 Takeda Pharmaceutial Company Limited チアゾロピリミジン誘導体
WO2008005303A2 (en) * 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
HUE026195T2 (en) 2008-01-22 2016-05-30 Dow Agrosciences Llc 4-Amino-5-fluoropyrimidine derivatives as fungicides
EP2647287A1 (en) 2008-08-01 2013-10-09 Dow AgroSciences LLC Use of 5-fluorocytosine and its derivatives as fungicides
ES2544803T3 (es) 2009-01-23 2015-09-04 Euro-Celtique S.A. Derivados del ácido hidroxámico
EA022289B1 (ru) * 2009-08-07 2015-12-30 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Производные n1-сульфонил-5-фторпиримидинона

Also Published As

Publication number Publication date
PL2519512T3 (pl) 2019-09-30
KR20120041786A (ko) 2012-05-02
KR101792285B1 (ko) 2017-10-31
IL217952A0 (en) 2012-03-29
SI2519512T1 (sl) 2019-09-30
MX2012001620A (es) 2012-04-11
CN102548981A (zh) 2012-07-04
IN2012DN00539A (OSRAM) 2015-06-12
EP2519512A1 (en) 2012-11-07
AU2010279402A1 (en) 2012-02-02
EA201270253A1 (ru) 2012-07-30
JP2013501723A (ja) 2013-01-17
ES2728966T3 (es) 2019-10-29
LT2519512T (lt) 2019-07-25
EA023411B1 (ru) 2016-06-30
IL217952A (en) 2017-11-30
US20110034490A1 (en) 2011-02-10
PE20120688A1 (es) 2012-06-06
CA2768510C (en) 2018-05-15
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
CL2012000316A1 (es) 2014-06-27
EP2519512A4 (en) 2013-01-16
PT2519512T (pt) 2019-06-04
JP5748754B2 (ja) 2015-07-15
US8470839B2 (en) 2013-06-25
HK1172894A1 (en) 2013-05-03
BR112012002810A2 (pt) 2015-09-15
CY1122115T1 (el) 2020-11-25
EP2519512B1 (en) 2019-03-20
CN102548981B (zh) 2015-05-13
DK2519512T3 (da) 2019-05-27
CA2768510A1 (en) 2011-02-10
CO6491117A2 (es) 2012-07-31
CR20120030A (es) 2012-03-28
NZ597570A (en) 2014-04-30
BR112012002810B1 (pt) 2018-12-11
WO2011017538A1 (en) 2011-02-10
HN2012000269A (es) 2015-04-27
AU2010279402B2 (en) 2015-04-16
HRP20190919T1 (hr) 2019-09-20
NI201200022A (es) 2012-05-22
TR201908180T4 (tr) 2019-06-21
ZA201200819B (en) 2013-05-29

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