IL160715A0 - Pharmaceutical compositions containing an a1 adenosine receptor antagonist - Google Patents

Pharmaceutical compositions containing an a1 adenosine receptor antagonist

Info

Publication number
IL160715A0
IL160715A0 IL16071502A IL16071502A IL160715A0 IL 160715 A0 IL160715 A0 IL 160715A0 IL 16071502 A IL16071502 A IL 16071502A IL 16071502 A IL16071502 A IL 16071502A IL 160715 A0 IL160715 A0 IL 160715A0
Authority
IL
Israel
Prior art keywords
pharmaceutical compositions
compositions containing
receptor antagonist
adenosine receptor
adenosine
Prior art date
Application number
IL16071502A
Other languages
English (en)
Original Assignee
Biogen Idec Inc
Musc Found For Res Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biogen Idec Inc, Musc Found For Res Dev filed Critical Biogen Idec Inc
Publication of IL160715A0 publication Critical patent/IL160715A0/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • A61K31/522Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL16071502A 2001-09-06 2002-09-06 Pharmaceutical compositions containing an a1 adenosine receptor antagonist IL160715A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31790801P 2001-09-06 2001-09-06
PCT/US2002/028580 WO2003022284A1 (fr) 2001-09-06 2002-09-06 Procedes de traitement des maladies pulmonaires

Publications (1)

Publication Number Publication Date
IL160715A0 true IL160715A0 (en) 2004-08-31

Family

ID=23235775

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16071502A IL160715A0 (en) 2001-09-06 2002-09-06 Pharmaceutical compositions containing an a1 adenosine receptor antagonist

Country Status (20)

Country Link
US (1) US20040259889A1 (fr)
EP (1) EP1429775A4 (fr)
JP (2) JP4388373B2 (fr)
KR (1) KR100979738B1 (fr)
CN (1) CN1564688A (fr)
AU (1) AU2002341618B2 (fr)
BR (1) BR0212329A (fr)
CA (1) CA2459533A1 (fr)
EA (1) EA014684B1 (fr)
GE (1) GEP20074132B (fr)
HU (1) HUP0401805A3 (fr)
IL (1) IL160715A0 (fr)
IS (1) IS7163A (fr)
MX (1) MXPA04002135A (fr)
NZ (1) NZ532083A (fr)
PL (1) PL368935A1 (fr)
UA (1) UA80258C2 (fr)
WO (1) WO2003022284A1 (fr)
YU (1) YU20104A (fr)
ZA (1) ZA200401765B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003105666A2 (fr) * 2002-06-12 2003-12-24 Biogen, Inc. Procede de traitement des lesions consecutives a la perfusion ischemique au moyen des antagonistes de recepteurs d'adenosine
US20040229901A1 (en) * 2003-02-24 2004-11-18 Lauren Otsuki Method of treatment of disease using an adenosine A1 receptor antagonist
RU2367442C2 (ru) * 2003-04-25 2009-09-20 Новокардия, Инк. Способ нормализации мочеиспускания при нарушении функции почек
CA2528385C (fr) * 2003-06-06 2011-03-15 Endacea, Inc. Antagonistes du recepteur d'adenosine a1
CN101420958A (zh) * 2006-04-06 2009-04-29 挪瓦卡尔迪阿公司 共投与腺苷a1受体拮抗剂和抗惊厥药
JP2009540003A (ja) * 2006-06-16 2009-11-19 ノヴァカーディア,インク. Aa1raの低頻度投与を含む腎機能の長期間にわたる改善
WO2007150026A2 (fr) 2006-06-23 2007-12-27 Incyte Corporation Dérivés de purinone en tant qu'agonistes de hm74a
BRPI0713619A2 (pt) 2006-06-23 2013-01-15 Incyte Corp composto ou prà-droga ou sal farmaceuticamente aceitÁvel do mesmo, composiÇço, e, uso do composto.
WO2008121882A1 (fr) * 2007-03-29 2008-10-09 Novacardia, Inc. Procédés améliorés d'administration d'antagonistes de récepteur d'adénosine a1
US20090197900A1 (en) * 2007-03-29 2009-08-06 Howard Dittrich Methods of treating heart failure and renal dysfunction in individuals with an adenosine a1 receptor antagonist
WO2009055021A1 (fr) * 2007-10-26 2009-04-30 New York University School Of Medicine Procédés et compositions pour le traitement de maladies hépatiques
US20090228097A1 (en) * 2008-03-07 2009-09-10 Abbott Cardiovascular Systems Inc. A1 Adenosine Receptor Antagonist-Coated Implantable Medical Device
WO2009152458A1 (fr) * 2008-06-13 2009-12-17 Biogen Idec Ma Inc. Formulation liquide appropriée pour une perfusion renfermant un antagoniste des récepteurs de l’adénosine destinée à traiter une insuffisance cardiaque ou une insuffisance rénale
CN103237548A (zh) * 2010-06-30 2013-08-07 吉利德科学股份有限公司 A2b腺苷受体拮抗剂用于治疗肺高血压的应用
US9598390B2 (en) * 2013-03-14 2017-03-21 Bristol-Myers Squibb Company Bicyclo[2.2.2]acid GPR120 modulators
CN111770926B (zh) 2018-01-04 2023-07-21 因佩蒂斯生物科学有限公司 三环化合物、组合物及其医药应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5208240A (en) * 1991-03-12 1993-05-04 Merrell Dow Pharmaceuticals Inc. 8-substituted purines as selective adenosine receptor agents
TW252044B (fr) * 1992-08-10 1995-07-21 Boehringer Ingelheim Kg
US5446046A (en) * 1993-10-28 1995-08-29 University Of Florida Research Foundation A1 adenosine receptor agonists and antagonists as diuretics
US5504090A (en) * 1994-03-30 1996-04-02 Trustees Of The University Of Pennsylvania Compositions and methods for the prevention and treatment of ischemia-reperfusion organ injury
SI0812844T1 (en) * 1996-06-07 2003-02-28 Hoechst Aktiengesellschaft Use of theophyllin derivatives for the treatment and prophylaxis fo shock conditions, novel xanthine compounds and processes for the production thereof
GB9723553D0 (en) * 1997-11-07 1998-01-07 Duff Gordon W Prediction of the risk of chronic obstructive airway disease
ZA9810766B (en) * 1997-11-28 1999-05-25 Mochida Pharm Co Ltd Novel compounds having cgmp-pde inhibitory activity
WO1999034803A1 (fr) * 1998-01-09 1999-07-15 The Trustees Of The University Of Pennsylvania Compositions et traitements convenant pour les lesions tissulaires liees a la reperfusion d'une ischemie ou dues a des endotoxines
EP0970696A1 (fr) * 1998-05-05 2000-01-12 Kyowa Hakko Kogyo Co., Ltd. Composition comprenant des diurétiques d'anse et des antagonists des recepteurs A1 de l'adenosine
SI1230243T1 (sl) * 1999-11-12 2009-08-31 Biogen Idec Inc Policikloalkilpurini kot antagonisti adenozinskega receptorja
PT1246623E (pt) * 1999-12-02 2006-12-29 Osi Pharm Inc Compostos específicos para o receptor de adenosina a1,a2a e a3 e as suas utilizações

Also Published As

Publication number Publication date
MXPA04002135A (es) 2005-03-07
KR20040040457A (ko) 2004-05-12
YU20104A (sh) 2006-08-17
US20040259889A1 (en) 2004-12-23
EA014684B1 (ru) 2010-12-30
EP1429775A1 (fr) 2004-06-23
HUP0401805A2 (hu) 2004-12-28
EA200400399A1 (ru) 2004-08-26
CN1564688A (zh) 2005-01-12
WO2003022284A1 (fr) 2003-03-20
UA80258C2 (en) 2007-09-10
EP1429775A4 (fr) 2007-04-11
KR100979738B1 (ko) 2010-09-09
BR0212329A (pt) 2004-09-21
ZA200401765B (en) 2005-04-05
HUP0401805A3 (en) 2007-05-02
AU2002341618B2 (en) 2008-06-26
JP2009209156A (ja) 2009-09-17
CA2459533A1 (fr) 2003-03-20
NZ532083A (en) 2005-10-28
JP2005501915A (ja) 2005-01-20
GEP20074132B (en) 2007-06-25
PL368935A1 (en) 2005-04-04
IS7163A (is) 2004-02-26
JP4388373B2 (ja) 2009-12-24

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