IL157413A0 - Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands - Google Patents

Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands

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Publication number
IL157413A0
IL157413A0 IL15741302A IL15741302A IL157413A0 IL 157413 A0 IL157413 A0 IL 157413A0 IL 15741302 A IL15741302 A IL 15741302A IL 15741302 A IL15741302 A IL 15741302A IL 157413 A0 IL157413 A0 IL 157413A0
Authority
IL
Israel
Prior art keywords
disorders
dopamine
compounds
substituted carbonyl
heterocyclic substituted
Prior art date
Application number
IL15741302A
Other languages
English (en)
Original Assignee
Aventis Pharmaceuticals Inc Av
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Publication date
Priority claimed from GBGB0117577.7A external-priority patent/GB0117577D0/en
Application filed by Aventis Pharmaceuticals Inc Av filed Critical Aventis Pharmaceuticals Inc Av
Publication of IL157413A0 publication Critical patent/IL157413A0/xx

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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D239/42—One nitrogen atom
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    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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IL15741302A 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands IL157413A0 (en)

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US26967201P 2001-02-16 2001-02-16
GBGB0117577.7A GB0117577D0 (en) 2001-02-16 2001-07-19 Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D receptor ligands
PCT/US2002/004713 WO2002066446A1 (en) 2001-02-16 2002-02-15 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands

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DE60235130D1 (de) 2010-03-04
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ATE313534T1 (de) 2006-01-15
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