IL154222A0 - Imidazolyl derivatives - Google Patents
Imidazolyl derivativesInfo
- Publication number
- IL154222A0 IL154222A0 IL15422201A IL15422201A IL154222A0 IL 154222 A0 IL154222 A0 IL 154222A0 IL 15422201 A IL15422201 A IL 15422201A IL 15422201 A IL15422201 A IL 15422201A IL 154222 A0 IL154222 A0 IL 154222A0
- Authority
- IL
- Israel
- Prior art keywords
- imidazolyl derivatives
- imidazolyl
- derivatives
- Prior art date
Links
- 125000002883 imidazolyl group Chemical group 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C—CHEMISTRY; METALLURGY
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- C—CHEMISTRY; METALLURGY
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- C—CHEMISTRY; METALLURGY
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- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
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Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Biomedical Technology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Oncology (AREA)
- Emergency Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Ophthalmology & Optometry (AREA)
- Pain & Pain Management (AREA)
- Transplantation (AREA)
- Communicable Diseases (AREA)
- Vascular Medicine (AREA)
- Dermatology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22258400P | 2000-08-01 | 2000-08-01 | |
PCT/US2001/023959 WO2002010140A2 (en) | 2000-08-01 | 2001-07-31 | Imidazolyl derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
IL154222A0 true IL154222A0 (en) | 2003-07-31 |
Family
ID=22832817
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL15422201A IL154222A0 (en) | 2000-08-01 | 2001-07-31 | Imidazolyl derivatives |
Country Status (15)
Country | Link |
---|---|
US (2) | US7566734B2 (no) |
EP (1) | EP1305294B1 (no) |
JP (1) | JP2004518613A (no) |
KR (1) | KR20030020960A (no) |
CN (1) | CN1444566A (no) |
AR (1) | AR035040A1 (no) |
AT (1) | ATE360620T1 (no) |
AU (2) | AU7909801A (no) |
CA (1) | CA2417204A1 (no) |
DE (1) | DE60128102T2 (no) |
ES (1) | ES2282275T3 (no) |
IL (1) | IL154222A0 (no) |
NO (1) | NO20030473L (no) |
NZ (1) | NZ523774A (no) |
WO (1) | WO2002010140A2 (no) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7291641B2 (en) * | 1999-10-11 | 2007-11-06 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Derivatives of heterocycles with 5 members, their preparation and their use as medicaments |
WO2003057214A1 (en) | 2001-12-28 | 2003-07-17 | Somatocor Pharmaceuticals, Inc. | Imidazolidin-2,4-dione derivatives as non-peptide somatostatin receptor ligands |
US7220862B2 (en) | 2002-06-05 | 2007-05-22 | Bristol-Myers Squibb Company | Calcitonin gene related peptide receptor antagonists |
US7842808B2 (en) | 2002-06-05 | 2010-11-30 | Bristol-Myers Squibb Company | Anti-migraine spirocycles |
WO2004032836A2 (en) * | 2002-10-07 | 2004-04-22 | Merck & Co., Inc. | Antidiabetic beta-amino heterocylcic dipeptidyl peptidase inhibitors |
CA2508947A1 (en) * | 2002-12-20 | 2004-07-15 | Merck & Co., Inc. | 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes |
WO2004071448A2 (en) * | 2003-02-12 | 2004-08-26 | Transtech Pharma Inc. | Substituted azole derivatives as inhibitors of protein tyrosine phosphatases |
AR046787A1 (es) * | 2003-12-05 | 2005-12-21 | Bristol Myers Squibb Co | Agentes antimigrana heterociclicos |
WO2005077373A2 (en) * | 2004-02-03 | 2005-08-25 | Astrazeneca Ab | Treatment of gastro-esophageal reflux disease (gerd) |
TW200533398A (en) | 2004-03-29 | 2005-10-16 | Bristol Myers Squibb Co | Novel therapeutic agents for the treatment of migraine |
US7453002B2 (en) | 2004-06-15 | 2008-11-18 | Bristol-Myers Squibb Company | Five-membered heterocycles useful as serine protease inhibitors |
RU2427572C2 (ru) | 2004-06-18 | 2011-08-27 | Чирон Корпорейшн | N-(1-(1-бензил-4-фенил-1н-имидазол-2-ил)-2,2-диметилпропил)бензамидные производные и родственные соединения в качестве ингибиторов кинезинового белка веретена (ksp) для лечения рака |
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2001
- 2001-07-31 KR KR10-2003-7001501A patent/KR20030020960A/ko not_active Application Discontinuation
- 2001-07-31 US US10/333,556 patent/US7566734B2/en not_active Expired - Fee Related
- 2001-07-31 WO PCT/US2001/023959 patent/WO2002010140A2/en active IP Right Grant
- 2001-07-31 IL IL15422201A patent/IL154222A0/xx unknown
- 2001-07-31 JP JP2002516272A patent/JP2004518613A/ja active Pending
- 2001-07-31 AR ARP010103657A patent/AR035040A1/es not_active Application Discontinuation
- 2001-07-31 EP EP01957342A patent/EP1305294B1/en not_active Expired - Lifetime
- 2001-07-31 ES ES01957342T patent/ES2282275T3/es not_active Expired - Lifetime
- 2001-07-31 CA CA002417204A patent/CA2417204A1/en not_active Abandoned
- 2001-07-31 CN CN01813618A patent/CN1444566A/zh active Pending
- 2001-07-31 NZ NZ523774A patent/NZ523774A/en unknown
- 2001-07-31 AT AT01957342T patent/ATE360620T1/de not_active IP Right Cessation
- 2001-07-31 AU AU7909801A patent/AU7909801A/xx active Pending
- 2001-07-31 AU AU2001279098A patent/AU2001279098B2/en not_active Expired - Fee Related
- 2001-07-31 DE DE60128102T patent/DE60128102T2/de not_active Expired - Fee Related
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2003
- 2003-01-30 NO NO20030473A patent/NO20030473L/no unknown
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2007
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AU2001279098B2 (en) | 2005-04-14 |
ATE360620T1 (de) | 2007-05-15 |
AR035040A1 (es) | 2004-04-14 |
NO20030473D0 (no) | 2003-01-30 |
NZ523774A (en) | 2004-09-24 |
NO20030473L (no) | 2003-01-30 |
CN1444566A (zh) | 2003-09-24 |
WO2002010140A3 (en) | 2002-08-08 |
DE60128102D1 (en) | 2007-06-06 |
KR20030020960A (ko) | 2003-03-10 |
WO2002010140A2 (en) | 2002-02-07 |
CA2417204A1 (en) | 2002-02-07 |
AU7909801A (en) | 2002-02-13 |
US7566734B2 (en) | 2009-07-28 |
JP2004518613A (ja) | 2004-06-24 |
EP1305294A2 (en) | 2003-05-02 |
US7638546B1 (en) | 2009-12-29 |
ES2282275T3 (es) | 2007-10-16 |
EP1305294B1 (en) | 2007-04-25 |
DE60128102T2 (de) | 2008-01-03 |
US20070032653A1 (en) | 2007-02-08 |
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