IL148807A0 - Tetrahydrothiopyran derivatives and pharmaceutical compositions containing the same - Google Patents
Tetrahydrothiopyran derivatives and pharmaceutical compositions containing the sameInfo
- Publication number
- IL148807A0 IL148807A0 IL14880700A IL14880700A IL148807A0 IL 148807 A0 IL148807 A0 IL 148807A0 IL 14880700 A IL14880700 A IL 14880700A IL 14880700 A IL14880700 A IL 14880700A IL 148807 A0 IL148807 A0 IL 148807A0
- Authority
- IL
- Israel
- Prior art keywords
- tetrahydrothiopyran
- derivatives
- same
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/502—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with carbocyclic ring systems, e.g. cinnoline, phthalazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP99121243 | 1999-10-25 | ||
| US20395000P | 2000-05-12 | 2000-05-12 | |
| PCT/EP2000/010445 WO2001030777A1 (en) | 1999-10-25 | 2000-10-24 | Tetrahydrothiopy ranphthalazinone derivatives as pde4 inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL148807A0 true IL148807A0 (en) | 2002-09-12 |
Family
ID=26153155
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL14880700A IL148807A0 (en) | 1999-10-25 | 2000-10-24 | Tetrahydrothiopyran derivatives and pharmaceutical compositions containing the same |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US6544993B1 (es) |
| EP (1) | EP1244654A1 (es) |
| JP (1) | JP2003512466A (es) |
| KR (1) | KR20020043238A (es) |
| CN (1) | CN1146562C (es) |
| AU (1) | AU781137B2 (es) |
| BR (1) | BR0014990A (es) |
| CA (1) | CA2388119A1 (es) |
| CZ (1) | CZ20021457A3 (es) |
| EA (1) | EA005856B1 (es) |
| HK (1) | HK1047276A1 (es) |
| HR (1) | HRP20020350A2 (es) |
| HU (1) | HUP0203487A2 (es) |
| IL (1) | IL148807A0 (es) |
| MX (1) | MXPA02003581A (es) |
| NO (1) | NO20021959L (es) |
| PL (1) | PL354979A1 (es) |
| SK (1) | SK7232002A3 (es) |
| TR (1) | TR200201128T2 (es) |
| WO (1) | WO2001030777A1 (es) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1146562C (zh) * | 1999-10-25 | 2004-04-21 | 奥坦纳医药公司 | 作为pde4抑制剂的四氢噻喃2,3-二氮杂萘酮类衍生物 |
| KR20030074817A (ko) * | 2001-02-15 | 2003-09-19 | 알타나 파마 아게 | Ｐｄｅ4 억제제로서의 프탈라지논-피페리디노-유도체 |
| JP4021329B2 (ja) | 2001-04-25 | 2007-12-12 | ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング | ピペラジノ誘導体およびｐｄｅ４阻害剤としてのその使用 |
| CN1503792A (zh) * | 2001-04-25 | 2004-06-09 | ��̹��ҽҩ��˾ | 新的酞嗪酮 |
| TWI347845B (en) * | 2002-03-06 | 2011-09-01 | Nycomed Gmbh | Pharmaceutical compositions,combinations,and kits for the treatment of respiratory diseases and use of the same |
| US20060167001A1 (en) * | 2002-08-10 | 2006-07-27 | Sterk Jan G | Pyridazinone-derivatives as pde4 inhibitors |
| AU2003255376A1 (en) * | 2002-08-10 | 2004-03-11 | Altana Pharma Ag | Piperidine-derivatives as pde4 inhibitors |
| CA2494643A1 (en) * | 2002-08-10 | 2004-03-04 | Altana Pharma Ag | Piperidine-n-oxide-derivatives |
| JP4555684B2 (ja) * | 2002-08-10 | 2010-10-06 | ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｐｄｅ４阻害剤としての、ピロリジンジオンにより置換されたピペリジン−フタラゾン |
| PL378247A1 (pl) * | 2003-01-14 | 2006-03-20 | Altana Pharma Ag | Inhibitory PDE4 w terapii nowotworów komórek limfoidalnych |
| EP1716123A1 (en) * | 2004-02-04 | 2006-11-02 | Altana Pharma AG | Pyridazinone derivatives and their use as pde4 inhibitors |
| ATE390419T1 (de) | 2004-02-04 | 2008-04-15 | Nycomed Gmbh | 2-(piperidin-4-yl)-4,5-dihydro-2h-pyridazin-3-o - derivate als pde4-inhibitoren |
| WO2005085225A1 (en) * | 2004-03-03 | 2005-09-15 | Altana Pharma Ag | Novel hydroxy-6-heteroarylphenanthridines and their use as pde4 inhibitors |
| WO2012080735A1 (en) * | 2010-12-16 | 2012-06-21 | Convergence Pharmaceuticals Limited | Ask1 inhibiting pyrrolopyrimidine derivatives |
| WO2013106547A1 (en) | 2012-01-10 | 2013-07-18 | President And Fellows Of Harvard College | Beta-cell replication promoting compounds and methods of their use |
| CA2906008C (en) | 2013-03-13 | 2019-07-09 | Flatley Discovery Lab, Llc | Pyridazinone compounds and methods for the treatment of cystic fibrosis |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9204808D0 (en) * | 1992-03-04 | 1992-04-15 | Rhone Poulenc Rorer Ltd | Novel compositions of matter |
| RU95113454A (ru) | 1992-12-02 | 1997-06-10 | Пфайзер Инк. (US) | Катехольные диэфиры как селективные ингибиторы фдэiv, фармацевтическая композиция, способы лечения |
| DE19533975A1 (de) | 1995-09-14 | 1997-03-20 | Merck Patent Gmbh | Arylalkyl-diazinone |
| SK283270B6 (sk) * | 1997-01-15 | 2003-04-01 | Altana Pharma Ag | Ftalazinóny, farmaceutické prostriedky s ich obsahom a ich použitie |
| WO1999031071A1 (en) | 1997-12-15 | 1999-06-24 | Byk Gulden Lomberg Chemische Fabrik Gmbh | New phthalazinones |
| EP1042319B1 (en) | 1997-12-15 | 2004-02-04 | ALTANA Pharma AG | Dihydrobenzofurans |
| EP1070056B1 (en) | 1998-03-14 | 2004-06-30 | ALTANA Pharma AG | Phthalazinone pde iii/iv inhibitors |
| CN1146562C (zh) * | 1999-10-25 | 2004-04-21 | 奥坦纳医药公司 | 作为pde4抑制剂的四氢噻喃2,3-二氮杂萘酮类衍生物 |
-
2000
- 2000-10-24 CN CNB008146977A patent/CN1146562C/zh not_active Expired - Fee Related
- 2000-10-24 TR TR2002/01128T patent/TR200201128T2/xx unknown
- 2000-10-24 CA CA002388119A patent/CA2388119A1/en not_active Abandoned
- 2000-10-24 PL PL00354979A patent/PL354979A1/xx not_active Application Discontinuation
- 2000-10-24 JP JP2001533131A patent/JP2003512466A/ja active Pending
- 2000-10-24 EP EP00977429A patent/EP1244654A1/en not_active Withdrawn
- 2000-10-24 WO PCT/EP2000/010445 patent/WO2001030777A1/en not_active Application Discontinuation
- 2000-10-24 AU AU15151/01A patent/AU781137B2/en not_active Ceased
- 2000-10-24 IL IL14880700A patent/IL148807A0/xx unknown
- 2000-10-24 BR BR0014990-0A patent/BR0014990A/pt not_active IP Right Cessation
- 2000-10-24 SK SK723-2002A patent/SK7232002A3/sk unknown
- 2000-10-24 KR KR1020027005200A patent/KR20020043238A/ko not_active Application Discontinuation
- 2000-10-24 CZ CZ20021457A patent/CZ20021457A3/cs unknown
- 2000-10-24 US US10/110,397 patent/US6544993B1/en not_active Expired - Fee Related
- 2000-10-24 EA EA200200381A patent/EA005856B1/ru not_active IP Right Cessation
- 2000-10-24 HU HU0203487A patent/HUP0203487A2/hu unknown
- 2000-10-24 MX MXPA02003581A patent/MXPA02003581A/es unknown
-
2002
- 2002-04-22 HR HR20020350A patent/HRP20020350A2/hr not_active Application Discontinuation
- 2002-04-25 NO NO20021959A patent/NO20021959L/no not_active Application Discontinuation
- 2002-12-04 HK HK02108822.5A patent/HK1047276A1/zh unknown
-
2003
- 2003-02-25 US US10/372,243 patent/US6846821B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CN1382137A (zh) | 2002-11-27 |
| MXPA02003581A (es) | 2002-10-23 |
| EP1244654A1 (en) | 2002-10-02 |
| WO2001030777A1 (en) | 2001-05-03 |
| US20030166655A1 (en) | 2003-09-04 |
| HUP0203487A2 (hu) | 2003-02-28 |
| JP2003512466A (ja) | 2003-04-02 |
| CN1146562C (zh) | 2004-04-21 |
| KR20020043238A (ko) | 2002-06-08 |
| NO20021959L (no) | 2002-05-29 |
| SK7232002A3 (en) | 2002-09-10 |
| AU1515101A (en) | 2001-05-08 |
| NO20021959D0 (no) | 2002-04-25 |
| CZ20021457A3 (cs) | 2002-07-17 |
| TR200201128T2 (tr) | 2002-08-21 |
| CA2388119A1 (en) | 2001-05-03 |
| HK1047276A1 (zh) | 2003-02-14 |
| HRP20020350A2 (en) | 2004-02-29 |
| AU781137B2 (en) | 2005-05-05 |
| US6846821B2 (en) | 2005-01-25 |
| BR0014990A (pt) | 2002-06-18 |
| US6544993B1 (en) | 2003-04-08 |
| PL354979A1 (en) | 2004-03-22 |
| EA005856B1 (ru) | 2005-06-30 |
| EA200200381A1 (ru) | 2002-10-31 |
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