IL144611A0 - Indole derivatives and their use as mcp-1 antagonists - Google Patents

Indole derivatives and their use as mcp-1 antagonists

Info

Publication number
IL144611A0
IL144611A0 IL14461100A IL14461100A IL144611A0 IL 144611 A0 IL144611 A0 IL 144611A0 IL 14461100 A IL14461100 A IL 14461100A IL 14461100 A IL14461100 A IL 14461100A IL 144611 A0 IL144611 A0 IL 144611A0
Authority
IL
Israel
Prior art keywords
mcp
antagonists
indole derivatives
indole
derivatives
Prior art date
Application number
IL14461100A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of IL144611A0 publication Critical patent/IL144611A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
IL14461100A 1999-02-05 2000-01-31 Indole derivatives and their use as mcp-1 antagonists IL144611A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9902461.4A GB9902461D0 (en) 1999-02-05 1999-02-05 Chemical compounds
PCT/GB2000/000265 WO2000046196A1 (en) 1999-02-05 2000-01-31 Indole derivatives and their use as mcp-1 antagonists

Publications (1)

Publication Number Publication Date
IL144611A0 true IL144611A0 (en) 2002-05-23

Family

ID=10847084

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14461100A IL144611A0 (en) 1999-02-05 2000-01-31 Indole derivatives and their use as mcp-1 antagonists

Country Status (27)

Country Link
US (1) US6737435B1 (no)
EP (1) EP1150952B1 (no)
JP (1) JP2002536359A (no)
KR (1) KR20010094755A (no)
CN (1) CN1339025A (no)
AR (1) AR022461A1 (no)
AT (1) ATE280757T1 (no)
AU (1) AU770856B2 (no)
BR (1) BR0007984A (no)
CA (1) CA2356898A1 (no)
CZ (1) CZ20012807A3 (no)
DE (1) DE60015296T2 (no)
EE (1) EE200100403A (no)
GB (1) GB9902461D0 (no)
HU (1) HUP0105079A3 (no)
ID (1) ID30401A (no)
IL (1) IL144611A0 (no)
IS (1) IS5980A (no)
MY (1) MY133209A (no)
NO (1) NO20013809L (no)
NZ (1) NZ512680A (no)
PL (1) PL350184A1 (no)
RU (1) RU2235090C2 (no)
SK (1) SK11152001A3 (no)
TR (1) TR200102233T2 (no)
WO (1) WO2000046196A1 (no)
ZA (1) ZA200105311B (no)

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GB0000626D0 (en) * 2000-01-13 2000-03-01 Zeneca Ltd Chemical compounds
GB0000625D0 (en) * 2000-01-13 2000-03-01 Zeneca Ltd Chemical compounds
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JP2005506949A (ja) 2000-12-20 2005-03-10 ブリストル−マイヤーズ・スクイブ・ファーマ・カンパニー ケモカイン受容体の調節剤としてのジアミン
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ES2812698T3 (es) 2017-09-29 2021-03-18 Probiodrug Ag Inhibidores de glutaminil ciclasa
KR20210095165A (ko) 2018-11-19 2021-07-30 프로제너티, 인크. 바이오의약품으로 질환을 치료하기 위한 방법 및 디바이스
CN115666704A (zh) 2019-12-13 2023-01-31 比奥拉治疗股份有限公司 用于将治疗剂递送至胃肠道的可摄取装置
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Also Published As

Publication number Publication date
WO2000046196A1 (en) 2000-08-10
ID30401A (id) 2001-11-29
DE60015296T2 (de) 2006-02-02
ZA200105311B (en) 2002-09-27
HUP0105079A3 (en) 2002-11-28
NO20013809L (no) 2001-10-02
SK11152001A3 (sk) 2001-12-03
NO20013809D0 (no) 2001-08-03
US6737435B1 (en) 2004-05-18
BR0007984A (pt) 2001-11-06
PL350184A1 (en) 2002-11-18
CZ20012807A3 (cs) 2001-10-17
CA2356898A1 (en) 2000-08-10
AU2121300A (en) 2000-08-25
EP1150952A1 (en) 2001-11-07
EP1150952B1 (en) 2004-10-27
KR20010094755A (ko) 2001-11-01
DE60015296D1 (de) 2004-12-02
RU2001124567A (ru) 2004-01-10
IS5980A (is) 2001-06-26
EE200100403A (et) 2002-10-15
AU770856B2 (en) 2004-03-04
NZ512680A (en) 2003-11-28
JP2002536359A (ja) 2002-10-29
RU2235090C2 (ru) 2004-08-27
TR200102233T2 (tr) 2001-12-21
ATE280757T1 (de) 2004-11-15
CN1339025A (zh) 2002-03-06
HUP0105079A2 (hu) 2002-04-29
GB9902461D0 (en) 1999-03-24
MY133209A (en) 2007-10-31
AR022461A1 (es) 2002-09-04

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