IL144044A0 - Macrolides with anti-inflammatory activity - Google Patents

Macrolides with anti-inflammatory activity

Info

Publication number
IL144044A0
IL144044A0 IL14404400A IL14404400A IL144044A0 IL 144044 A0 IL144044 A0 IL 144044A0 IL 14404400 A IL14404400 A IL 14404400A IL 14404400 A IL14404400 A IL 14404400A IL 144044 A0 IL144044 A0 IL 144044A0
Authority
IL
Israel
Prior art keywords
macrolides
inflammatory activity
oxyimino
endowed
dimethylamino
Prior art date
Application number
IL14404400A
Other languages
English (en)
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of IL144044A0 publication Critical patent/IL144044A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL14404400A 1999-01-15 2000-01-12 Macrolides with anti-inflammatory activity IL144044A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT1999MI000061A IT1306205B1 (it) 1999-01-15 1999-01-15 Macrolidi ad attivita' antiinfiammatoria.
PCT/EP2000/000163 WO2000042055A2 (en) 1999-01-15 2000-01-12 Macrolides with anti-inflammatory activity

Publications (1)

Publication Number Publication Date
IL144044A0 true IL144044A0 (en) 2002-04-21

Family

ID=11381492

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14404400A IL144044A0 (en) 1999-01-15 2000-01-12 Macrolides with anti-inflammatory activity
IL144044A IL144044A (en) 1999-01-15 2001-06-28 Anti- inflammatory 3' - de (dimethylamino) - erythromycin a-9-oxime derivatives and pharmaceutical compositions containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL144044A IL144044A (en) 1999-01-15 2001-06-28 Anti- inflammatory 3' - de (dimethylamino) - erythromycin a-9-oxime derivatives and pharmaceutical compositions containing them

Country Status (19)

Country Link
US (1) US6455576B1 (https=)
EP (1) EP1144427B1 (https=)
JP (1) JP4568433B2 (https=)
CN (1) CN1151165C (https=)
AT (1) ATE308552T1 (https=)
AU (1) AU769006B2 (https=)
BR (1) BR0007514A (https=)
CA (1) CA2368400C (https=)
DE (1) DE60023647T2 (https=)
ES (1) ES2251966T3 (https=)
HU (1) HU229228B1 (https=)
IL (2) IL144044A0 (https=)
IT (1) IT1306205B1 (https=)
MX (1) MXPA01007164A (https=)
NO (1) NO318982B1 (https=)
RU (1) RU2243230C2 (https=)
SK (1) SK286772B6 (https=)
WO (1) WO2000042055A2 (https=)
ZA (1) ZA200105748B (https=)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20010018A2 (en) 2001-01-09 2002-12-31 Pliva D D Novel anti-inflammatory compounds
AU2003264917A1 (en) 2002-07-08 2004-01-23 Pliva - Istrazivacki Institut D.O.O. Hybrid molecules of macrolides with steroid/non-steroid anti-inflammatory, antineoplastic and antiviral active molecules
RS20050008A (sr) 2002-07-08 2007-06-04 Pliva-Istraživački Institut D.O.O., Nova jedinjenja,kompozicije i metode za lečenje inflamatornih oboljenja i stanja
EP1521763A2 (en) * 2002-07-08 2005-04-13 Pliva - Istrazivacki Institut d.o.o. Novel nonsteroidal anti-inflammatory substances, compositions and methods for their use
ITMI20021726A1 (it) 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
TW200420573A (en) 2002-09-26 2004-10-16 Rib X Pharmaceuticals Inc Bifunctional heterocyclic compounds and methods of making and using same
ITMI20022292A1 (it) * 2002-10-29 2004-04-30 Zambon Spa 9a-azalidi ad attivita' antiinfiammatoria.
BRPI0410638A (pt) * 2003-04-17 2006-06-13 Sandoz Ag derivados de azitromicina
HRP20030324A2 (en) 2003-04-24 2005-02-28 Pliva-Istra�iva�ki institut d.o.o. Compounds of antiinflammatory effect
ITMI20040124A1 (it) * 2004-01-29 2004-04-29 Zambon Spa Macrolidi ad attivita' antiinfiammatoria
WO2006130128A2 (en) * 2004-02-18 2006-12-07 Chiron Corporation Methods of identifying anti-inflammatory macrolides
EP1723159B1 (en) 2004-02-27 2019-06-12 Melinta Therapeutics, Inc. Macrocyclic compounds and methods of making and using the same
WO2006035301A2 (en) * 2004-09-27 2006-04-06 Ranbaxy Laboratories Limited Erythromycin a derivatives as antibacterial agents
ES2337915T3 (es) 2004-10-27 2010-04-30 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. Conjugados con adtividad antiinflamatoria.
US20080249034A1 (en) * 2005-03-21 2008-10-09 Zambon S.P.A. Use of Macrolides for Treating Intestinal Inflammation
US7582611B2 (en) * 2005-05-24 2009-09-01 Pfizer Inc. Motilide compounds
US20110178287A1 (en) 2010-01-19 2011-07-21 Cerulean Pharma Inc. Cyclodextrin-based polymers for therapeutic delivery
RU2455309C2 (ru) * 2010-07-20 2012-07-10 Открытое Акционерное Общество "Татхимфармпрепараты" Способ получения аморфной формы рокситромицина
GB201608236D0 (en) 2016-05-11 2016-06-22 Fidelta D O O Seco macrolide compounds
TWI830987B (zh) 2020-03-12 2024-02-01 美商碩騰服務公司 免疫調節脲氮雜內酯
WO2021195126A1 (en) 2020-03-24 2021-09-30 Burnet Michael W Anti-infective and anti-viral compounds and compositions

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3928387A (en) * 1974-02-04 1975-12-23 Hoffmann La Roche Antibiotic 1745A/X and methods for the production thereof
IT1189285B (it) * 1982-05-28 1988-02-04 Nuovo Consor Sanitar Nazionale Sali dell'antibiotico eritromicina e del suo estere propionico con acidi ad attivita' terapeutica coadiuvante
EP0254534A3 (en) * 1986-07-24 1991-04-17 William S. Robinson Erythromycin derivatives and compositions and use for inhibiting virus replication and disease
FR2697524B1 (fr) * 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
IT1276901B1 (it) * 1994-12-13 1997-11-03 Zambon Spa Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica
KR19980701895A (ko) * 1995-03-08 1998-06-25 이라우치지마 가즈다카 면역관련병 처치제 및 그의 탐색 방법

Also Published As

Publication number Publication date
CN1151165C (zh) 2004-05-26
AU2663600A (en) 2000-08-01
ATE308552T1 (de) 2005-11-15
DE60023647T2 (de) 2006-08-10
ES2251966T3 (es) 2006-05-16
NO20013517D0 (no) 2001-07-16
JP4568433B2 (ja) 2010-10-27
HUP0105105A2 (hu) 2002-04-29
EP1144427B1 (en) 2005-11-02
CA2368400A1 (en) 2000-07-20
BR0007514A (pt) 2001-11-20
IL144044A (en) 2006-12-31
MXPA01007164A (es) 2002-03-27
IT1306205B1 (it) 2001-05-30
RU2243230C2 (ru) 2004-12-27
SK286772B6 (sk) 2009-05-07
HU229228B1 (en) 2013-09-30
ZA200105748B (en) 2002-10-14
EP1144427A2 (en) 2001-10-17
HUP0105105A3 (en) 2003-05-28
JP2002534531A (ja) 2002-10-15
DE60023647D1 (de) 2005-12-08
US6455576B1 (en) 2002-09-24
CN1336932A (zh) 2002-02-20
ITMI990061A1 (it) 2000-07-15
SK9812001A3 (en) 2002-01-07
WO2000042055A2 (en) 2000-07-20
EP1144427A3 (en) 2002-08-28
WO2000042055A3 (en) 2001-09-07
NO20013517L (no) 2001-07-16
NO318982B1 (no) 2005-05-30
AU769006B2 (en) 2004-01-15
CA2368400C (en) 2007-06-05

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Legal Events

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