IL140586A - Phenyl ester derivatives of a-amino acid and pharmaceuticals containing them - Google Patents

Phenyl ester derivatives of a-amino acid and pharmaceuticals containing them

Info

Publication number
IL140586A
IL140586A IL14058699A IL14058699A IL140586A IL 140586 A IL140586 A IL 140586A IL 14058699 A IL14058699 A IL 14058699A IL 14058699 A IL14058699 A IL 14058699A IL 140586 A IL140586 A IL 140586A
Authority
IL
Israel
Prior art keywords
acid
amino acid
alkoxy
alkyl
acid phenyl
Prior art date
Application number
IL14058699A
Other languages
English (en)
Hebrew (he)
Other versions
IL140586A0 (en
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of IL140586A0 publication Critical patent/IL140586A0/xx
Publication of IL140586A publication Critical patent/IL140586A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/38Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/06Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
    • C07C229/10Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
    • C07C229/12Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of acyclic carbon skeletons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/06Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
    • C07C229/10Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
    • C07C229/16Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of hydrocarbon radicals substituted by amino or carboxyl groups, e.g. ethylenediamine-tetra-acetic acid, iminodiacetic acids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL14058699A 1998-07-22 1999-07-16 Phenyl ester derivatives of a-amino acid and pharmaceuticals containing them IL140586A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP98305837 1998-07-22
PCT/EP1999/005051 WO2000005196A1 (en) 1998-07-22 1999-07-16 α-AMINO ACID PHENYL ESTER DERIVATIVES

Publications (2)

Publication Number Publication Date
IL140586A0 IL140586A0 (en) 2002-02-10
IL140586A true IL140586A (en) 2004-06-01

Family

ID=8234960

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14058699A IL140586A (en) 1998-07-22 1999-07-16 Phenyl ester derivatives of a-amino acid and pharmaceuticals containing them

Country Status (27)

Country Link
US (1) US6451854B1 (no)
EP (1) EP1098871B1 (no)
JP (1) JP2002521358A (no)
KR (1) KR100599142B1 (no)
CN (1) CN1183101C (no)
AR (1) AR021165A1 (no)
AT (1) ATE244697T1 (no)
AU (1) AU758808B2 (no)
BR (1) BR9912291A (no)
CA (1) CA2337945A1 (no)
CO (1) CO5080742A1 (no)
DE (1) DE69909486T2 (no)
DK (1) DK1098871T3 (no)
ES (1) ES2203163T3 (no)
HU (1) HUP0102705A3 (no)
ID (1) ID27261A (no)
IL (1) IL140586A (no)
NO (1) NO20010280L (no)
NZ (1) NZ509327A (no)
PE (1) PE20000880A1 (no)
PL (1) PL345621A1 (no)
PT (1) PT1098871E (no)
RU (1) RU2223947C2 (no)
SK (1) SK1032001A3 (no)
TR (1) TR200100166T2 (no)
TW (1) TW565546B (no)
WO (1) WO2000005196A1 (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR031473A1 (es) * 2000-11-20 2003-09-24 Lundbeck & Co As H Intensificadores de gaba en el tratamiento de enfermedades relacionadas con una reducida actividad neuroesteroide
ATE328864T1 (de) 2001-01-19 2006-06-15 Akzo Nobel Nv Alanin-2,6-dialkoxyphenylesterderivate als hypnotika

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1102011A (en) 1964-05-21 1968-02-07 Richardson Merrell Spa Phenol esters of amino acids
GB1160468A (en) 1967-05-08 1969-08-06 May & Baker Ltd Morpholine Derivative

Also Published As

Publication number Publication date
TW565546B (en) 2003-12-11
AR021165A1 (es) 2002-07-03
AU758808B2 (en) 2003-03-27
AU5160299A (en) 2000-02-14
CN1311770A (zh) 2001-09-05
PT1098871E (pt) 2003-11-28
BR9912291A (pt) 2001-04-17
WO2000005196A1 (en) 2000-02-03
EP1098871A1 (en) 2001-05-16
TR200100166T2 (tr) 2001-05-21
CO5080742A1 (es) 2001-09-25
EP1098871B1 (en) 2003-07-09
SK1032001A3 (en) 2001-08-06
HUP0102705A2 (hu) 2001-12-28
ATE244697T1 (de) 2003-07-15
NZ509327A (en) 2003-04-29
CN1183101C (zh) 2005-01-05
KR100599142B1 (ko) 2006-07-12
DE69909486D1 (de) 2003-08-14
KR20010071905A (ko) 2001-07-31
JP2002521358A (ja) 2002-07-16
IL140586A0 (en) 2002-02-10
HUP0102705A3 (en) 2002-11-28
NO20010280L (no) 2001-03-08
CA2337945A1 (en) 2000-02-03
PE20000880A1 (es) 2000-09-12
US6451854B1 (en) 2002-09-17
ES2203163T3 (es) 2004-04-01
DE69909486T2 (de) 2004-05-27
DK1098871T3 (da) 2003-10-27
NO20010280D0 (no) 2001-01-17
ID27261A (id) 2001-03-22
RU2223947C2 (ru) 2004-02-20
PL345621A1 (en) 2002-01-02

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees