IL138691A - Process for the preparation of 3-acyl-indoles - Google Patents

Process for the preparation of 3-acyl-indoles

Info

Publication number
IL138691A
IL138691A IL13869100A IL13869100A IL138691A IL 138691 A IL138691 A IL 138691A IL 13869100 A IL13869100 A IL 13869100A IL 13869100 A IL13869100 A IL 13869100A IL 138691 A IL138691 A IL 138691A
Authority
IL
Israel
Prior art keywords
indoles
acyl
preparation
Prior art date
Application number
IL13869100A
Other languages
English (en)
Other versions
IL138691A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL138691A0 publication Critical patent/IL138691A0/xx
Publication of IL138691A publication Critical patent/IL138691A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL13869100A 1999-10-01 2000-09-25 Process for the preparation of 3-acyl-indoles IL138691A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9923314.0A GB9923314D0 (en) 1999-10-01 1999-10-01 Acylation process

Publications (2)

Publication Number Publication Date
IL138691A0 IL138691A0 (en) 2001-10-31
IL138691A true IL138691A (en) 2005-03-20

Family

ID=10861993

Family Applications (1)

Application Number Title Priority Date Filing Date
IL13869100A IL138691A (en) 1999-10-01 2000-09-25 Process for the preparation of 3-acyl-indoles

Country Status (24)

Country Link
US (2) US6441192B1 (cs)
EP (1) EP1088817B1 (cs)
JP (1) JP3374125B2 (cs)
KR (1) KR100365458B1 (cs)
CN (1) CN1142140C (cs)
AR (1) AR035993A1 (cs)
AT (1) ATE233238T1 (cs)
AU (1) AU778663B2 (cs)
BR (1) BR0004578A (cs)
CA (1) CA2322346C (cs)
CZ (1) CZ297897B6 (cs)
DE (1) DE60001477T2 (cs)
DK (1) DK1088817T3 (cs)
ES (1) ES2188482T3 (cs)
GB (1) GB9923314D0 (cs)
HU (1) HUP0003862A3 (cs)
ID (1) ID27404A (cs)
IL (1) IL138691A (cs)
PL (1) PL342875A1 (cs)
RS (1) RS49983B (cs)
RU (1) RU2197480C2 (cs)
TR (1) TR200002834A2 (cs)
TW (1) TWI265923B (cs)
ZA (1) ZA200005216B (cs)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9923314D0 (en) * 1999-10-01 1999-12-08 Pfizer Ltd Acylation process
US6927296B2 (en) 2003-07-23 2005-08-09 Pfizer Inc. Process
IT1393700B1 (it) * 2009-04-22 2012-05-08 F S I Fabbrica Italiana Sint Sintesi di 3-{[(2r)-1-metilpirrolidin-2-il]metil}-5-[2-(fenilsulfonil)etil]-1h-indolo
WO2011024039A1 (en) * 2009-08-25 2011-03-03 Ramesh Babu Potluri Synthesis of novel 5-(2-(phenylsulfonyl)ethyl)-1h-indole derivatives
WO2011089614A1 (en) 2010-01-19 2011-07-28 Sms Pharmaceuticals Limited PROCESS FOR PREPARING ELETRIPTAN HYDROBROMIDE HAVING α-FORM
AU2021215709A1 (en) 2020-02-04 2022-09-01 Mindset Pharma Inc. 3-pyrrolidine-indole derivatives as serotonergic psychedelic agents for the treatment of CNS disorders

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK425384A (da) * 1983-09-28 1985-03-29 Nippon Zoki Pharmaceutical Co Acylindol-derivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater som indeholder dem
JPS625012A (ja) * 1985-06-28 1987-01-12 Chugai Ro Kogyo Kaisha Ltd 排熱回収バ−ナ
US5607951A (en) 1990-10-15 1997-03-04 Pfizer Inc Indole derivatives
US5559246A (en) 1990-10-15 1996-09-24 Pfizer Inc. Indole derivatives
US5578612A (en) 1990-10-15 1996-11-26 Pfizer Inc. Indole derivatives
US5559129A (en) 1990-10-15 1996-09-24 Pfizer Inc Indole derivatives
DE10299004I2 (de) * 1990-10-15 2006-03-16 Pfizer Indolderivate
US5545644A (en) 1990-10-15 1996-08-13 Pfizer Inc. Indole derivatives
JPH05154271A (ja) * 1991-12-05 1993-06-22 Mitsubishi Heavy Ind Ltd 連続式水洗機
GB9207930D0 (en) * 1992-04-10 1992-05-27 Pfizer Ltd Indoles
JPH064167A (ja) * 1992-06-18 1994-01-14 Nec Corp ディスク媒体障害の復旧方式
GB9417310D0 (en) 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
FR2735774B1 (fr) * 1995-06-21 1997-09-12 Sanofi Sa Utilisation de composes agonistes du recepteur cb2 humain pour la preparation de medicaments immunomodulateurs, nouveaux composes agonistes du recepteur cb2 et les compositions pharmaceutiques les contenant
US5998462A (en) * 1996-12-16 1999-12-07 Allelix Biopharmaceuticals Inc. 5-alkyl indole compounds
JPH10195048A (ja) * 1997-01-17 1998-07-28 Sumitomo Chem Co Ltd ３−（ニトロベンゾイル）インドール誘導体の製造法
HRP990416B1 (en) 1997-07-03 2002-04-30 Pfizer Pharmaceutical compositions containing eletriptan hemisulphate and caffeine
GB9923314D0 (en) * 1999-10-01 1999-12-08 Pfizer Ltd Acylation process

Also Published As

Publication number Publication date
EP1088817A3 (en) 2001-08-29
AR035993A1 (es) 2004-08-04
JP3374125B2 (ja) 2003-02-04
US20020188138A1 (en) 2002-12-12
ID27404A (id) 2001-04-05
JP2001131146A (ja) 2001-05-15
AU5951100A (en) 2001-04-05
EP1088817A2 (en) 2001-04-04
HK1034970A1 (en) 2001-11-09
DE60001477T2 (de) 2003-08-28
US6914145B2 (en) 2005-07-05
KR100365458B1 (ko) 2002-12-18
EP1088817B1 (en) 2003-02-26
GB9923314D0 (en) 1999-12-08
ATE233238T1 (de) 2003-03-15
CZ20003572A3 (cs) 2002-05-15
DK1088817T3 (da) 2003-04-22
RS49983B (sr) 2008-09-29
ZA200005216B (en) 2002-03-28
CN1142140C (zh) 2004-03-17
AU778663B2 (en) 2004-12-16
DE60001477D1 (de) 2003-04-03
YU53500A (sh) 2003-02-28
US6441192B1 (en) 2002-08-27
CA2322346A1 (en) 2001-04-01
CN1290697A (zh) 2001-04-11
CA2322346C (en) 2004-08-10
IL138691A0 (en) 2001-10-31
BR0004578A (pt) 2001-05-29
TWI265923B (en) 2006-11-11
KR20010050785A (ko) 2001-06-25
HUP0003862A3 (en) 2002-02-28
HUP0003862A2 (hu) 2001-12-28
CZ297897B6 (cs) 2007-04-25
HU0003862D0 (en) 2000-12-28
PL342875A1 (en) 2001-04-09
TR200002834A2 (tr) 2001-04-20
RU2197480C2 (ru) 2003-01-27
ES2188482T3 (es) 2003-07-01

Similar Documents

Publication Publication Date Title
HUP0100215A3 (en) Process for the preparation of substantially amorphous alpha-ol
HUP0202435A3 (en) Process for the preparation of naproxene nitroxyalkylesters
IL129906A0 (en) Process for the preparation of beta-isophorone
IL187126A0 (en) Process for the preparation of 4 - haloalkylnicotinonitriles
AU8824201A (en) Process for the preparation of dinapsoline
IL139023A0 (en) Process for the preparation of 2,3,5-trimethyl-p- benzoquinone
HUP0203407A3 (en) Process for the preparation of pyrazolopyridazine derivatives
IL145888A0 (en) Process for the preparation of substituted pyrimidines
AU5831500A (en) Process for the preparation of polyols
HUP0202865A3 (en) Process for the preparation of 2-cyanopyridines
GB2363605B (en) Process for the preparation of alpha-aminoketone derivatives
IL138691A (en) Process for the preparation of 3-acyl-indoles
HUP0203384A3 (en) Process for the preparation of ketimines
GB9909592D0 (en) Process for the preparation of calanolide precursors
IL150897A0 (en) Process for the preparation of acetyl-amidiniophenylalanyl cyclohexylglycyl-pyridinioalaninamides
GB0121486D0 (en) Processes for the preparation of Α-Aminoketones
IL149527A0 (en) Process for the preparation of ketimines
HUP9902745A3 (en) Process for the preparation of benzylcarbazate
IL190807A0 (en) Process for the preparation of 2-aminoethylpyridines
HUP0201518A3 (en) Process for the preparation of tetrafluorohalogenbenzenes
HUP0201574A3 (en) Process for the preparation of fumagillin
HU9904575D0 (en) Process for preparation of n-alkoxy-methyl-acidamides
AU6275300A (en) Process for the preparation of 2-cyano-5-hydroxypyrazine
GB0012249D0 (en) Process for the preparation of 11-oxaprostaglandins
IL140300A0 (en) Process for the preparation of amides

Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees