BR0004578A - Processo de acilação - Google Patents

Processo de acilação

Info

Publication number
BR0004578A
BR0004578A BR0004578-0A BR0004578A BR0004578A BR 0004578 A BR0004578 A BR 0004578A BR 0004578 A BR0004578 A BR 0004578A BR 0004578 A BR0004578 A BR 0004578A
Authority
BR
Brazil
Prior art keywords
acylation process
indols
acylation
acillation
indoles
Prior art date
Application number
BR0004578-0A
Other languages
English (en)
Inventor
Jolyon Francis Perkins
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of BR0004578A publication Critical patent/BR0004578A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Patente de Invenção: <B>"PROCESSO DE ACILAçãO"<D>. A presente invenção refere-se à acilação de indóis, especificamente à preparação de indóis acilados na posição 3 que podem ainda ser tratados para proporcionar indóis possuindo um substituinte alternativo na posição 3.
BR0004578-0A 1999-10-01 2000-10-02 Processo de acilação BR0004578A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9923314.0A GB9923314D0 (en) 1999-10-01 1999-10-01 Acylation process

Publications (1)

Publication Number Publication Date
BR0004578A true BR0004578A (pt) 2001-05-29

Family

ID=10861993

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0004578-0A BR0004578A (pt) 1999-10-01 2000-10-02 Processo de acilação

Country Status (25)

Country Link
US (2) US6441192B1 (pt)
EP (1) EP1088817B1 (pt)
JP (1) JP3374125B2 (pt)
KR (1) KR100365458B1 (pt)
CN (1) CN1142140C (pt)
AR (1) AR035993A1 (pt)
AT (1) ATE233238T1 (pt)
AU (1) AU778663B2 (pt)
BR (1) BR0004578A (pt)
CA (1) CA2322346C (pt)
CZ (1) CZ297897B6 (pt)
DE (1) DE60001477T2 (pt)
DK (1) DK1088817T3 (pt)
ES (1) ES2188482T3 (pt)
GB (1) GB9923314D0 (pt)
HK (1) HK1034970A1 (pt)
HU (1) HUP0003862A3 (pt)
ID (1) ID27404A (pt)
IL (1) IL138691A (pt)
PL (1) PL342875A1 (pt)
RS (1) RS49983B (pt)
RU (1) RU2197480C2 (pt)
TR (1) TR200002834A2 (pt)
TW (1) TWI265923B (pt)
ZA (1) ZA200005216B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9923314D0 (en) * 1999-10-01 1999-12-08 Pfizer Ltd Acylation process
US6927296B2 (en) 2003-07-23 2005-08-09 Pfizer Inc. Process
IT1393700B1 (it) * 2009-04-22 2012-05-08 F S I Fabbrica Italiana Sint Sintesi di 3-{[(2r)-1-metilpirrolidin-2-il]metil}-5-[2-(fenilsulfonil)etil]-1h-indolo
WO2011024039A1 (en) * 2009-08-25 2011-03-03 Ramesh Babu Potluri Synthesis of novel 5-(2-(phenylsulfonyl)ethyl)-1h-indole derivatives
WO2011089614A1 (en) 2010-01-19 2011-07-28 Sms Pharmaceuticals Limited PROCESS FOR PREPARING ELETRIPTAN HYDROBROMIDE HAVING α-FORM
IL295374A (en) 2020-02-04 2022-10-01 Mindset Pharma Inc 3-pyrrolidine indole derivatives as serotonergic psychedelics for the treatment of central nervous system disorders

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK425384A (da) * 1983-09-28 1985-03-29 Nippon Zoki Pharmaceutical Co Acylindol-derivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater som indeholder dem
JPS625012A (ja) * 1985-06-28 1987-01-12 Chugai Ro Kogyo Kaisha Ltd 排熱回収バ−ナ
US5607951A (en) 1990-10-15 1997-03-04 Pfizer Inc Indole derivatives
US5559246A (en) 1990-10-15 1996-09-24 Pfizer Inc. Indole derivatives
WO1992006973A1 (en) * 1990-10-15 1992-04-30 Pfizer Inc. Indole derivatives
US5545644A (en) 1990-10-15 1996-08-13 Pfizer Inc. Indole derivatives
US5578612A (en) 1990-10-15 1996-11-26 Pfizer Inc. Indole derivatives
US5559129A (en) 1990-10-15 1996-09-24 Pfizer Inc Indole derivatives
JPH05154271A (ja) * 1991-12-05 1993-06-22 Mitsubishi Heavy Ind Ltd 連続式水洗機
GB9207930D0 (en) * 1992-04-10 1992-05-27 Pfizer Ltd Indoles
JPH064167A (ja) * 1992-06-18 1994-01-14 Nec Corp ディスク媒体障害の復旧方式
GB9417310D0 (en) 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
FR2735774B1 (fr) * 1995-06-21 1997-09-12 Sanofi Sa Utilisation de composes agonistes du recepteur cb2 humain pour la preparation de medicaments immunomodulateurs, nouveaux composes agonistes du recepteur cb2 et les compositions pharmaceutiques les contenant
US5998462A (en) * 1996-12-16 1999-12-07 Allelix Biopharmaceuticals Inc. 5-alkyl indole compounds
JPH10195048A (ja) * 1997-01-17 1998-07-28 Sumitomo Chem Co Ltd ３−（ニトロベンゾイル）インドール誘導体の製造法
ID24528A (id) 1997-07-03 2000-07-20 Pfizer Komposisi-komposisi obat farmasi yang mengandung eletriptan hemisulfat dan kafein
GB9923314D0 (en) * 1999-10-01 1999-12-08 Pfizer Ltd Acylation process

Also Published As

Publication number Publication date
EP1088817B1 (en) 2003-02-26
IL138691A (en) 2005-03-20
CZ297897B6 (cs) 2007-04-25
ES2188482T3 (es) 2003-07-01
HU0003862D0 (en) 2000-12-28
EP1088817A3 (en) 2001-08-29
ZA200005216B (en) 2002-03-28
CA2322346C (en) 2004-08-10
TWI265923B (en) 2006-11-11
DE60001477T2 (de) 2003-08-28
RS49983B (sr) 2008-09-29
RU2197480C2 (ru) 2003-01-27
KR20010050785A (ko) 2001-06-25
HK1034970A1 (en) 2001-11-09
ATE233238T1 (de) 2003-03-15
JP3374125B2 (ja) 2003-02-04
CZ20003572A3 (cs) 2002-05-15
US6441192B1 (en) 2002-08-27
HUP0003862A2 (hu) 2001-12-28
AR035993A1 (es) 2004-08-04
US6914145B2 (en) 2005-07-05
TR200002834A2 (tr) 2001-04-20
JP2001131146A (ja) 2001-05-15
YU53500A (sh) 2003-02-28
CN1142140C (zh) 2004-03-17
GB9923314D0 (en) 1999-12-08
CA2322346A1 (en) 2001-04-01
AU778663B2 (en) 2004-12-16
CN1290697A (zh) 2001-04-11
EP1088817A2 (en) 2001-04-04
ID27404A (id) 2001-04-05
DK1088817T3 (da) 2003-04-22
IL138691A0 (en) 2001-10-31
US20020188138A1 (en) 2002-12-12
KR100365458B1 (ko) 2002-12-18
PL342875A1 (en) 2001-04-09
DE60001477D1 (de) 2003-04-03
HUP0003862A3 (en) 2002-02-28
AU5951100A (en) 2001-04-05

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 10A ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2116 DE 26/07/2011.