IL120844A0 - Fluorinated vitamin D3 analogs and their uses - Google Patents

Fluorinated vitamin D3 analogs and their uses

Info

Publication number
IL120844A0
IL120844A0 IL12084497A IL12084497A IL120844A0 IL 120844 A0 IL120844 A0 IL 120844A0 IL 12084497 A IL12084497 A IL 12084497A IL 12084497 A IL12084497 A IL 12084497A IL 120844 A0 IL120844 A0 IL 120844A0
Authority
IL
Israel
Prior art keywords
analogs
fluorinated vitamin
fluorinated
vitamin
Prior art date
Application number
IL12084497A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of IL120844A0 publication Critical patent/IL120844A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/59Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804Compounds having Si-O-C linkages
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Nutrition Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL12084497A 1996-05-23 1997-05-16 Fluorinated vitamin D3 analogs and their uses IL120844A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1821996P 1996-05-23 1996-05-23
US3990197P 1997-03-19 1997-03-19

Publications (1)

Publication Number Publication Date
IL120844A0 true IL120844A0 (en) 1997-09-30

Family

ID=26690870

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12084497A IL120844A0 (en) 1996-05-23 1997-05-16 Fluorinated vitamin D3 analogs and their uses

Country Status (26)

Country Link
EP (1) EP0808832B1 (ja)
JP (1) JP2859248B2 (ja)
KR (1) KR100253961B1 (ja)
CN (1) CN100402497C (ja)
AR (1) AR007776A1 (ja)
AT (1) ATE238278T1 (ja)
AU (1) AU733970B2 (ja)
BR (1) BR9703385A (ja)
CA (1) CA2205315C (ja)
CO (1) CO4940503A1 (ja)
CZ (1) CZ157797A3 (ja)
DE (1) DE69721123T2 (ja)
DK (1) DK0808832T3 (ja)
ES (1) ES2195049T3 (ja)
HR (1) HRP970272A2 (ja)
HU (1) HUP9700928A3 (ja)
IL (1) IL120844A0 (ja)
MA (1) MA24250A1 (ja)
NO (1) NO972278L (ja)
NZ (1) NZ314840A (ja)
PE (1) PE66798A1 (ja)
PL (1) PL320130A1 (ja)
PT (1) PT808832E (ja)
SG (1) SG70010A1 (ja)
TR (1) TR199700416A2 (ja)
YU (1) YU20097A (ja)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6008209A (en) * 1997-04-28 1999-12-28 Hoffmann-La Roche Inc. Method of using vitamin D3 analogs with bis C-20 side chains
DE19935771A1 (de) 1999-07-23 2001-02-01 Schering Ag Neue Vitamin D-Derivate mit cyclischen Substrukturen in den Seitenketten, Verfahren und Zwischenprodukte zu ihrer Herstellung und die Verwendung zur Herstellung von Arzneimitteln
AU2001278744A1 (en) * 2000-08-17 2002-02-25 Chugai Seiyaku Kabushiki Kaisha Remedial agent for osteoporosis
JP2005503434A (ja) * 2001-09-21 2005-02-03 エフ.ホフマン−ラ ロシュ アーゲー 3−デスオキシ−ビタミンd3類似体
AU2004203436A1 (en) 2003-09-24 2005-04-14 Bioxell Spa Compound and use in treatment
US20080318911A1 (en) * 2004-09-24 2008-12-25 Bioxell S.P.A. 20-Cyclopropyl, 26,27-Alkyl/Haloalkyl Vitamin D3 Compounds and Methods of Use Thereof
JP2008538114A (ja) * 2005-03-23 2008-10-09 ビオクセル エッセ ピ ア 20−アルキル、ジェミニビタミンd3化合物及びその使用方法
AU2011321624B2 (en) 2010-10-25 2015-03-26 Teijin Limited 23-yne-vitamin D3 derivative

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4141746A1 (de) * 1991-12-13 1993-06-17 Schering Ag 20-methyl-substituierte vitamin d-derivate
DE4220757A1 (de) * 1992-06-24 1994-01-05 Schering Ag Derivate in der Vitamin D-Reihe mit Modifikationen in der 20-Position, Verfahren zu ihrer Herstellung, Zwischenprodukte für dieses Verfahren, diese Derivate enthaltende pharmazeutische Präparate sowie deren Verwendung zur Herstellung von Arzneimitteln
US5428029A (en) * 1993-11-24 1995-06-27 Hoffmann-La Roche Inc. Vitamin D3 fluorinated analogs
US5384314B1 (en) * 1994-03-11 1997-08-05 Hoffmann La Roche 1alpha-fluoro-25-hydroxy-16-ene-23-yne-cholecalciferol
AU7295696A (en) * 1995-10-27 1997-05-22 F. Hoffmann-La Roche Ag Pharmaceutical composition for treating osteoporosis

Also Published As

Publication number Publication date
AR007776A1 (es) 1999-11-24
CZ157797A3 (en) 1997-12-17
EP0808832A3 (en) 1999-02-03
CA2205315C (en) 2006-10-24
HRP970272A2 (en) 1998-04-30
MX9703775A (es) 1998-06-30
HUP9700928A3 (en) 1999-07-28
SG70010A1 (en) 2000-01-25
JP2859248B2 (ja) 1999-02-17
ES2195049T3 (es) 2003-12-01
TR199700416A2 (xx) 1997-12-21
AU733970B2 (en) 2001-05-31
HU9700928D0 (en) 1997-07-28
PE66798A1 (es) 1998-10-22
AU2357697A (en) 1997-11-27
KR100253961B1 (ko) 2000-04-15
KR970074764A (ko) 1997-12-10
BR9703385A (pt) 1998-09-15
EP0808832B1 (en) 2003-04-23
DK0808832T3 (da) 2003-08-11
CA2205315A1 (en) 1997-11-23
ATE238278T1 (de) 2003-05-15
CN1172801A (zh) 1998-02-11
PT808832E (pt) 2003-07-31
NO972278L (no) 1997-11-24
DE69721123D1 (de) 2003-05-28
PL320130A1 (en) 1997-11-24
HUP9700928A2 (hu) 1998-01-28
NO972278D0 (no) 1997-05-20
NZ314840A (en) 1998-11-25
MA24250A1 (fr) 1998-04-01
DE69721123T2 (de) 2004-01-08
YU20097A (sh) 1999-09-27
JPH1045714A (ja) 1998-02-17
CO4940503A1 (es) 2000-07-24
CN100402497C (zh) 2008-07-16
EP0808832A2 (en) 1997-11-26

Similar Documents

Publication Publication Date Title
IL120843A0 (en) Vitamin D3 analogs and their uses
PL328822A1 (en) Human bikinine
EP0888151A4 (en) MECHANICAL BRAKE FOR RECALL
IL137793A0 (en) Fluorinated ionomers and their uses
GR3034832T3 (en) Fluorinated vitamin D3 analogs
ZA959517B (en) Leutherobin and analogs thereof
IL120844A0 (en) Fluorinated vitamin D3 analogs and their uses
HUT65350A (en) Fluorine-containing vitamin d3 analogues
GB9622842D0 (en) Shoe-sole
AU6735494A (en) Sports boarding
SG24096A1 (en) Fluorinated vitamin D3 derivative
ZA974332B (en) Fluorinated vitamin D3 analogs.
ZA933357B (en) Vitamin D3 fluorinated analogs
GB9619750D0 (en) Respirator faceseal
AU128539S (en) Handrail
AU129740S (en) Handrail
PL105498U1 (en) Footrest
TW295232U (en) Assembled-type emergency jacklight
GB9614397D0 (en) Emergency pinpointer
GB9423003D0 (en) Rescue fawiclos
GB9611001D0 (en) Balustrade
TW354901U (en) Improvement of respirator
HU9401780D0 (en) Orthoped shoe-sole
GB9617437D0 (en) Aircraft
AU132261S (en) Aircraft