IL119053A0 - Process for the preparation of some 4-hydroxypyrrolo Ú2,3-d¾ pyrimidine-L-glutamic acid derivatives and compounds prepared thereby - Google Patents

Process for the preparation of some 4-hydroxypyrrolo Ú2,3-d¾ pyrimidine-L-glutamic acid derivatives and compounds prepared thereby

Info

Publication number
IL119053A0
IL119053A0 IL11905396A IL11905396A IL119053A0 IL 119053 A0 IL119053 A0 IL 119053A0 IL 11905396 A IL11905396 A IL 11905396A IL 11905396 A IL11905396 A IL 11905396A IL 119053 A0 IL119053 A0 IL 119053A0
Authority
IL
Israel
Prior art keywords
hydroxypyrrolo
pyrimidine
preparation
glutamic acid
acid derivatives
Prior art date
Application number
IL11905396A
Other languages
English (en)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of IL119053A0 publication Critical patent/IL119053A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
IL11905396A 1992-06-22 1996-08-12 Process for the preparation of some 4-hydroxypyrrolo Ú2,3-d¾ pyrimidine-L-glutamic acid derivatives and compounds prepared thereby IL119053A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/902,116 US5235053A (en) 1992-06-22 1992-06-22 Process for the synthesis of 4-hydroxy-5-halopyrrold[2,3-d]pyrimidine intermediates
IL10605496 1996-08-12

Publications (1)

Publication Number Publication Date
IL119053A0 true IL119053A0 (en) 1996-11-14

Family

ID=25415324

Family Applications (3)

Application Number Title Priority Date Filing Date
IL11905393A IL119053A (en) 1992-06-22 1993-06-17 Process for the preparation of several derivatives of acid 4 - hydroxypyrrolo] D - 3, 2 [pyrimidine - L - glutamic, and compounds prepared by it
IL106054A IL106054A (en) 1992-06-22 1993-06-17 REGIOSELECTIVE PROCESS FOR THE PREPARATION OF 4-HYDROXY-5-HALO-7H- PYRROLO £2, 3-d| PYRIMIDINES
IL11905396A IL119053A0 (en) 1992-06-22 1996-08-12 Process for the preparation of some 4-hydroxypyrrolo Ú2,3-d¾ pyrimidine-L-glutamic acid derivatives and compounds prepared thereby

Family Applications Before (2)

Application Number Title Priority Date Filing Date
IL11905393A IL119053A (en) 1992-06-22 1993-06-17 Process for the preparation of several derivatives of acid 4 - hydroxypyrrolo] D - 3, 2 [pyrimidine - L - glutamic, and compounds prepared by it
IL106054A IL106054A (en) 1992-06-22 1993-06-17 REGIOSELECTIVE PROCESS FOR THE PREPARATION OF 4-HYDROXY-5-HALO-7H- PYRROLO £2, 3-d| PYRIMIDINES

Country Status (15)

Country Link
US (1) US5235053A (xx)
EP (1) EP0576211B1 (xx)
JP (1) JPH0656838A (xx)
KR (1) KR100285891B1 (xx)
AT (1) ATE204577T1 (xx)
BR (1) BR9302432A (xx)
CA (1) CA2098694A1 (xx)
DE (1) DE69330627T2 (xx)
DK (1) DK0576211T3 (xx)
ES (1) ES2160589T3 (xx)
HU (1) HU214019B (xx)
IL (3) IL119053A (xx)
MX (1) MX9303671A (xx)
PT (1) PT576211E (xx)
TW (1) TW226376B (xx)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL107041A (en) * 1992-09-25 2000-02-17 Lilly Co Eli Process for preparing omega(2-amino-4,7-dihydro-4-oxo-3H-pyrrolo-6-¬2,3-d¾pyrimidin-5-YL)alkarylcarboxylic acids and N-(omega-(2-amino-4,7-dihydro-4-oxo-3H-pyrrolo¬2,3-d¾pyrimidin-5-YL)alk-aroyl-4-glutamic acids
US5426187A (en) * 1993-11-30 1995-06-20 Eli Lilly And Company Process for the preparation of 4-hydroxy-5-substituted ethynylpyrrolo [2,3-d]pyrimidine intermediates
US6002004A (en) * 1995-03-28 1999-12-14 Witco Vinyl Additives Gmbh Pyrrolodiazine derivatives as stabilizers for chilorine-containing polymers
JP3711238B2 (ja) * 1997-08-05 2005-11-02 ファイザー・プロダクツ・インク 神経ペプチドＹ受容体アンタゴニストとしての４−アミノピロ−ル（３，２−ｄ）ピリミジン
CN100374441C (zh) * 2003-06-06 2008-03-12 天津倍方科技发展有限公司 二氢吡咯[2，3-d]嘧啶-4-酮衍生物，其制备方法及其制药用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO169490C (no) 1988-03-24 1992-07-01 Takeda Chemical Industries Ltd Analogifremgangsmaate for fremstilling av terapeutisk aktive pyrrolopyrimidinderivater
IL96531A (en) * 1989-12-11 1995-08-31 Univ Princeton History of Acid N- (Diomeric-H1-Pyrolo] D-2,3 [Pyrimidine-3-Ilacyl (-glutamic, preparation and pharmaceutical preparations containing them)
US5028608A (en) 1989-12-11 1991-07-02 The Trustees Of Princeton University N-(6-Amino-(pyrrolo(2,3-d)pyrimidin-3-ylacyl) )-glutamic acid derivatives

Also Published As

Publication number Publication date
DK0576211T3 (da) 2001-10-08
US5235053A (en) 1993-08-10
JPH0656838A (ja) 1994-03-01
IL119053A (en) 1998-12-06
IL106054A0 (en) 1993-10-20
BR9302432A (pt) 1994-01-11
TW226376B (xx) 1994-07-11
EP0576211B1 (en) 2001-08-22
PT576211E (pt) 2001-12-28
MX9303671A (es) 1993-12-01
IL106054A (en) 1997-07-13
EP0576211A3 (en) 1994-06-15
ES2160589T3 (es) 2001-11-16
CA2098694A1 (en) 1993-12-23
HUT65439A (en) 1994-06-28
DE69330627T2 (de) 2002-06-13
KR100285891B1 (ko) 2001-04-16
EP0576211A2 (en) 1993-12-29
KR940000461A (ko) 1994-01-03
DE69330627D1 (de) 2001-09-27
HU214019B (hu) 2000-06-28
HU9301829D0 (en) 1993-09-28
ATE204577T1 (de) 2001-09-15

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