IL113808A - Synthesis of enantiomeric benzoquinolinones - Google Patents

Synthesis of enantiomeric benzoquinolinones

Info

Publication number
IL113808A
IL113808A IL11380895A IL11380895A IL113808A IL 113808 A IL113808 A IL 113808A IL 11380895 A IL11380895 A IL 11380895A IL 11380895 A IL11380895 A IL 11380895A IL 113808 A IL113808 A IL 113808A
Authority
IL
Israel
Prior art keywords
compound
formula
reaction mixture
reaction
mixture
Prior art date
Application number
IL11380895A
Other languages
English (en)
Hebrew (he)
Other versions
IL113808A0 (en
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of IL113808A0 publication Critical patent/IL113808A0/xx
Publication of IL113808A publication Critical patent/IL113808A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/39Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton
    • C07C211/41Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems
    • C07C211/42Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems with six-membered aromatic rings being part of the condensed ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C07C319/20Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by reactions not involving the formation of sulfide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04Ortho- or peri-condensed ring systems
    • C07D221/06Ring systems of three rings
    • C07D221/10Aza-phenanthrenes
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00Systems containing two condensed rings
    • C07C2602/02Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Catalysts (AREA)
IL11380895A 1994-05-26 1995-05-22 Synthesis of enantiomeric benzoquinolinones IL113808A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24958294A 1994-05-26 1994-05-26

Publications (2)

Publication Number Publication Date
IL113808A0 IL113808A0 (en) 1995-08-31
IL113808A true IL113808A (en) 1998-12-06

Family

ID=22944128

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11380895A IL113808A (en) 1994-05-26 1995-05-22 Synthesis of enantiomeric benzoquinolinones

Country Status (14)

Country Link
EP (1) EP0684234B1 (fr)
JP (1) JPH07316136A (fr)
AT (1) ATE194979T1 (fr)
BR (1) BR9502557A (fr)
CA (1) CA2149988A1 (fr)
DE (1) DE69518112T2 (fr)
DK (1) DK0684234T3 (fr)
ES (1) ES2148438T3 (fr)
FI (1) FI952535A (fr)
GR (1) GR3034634T3 (fr)
HU (1) HU219450B (fr)
IL (1) IL113808A (fr)
PT (1) PT684234E (fr)
SI (1) SI0684234T1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5574160A (en) * 1994-05-26 1996-11-12 Eli Lilly And Company Syntheis of benzoquinolinones
AU754604B2 (en) * 1998-07-29 2002-11-21 Merck & Co., Inc. Tricyclic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL105168A0 (en) * 1992-04-03 1993-07-08 Lilly Co Eli Heteroannulation process

Also Published As

Publication number Publication date
FI952535A0 (fi) 1995-05-24
HUT72331A (en) 1996-04-29
GR3034634T3 (en) 2001-01-31
PT684234E (pt) 2000-12-29
JPH07316136A (ja) 1995-12-05
IL113808A0 (en) 1995-08-31
ATE194979T1 (de) 2000-08-15
HU9501509D0 (en) 1995-07-28
DE69518112D1 (de) 2000-08-31
EP0684234A1 (fr) 1995-11-29
HU219450B (hu) 2001-04-28
EP0684234B1 (fr) 2000-07-26
DE69518112T2 (de) 2001-03-15
BR9502557A (pt) 1996-06-04
SI0684234T1 (en) 2001-02-28
CA2149988A1 (fr) 1995-11-27
ES2148438T3 (es) 2000-10-16
FI952535A (fi) 1995-11-27
DK0684234T3 (da) 2000-09-18

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees