DE69518112T2 - Benzochinolinone Synthese - Google Patents

Benzochinolinone Synthese

Info

Publication number
DE69518112T2
DE69518112T2 DE69518112T DE69518112T DE69518112T2 DE 69518112 T2 DE69518112 T2 DE 69518112T2 DE 69518112 T DE69518112 T DE 69518112T DE 69518112 T DE69518112 T DE 69518112T DE 69518112 T2 DE69518112 T2 DE 69518112T2
Authority
DE
Germany
Prior art keywords
formula
compound
chem
prepare
combining
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69518112T
Other languages
English (en)
Other versions
DE69518112D1 (de
Inventor
James Edmund Audia
James Joseph Droste
Perry Clark Heath
Leland Otto Weigel
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Application granted granted Critical
Publication of DE69518112D1 publication Critical patent/DE69518112D1/de
Publication of DE69518112T2 publication Critical patent/DE69518112T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/39—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton
    • C07C211/41—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems
    • C07C211/42—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems with six-membered aromatic rings being part of the condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C07C319/20—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by reactions not involving the formation of sulfide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/10—Aza-phenanthrenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Catalysts (AREA)
DE69518112T 1994-05-26 1995-05-23 Benzochinolinone Synthese Expired - Fee Related DE69518112T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24958294A 1994-05-26 1994-05-26

Publications (2)

Publication Number Publication Date
DE69518112D1 DE69518112D1 (de) 2000-08-31
DE69518112T2 true DE69518112T2 (de) 2001-03-15

Family

ID=22944128

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69518112T Expired - Fee Related DE69518112T2 (de) 1994-05-26 1995-05-23 Benzochinolinone Synthese

Country Status (14)

Country Link
EP (1) EP0684234B1 (de)
JP (1) JPH07316136A (de)
AT (1) ATE194979T1 (de)
BR (1) BR9502557A (de)
CA (1) CA2149988A1 (de)
DE (1) DE69518112T2 (de)
DK (1) DK0684234T3 (de)
ES (1) ES2148438T3 (de)
FI (1) FI952535A (de)
GR (1) GR3034634T3 (de)
HU (1) HU219450B (de)
IL (1) IL113808A (de)
PT (1) PT684234E (de)
SI (1) SI0684234T1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5574160A (en) * 1994-05-26 1996-11-12 Eli Lilly And Company Syntheis of benzoquinolinones
US6048869A (en) * 1998-07-29 2000-04-11 Merck & Co., Inc. Tricyclic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL105168A0 (en) * 1992-04-03 1993-07-08 Lilly Co Eli Heteroannulation process

Also Published As

Publication number Publication date
HUT72331A (en) 1996-04-29
HU219450B (hu) 2001-04-28
GR3034634T3 (en) 2001-01-31
FI952535A0 (fi) 1995-05-24
PT684234E (pt) 2000-12-29
FI952535A (fi) 1995-11-27
JPH07316136A (ja) 1995-12-05
DK0684234T3 (da) 2000-09-18
IL113808A (en) 1998-12-06
SI0684234T1 (en) 2001-02-28
IL113808A0 (en) 1995-08-31
EP0684234B1 (de) 2000-07-26
EP0684234A1 (de) 1995-11-29
DE69518112D1 (de) 2000-08-31
HU9501509D0 (en) 1995-07-28
BR9502557A (pt) 1996-06-04
CA2149988A1 (en) 1995-11-27
ATE194979T1 (de) 2000-08-15
ES2148438T3 (es) 2000-10-16

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee