IL105255A - Perhydroisoindole derivatives their preparation and pharmaceutical compositions containing them - Google Patents

Perhydroisoindole derivatives their preparation and pharmaceutical compositions containing them

Info

Publication number
IL105255A
IL105255A IL10525593A IL10525593A IL105255A IL 105255 A IL105255 A IL 105255A IL 10525593 A IL10525593 A IL 10525593A IL 10525593 A IL10525593 A IL 10525593A IL 105255 A IL105255 A IL 105255A
Authority
IL
Israel
Prior art keywords
optionally
pct
preparation
date oct
optionally substituted
Prior art date
Application number
IL10525593A
Other languages
English (en)
Other versions
IL105255A0 (en
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of IL105255A0 publication Critical patent/IL105255A0/xx
Publication of IL105255A publication Critical patent/IL105255A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL10525593A 1992-04-10 1993-04-01 Perhydroisoindole derivatives their preparation and pharmaceutical compositions containing them IL105255A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR929204390A FR2689888B1 (fr) 1992-04-10 1992-04-10 Nouveaux derives de perhydroisoindole, leur preparation et les compositions pharmaceutiques qui les contiennent.

Publications (2)

Publication Number Publication Date
IL105255A0 IL105255A0 (en) 1993-08-18
IL105255A true IL105255A (en) 1997-02-18

Family

ID=9428707

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10525593A IL105255A (en) 1992-04-10 1993-04-01 Perhydroisoindole derivatives their preparation and pharmaceutical compositions containing them

Country Status (24)

Country Link
US (1) US5484804A (no)
EP (1) EP0635003B1 (no)
JP (1) JP3205557B2 (no)
KR (1) KR950700880A (no)
AT (1) ATE167472T1 (no)
AU (1) AU667214B2 (no)
CA (1) CA2133840A1 (no)
CZ (1) CZ284213B6 (no)
DE (1) DE69319235T2 (no)
DK (1) DK0635003T3 (no)
ES (1) ES2118232T3 (no)
FI (1) FI105023B (no)
FR (1) FR2689888B1 (no)
HU (1) HUT71354A (no)
IL (1) IL105255A (no)
MX (1) MX9301986A (no)
NO (1) NO300417B1 (no)
NZ (1) NZ251730A (no)
PL (1) PL172754B1 (no)
RU (1) RU2127260C1 (no)
SK (1) SK279032B6 (no)
TW (1) TW234119B (no)
WO (1) WO1993021155A1 (no)
ZA (1) ZA932527B (no)

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FR2700472B1 (fr) 1993-01-19 1995-02-17 Rhone Poulenc Rorer Sa Association synergisante ayant un effet antagoniste des récepteurs NK1 et NK2.
FR2703679B1 (fr) * 1993-04-05 1995-06-23 Rhone Poulenc Rorer Sa Nouveaux derives de perhydroisoindole, leur preparation et les compositions pharmaceutiques qui les contiennent.
FR2709752B1 (fr) * 1993-07-30 1995-10-06 Rhone Poulenc Rorer Sa Nouveaux dérivés de perhydroisoindole, leur préparation et les compositions pharmaceutiques qui les contiennent.
TW365603B (en) * 1993-07-30 1999-08-01 Rhone Poulenc Rorer Sa Novel perhydroisoindole derivatives, their preparation and pharmaceutical compositions which contain them
FR2710913B1 (fr) * 1993-10-07 1995-11-24 Rhone Poulenc Rorer Sa Nouveaux dérivés de perhydroisoindole, leur préparation et les compositions pharmaceutiques qui les contiennent.
FR2710842B1 (fr) * 1993-10-07 1995-11-24 Rhone Poulenc Rorer Sa Nouvelle application thérapeutique de dérivés de perhydroisoindole.
FR2725900B1 (fr) * 1994-10-21 1997-07-18 Sanofi Sa Utilisation d'antagonistes des recepteurs nk1 pour la preparation de medicaments a action cardioregulatrice
FR2727411B1 (fr) * 1994-11-30 1997-01-03 Rhone Poulenc Rorer Sa Nouveaux derives de perhydroisoindole, leur preparation et les compositions pharmaceutiques qui les contiennent
US6107325A (en) * 1995-01-17 2000-08-22 Qlt Phototherapeutics, Inc. Green porphyrins as immunomodulators
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Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR514273A (fr) * 1920-04-23 1921-03-07 Georges Loutz Bougie d'allumage électrique pour moteurs à explosions
US4042707A (en) * 1976-02-19 1977-08-16 E. I. Du Pont De Nemours And Company 3α-Arylhydroisoindoles
FR2654725B1 (fr) * 1989-11-23 1992-02-14 Rhone Poulenc Sante Nouveaux derives de l'isoindolone, leur preparation et les compositions pharmaceutiques qui les contiennent.
FR2676442B1 (fr) * 1991-05-17 1993-08-06 Rhone Poulenc Rorer Sa Nouveau derives de perhydroisoindole, leur preparation et les compositions pharmaceutiques qui les contiennent.
FR2689889B1 (fr) * 1992-04-10 1994-06-10 Rhone Poulenc Rorer Sa Nouveaux derives de perhydroisoindole, et leur preparation.

Also Published As

Publication number Publication date
HUT71354A (en) 1995-11-28
SK122094A3 (en) 1995-05-10
US5484804A (en) 1996-01-16
SK279032B6 (sk) 1998-05-06
CZ248294A3 (en) 1995-11-15
DE69319235D1 (de) 1998-07-23
ZA932527B (en) 1993-11-08
HU9402911D0 (en) 1995-01-30
NO943692D0 (no) 1994-10-03
FR2689888A1 (fr) 1993-10-15
FR2689888B1 (fr) 1994-06-10
IL105255A0 (en) 1993-08-18
JPH07505410A (ja) 1995-06-15
DE69319235T2 (de) 1999-01-07
WO1993021155A1 (fr) 1993-10-28
RU94045855A (ru) 1996-09-10
CA2133840A1 (fr) 1993-10-28
FI944729A0 (fi) 1994-10-07
TW234119B (no) 1994-11-11
AU667214B2 (en) 1996-03-14
NO300417B1 (no) 1997-05-26
FI105023B (fi) 2000-05-31
JP3205557B2 (ja) 2001-09-04
NO943692L (no) 1994-10-03
RU2127260C1 (ru) 1999-03-10
NZ251730A (en) 1995-08-28
AU3956593A (en) 1993-11-18
MX9301986A (es) 1994-05-31
CZ284213B6 (cs) 1998-09-16
EP0635003A1 (fr) 1995-01-25
FI944729L (fi) 1994-10-07
PL172754B1 (pl) 1997-11-28
ATE167472T1 (de) 1998-07-15
EP0635003B1 (fr) 1998-06-17
KR950700880A (ko) 1995-02-20
DK0635003T3 (da) 1999-02-15
ES2118232T3 (es) 1998-09-16

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