IL103440A - Thiano] B-2,3 [Pirazine-H4, H) -12,3 (Discussions and Pharmaceuticals Containing Them - Google Patents

Thiano] B-2,3 [Pirazine-H4, H) -12,3 (Discussions and Pharmaceuticals Containing Them

Info

Publication number
IL103440A
IL103440A IL10344092A IL10344092A IL103440A IL 103440 A IL103440 A IL 103440A IL 10344092 A IL10344092 A IL 10344092A IL 10344092 A IL10344092 A IL 10344092A IL 103440 A IL103440 A IL 103440A
Authority
IL
Israel
Prior art keywords
pyrazine
dione
mmol
ethyl
mixture
Prior art date
Application number
IL10344092A
Other languages
English (en)
Hebrew (he)
Other versions
IL103440A0 (en
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of IL103440A0 publication Critical patent/IL103440A0/xx
Publication of IL103440A publication Critical patent/IL103440A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL10344092A 1991-10-23 1992-10-15 Thiano] B-2,3 [Pirazine-H4, H) -12,3 (Discussions and Pharmaceuticals Containing Them IL103440A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK911771A DK177191D0 (da) 1991-10-23 1991-10-23 Heterocyclic compounds and their preparation and use

Publications (2)

Publication Number Publication Date
IL103440A0 IL103440A0 (en) 1993-03-15
IL103440A true IL103440A (en) 1996-03-31

Family

ID=8107934

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10344092A IL103440A (en) 1991-10-23 1992-10-15 Thiano] B-2,3 [Pirazine-H4, H) -12,3 (Discussions and Pharmaceuticals Containing Them

Country Status (17)

Country Link
US (1) US5284847A (es)
EP (1) EP0609371B1 (es)
JP (1) JP2519020B2 (es)
AT (1) ATE137239T1 (es)
AU (1) AU659243B2 (es)
CA (1) CA2121845A1 (es)
DE (1) DE69210255T2 (es)
DK (2) DK177191D0 (es)
ES (1) ES2088162T3 (es)
FI (1) FI941877A0 (es)
GR (1) GR3020487T3 (es)
IL (1) IL103440A (es)
NO (1) NO941476D0 (es)
NZ (1) NZ244849A (es)
PT (1) PT101002A (es)
WO (1) WO1993008197A1 (es)
ZA (1) ZA928096B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6037340A (en) * 1997-05-28 2000-03-14 Cadus Pharmaceutical Corporation Synthesis and use of thiophene- and pyrrole-based heteroaromatic compounds
US20020002199A1 (en) * 1998-03-12 2002-01-03 Lone Jeppesen Modulators of protein tyrosine phosphatases (ptpases)
ZA200605471B (en) * 2003-12-23 2007-11-28 Dow Agrosciences Llc Process for the preparation of pyridine derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO179551C (no) * 1987-11-10 1996-10-30 Novo Nordisk As Analogifremgangsmåte for fremstilling av terapeutisk virksomme kinoxalinforbindelser
US4902685A (en) * 1988-08-17 1990-02-20 American Home Products Corporation 2-amino-3-cyano-bicyclic pyridines/pyrazines as inhibitors of interleukin 1

Also Published As

Publication number Publication date
WO1993008197A1 (en) 1993-04-29
JP2519020B2 (ja) 1996-07-31
NO941476D0 (no) 1994-04-22
EP0609371B1 (en) 1996-04-24
ATE137239T1 (de) 1996-05-15
ZA928096B (en) 1994-04-20
NZ244849A (en) 1995-02-24
GR3020487T3 (en) 1996-10-31
AU2902592A (en) 1993-05-21
DK0609371T3 (da) 1996-08-12
IL103440A0 (en) 1993-03-15
FI941877A (fi) 1994-04-22
EP0609371A1 (en) 1994-08-10
DK177191D0 (da) 1991-10-23
JPH06510789A (ja) 1994-12-01
US5284847A (en) 1994-02-08
FI941877A0 (fi) 1994-04-22
ES2088162T3 (es) 1996-08-01
DE69210255T2 (de) 1996-11-28
NO941476L (es) 1994-06-22
AU659243B2 (en) 1995-05-11
DE69210255D1 (de) 1996-05-30
CA2121845A1 (en) 1993-04-29
PT101002A (pt) 1994-01-31

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
RH Patent void