IE51707B1 - Piperidine derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

Piperidine derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number
IE51707B1
IE51707B1 IE2500/81A IE250081A IE51707B1 IE 51707 B1 IE51707 B1 IE 51707B1 IE 2500/81 A IE2500/81 A IE 2500/81A IE 250081 A IE250081 A IE 250081A IE 51707 B1 IE51707 B1 IE 51707B1
Authority
IE
Ireland
Prior art keywords
radical
general formula
alkyl
piperidine derivative
acid addition
Prior art date
Application number
IE2500/81A
Other languages
English (en)
Other versions
IE812500L (en
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Priority to DK469381A priority Critical patent/DK157853C/da
Priority to FI813330A priority patent/FI77850C/fi
Priority to ES506500A priority patent/ES506500A0/es
Priority to IE2500/81A priority patent/IE51707B1/en
Priority to ZA817373A priority patent/ZA817373B/xx
Priority to NZ198748A priority patent/NZ198748A/en
Priority to NO813577A priority patent/NO153890C/no
Priority to AU76769/81A priority patent/AU545739B2/en
Priority to JP56170536A priority patent/JPS5872565A/ja
Priority to CA000388595A priority patent/CA1173039A/en
Priority to GR66337A priority patent/GR75364B/el
Priority to PT73875A priority patent/PT73875B/pt
Publication of IE812500L publication Critical patent/IE812500L/xx
Publication of IE51707B1 publication Critical patent/IE51707B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IE2500/81A 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them IE51707B1 (en)

Priority Applications (12)

Application Number Priority Date Filing Date Title
DK469381A DK157853C (da) 1981-10-23 1981-10-23 Analogifremgangsmaade til fremstilling af 4-benzyloxypiperidinderivater
FI813330A FI77850C (fi) 1981-10-23 1981-10-23 Foerfarande foer framstaellning av 4-bensyloxi- eller 4-naftylmetoxipiperidinderivat, vilka har antidepressiv verkan.
ES506500A ES506500A0 (es) 1981-10-23 1981-10-23 Procedimiento de preparacion de derivados de piperidina
IE2500/81A IE51707B1 (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
ZA817373A ZA817373B (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
NZ198748A NZ198748A (en) 1981-10-23 1981-10-23 Piperidine derivatives and pharmaceutical compositions
NO813577A NO153890C (no) 1981-10-23 1981-10-23 Analogifremgangsmaate for fremstilling av terapeutisk aktive piperidinderivater.
AU76769/81A AU545739B2 (en) 1981-10-23 1981-10-23 Piperidine derivatives
JP56170536A JPS5872565A (ja) 1981-10-23 1981-10-23 ピペリジン誘導体およびその製造方法
CA000388595A CA1173039A (en) 1981-10-23 1981-10-23 4-benzyloxypiperidine compounds
GR66337A GR75364B (enrdf_load_stackoverflow) 1981-10-23 1981-10-23
PT73875A PT73875B (fr) 1981-10-23 1981-10-23 Procede de preparation de derives de piperidine applicables en therapeutique

Applications Claiming Priority (12)

Application Number Priority Date Filing Date Title
DK469381A DK157853C (da) 1981-10-23 1981-10-23 Analogifremgangsmaade til fremstilling af 4-benzyloxypiperidinderivater
FI813330A FI77850C (fi) 1981-10-23 1981-10-23 Foerfarande foer framstaellning av 4-bensyloxi- eller 4-naftylmetoxipiperidinderivat, vilka har antidepressiv verkan.
ES506500A ES506500A0 (es) 1981-10-23 1981-10-23 Procedimiento de preparacion de derivados de piperidina
IE2500/81A IE51707B1 (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
ZA817373A ZA817373B (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
NZ198748A NZ198748A (en) 1981-10-23 1981-10-23 Piperidine derivatives and pharmaceutical compositions
NO813577A NO153890C (no) 1981-10-23 1981-10-23 Analogifremgangsmaate for fremstilling av terapeutisk aktive piperidinderivater.
AU76769/81A AU545739B2 (en) 1981-10-23 1981-10-23 Piperidine derivatives
JP56170536A JPS5872565A (ja) 1981-10-23 1981-10-23 ピペリジン誘導体およびその製造方法
CA000388595A CA1173039A (en) 1981-10-23 1981-10-23 4-benzyloxypiperidine compounds
GR66337A GR75364B (enrdf_load_stackoverflow) 1981-10-23 1981-10-23
PT73875A PT73875B (fr) 1981-10-23 1981-10-23 Procede de preparation de derives de piperidine applicables en therapeutique

Publications (2)

Publication Number Publication Date
IE812500L IE812500L (en) 1983-04-21
IE51707B1 true IE51707B1 (en) 1987-02-18

Family

ID=27582840

Family Applications (1)

Application Number Title Priority Date Filing Date
IE2500/81A IE51707B1 (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them

Country Status (12)

Country Link
JP (1) JPS5872565A (enrdf_load_stackoverflow)
AU (1) AU545739B2 (enrdf_load_stackoverflow)
CA (1) CA1173039A (enrdf_load_stackoverflow)
DK (1) DK157853C (enrdf_load_stackoverflow)
ES (1) ES506500A0 (enrdf_load_stackoverflow)
FI (1) FI77850C (enrdf_load_stackoverflow)
GR (1) GR75364B (enrdf_load_stackoverflow)
IE (1) IE51707B1 (enrdf_load_stackoverflow)
NO (1) NO153890C (enrdf_load_stackoverflow)
NZ (1) NZ198748A (enrdf_load_stackoverflow)
PT (1) PT73875B (enrdf_load_stackoverflow)
ZA (1) ZA817373B (enrdf_load_stackoverflow)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02148948U (enrdf_load_stackoverflow) * 1989-05-17 1990-12-18
US5169855A (en) * 1990-03-28 1992-12-08 Du Pont Merck Pharmaceutical Company Piperidine ether derivatives as psychotropic drugs or plant fungicides
JPH0535676U (ja) * 1991-06-06 1993-05-14 株式会社カネマス 乾燥海草の水戻し用パツク

Also Published As

Publication number Publication date
FI77850B (fi) 1989-01-31
GR75364B (enrdf_load_stackoverflow) 1984-07-13
DK469381A (da) 1983-04-24
AU7676981A (en) 1983-04-28
NO153890B (no) 1986-03-03
FI77850C (fi) 1989-05-10
ZA817373B (en) 1983-03-30
JPS5872565A (ja) 1983-04-30
NO153890C (no) 1986-06-11
PT73875B (fr) 1983-01-25
ES8206476A1 (es) 1982-08-16
PT73875A (fr) 1981-11-01
DK157853C (da) 1990-08-06
ES506500A0 (es) 1982-08-16
JPS6135177B2 (enrdf_load_stackoverflow) 1986-08-12
AU545739B2 (en) 1985-08-01
FI813330L (fi) 1983-04-24
NZ198748A (en) 1984-08-24
IE812500L (en) 1983-04-21
DK157853B (da) 1990-02-26
CA1173039A (en) 1984-08-21
NO813577L (no) 1983-04-25

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