IE49697B1 - Oxazoline and thiazoline derivatives and processes for their preparation - Google Patents
Oxazoline and thiazoline derivatives and processes for their preparationInfo
- Publication number
- IE49697B1 IE49697B1 IE787/80A IE78780A IE49697B1 IE 49697 B1 IE49697 B1 IE 49697B1 IE 787/80 A IE787/80 A IE 787/80A IE 78780 A IE78780 A IE 78780A IE 49697 B1 IE49697 B1 IE 49697B1
- Authority
- IE
- Ireland
- Prior art keywords
- alkyl
- formula
- compound
- phenyl
- halogen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/48—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Emergency Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Endocrinology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7913864 | 1979-04-20 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE800787L IE800787L (en) | 1980-10-20 |
| IE49697B1 true IE49697B1 (en) | 1985-11-27 |
Family
ID=10504680
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE787/80A IE49697B1 (en) | 1979-04-20 | 1980-04-18 | Oxazoline and thiazoline derivatives and processes for their preparation |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US4409216A (en, 2012) |
| EP (1) | EP0018107B1 (en, 2012) |
| JP (1) | JPS55141474A (en, 2012) |
| AT (1) | ATE2075T1 (en, 2012) |
| AU (1) | AU5758880A (en, 2012) |
| DE (1) | DE3061396D1 (en, 2012) |
| DK (1) | DK167580A (en, 2012) |
| ES (2) | ES8105306A1 (en, 2012) |
| FI (1) | FI801253A7 (en, 2012) |
| GR (1) | GR67301B (en, 2012) |
| IE (1) | IE49697B1 (en, 2012) |
| IL (1) | IL59803A0 (en, 2012) |
| NO (1) | NO801131L (en, 2012) |
| ZA (1) | ZA801970B (en, 2012) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2075805B1 (es) * | 1993-12-30 | 1996-10-16 | Univ Murcia | Procedimiento para la obtencion de iminooxazolinas n-n'-sustituidas. |
| DE102004008141A1 (de) | 2004-02-19 | 2005-09-01 | Abbott Gmbh & Co. Kg | Guanidinverbindungen und ihre Verwendung als Bindungspartner für 5-HT5-Rezeptoren |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3023103A (en) * | 1960-08-02 | 1962-02-27 | Gen Aniline & Film Corp | Antifoggants and stabilizers for photographic silver halide emulsions |
| DE2205744A1 (de) | 1972-02-08 | 1973-08-09 | Thomae Gmbh Dr K | Neue durch einen guanidinylidenrest substituierte heterocyclen und verfahren zu ihrer herstellung |
| NZ183570A (en) * | 1976-03-19 | 1979-06-08 | Mcneilab Inc | Heterocyclic guanidine derivatives, having anti-secretory and hypogliycaemic activity |
| CS225804B2 (cs) | 1976-03-19 | 1984-02-13 | Mcneilab Inc | Způsob výroby heterocyklických derivátů guanidinu |
| US4089965A (en) * | 1976-03-26 | 1978-05-16 | American Cyanamid Company | Thiazolylphenylguanidines as antirhinovirus agents |
| CA1201119A (en) * | 1978-09-18 | 1986-02-25 | Mcneilab, Inc. | Diaza-cyclic derivatives of guanidine |
| AU5263779A (en) * | 1978-11-29 | 1980-05-29 | Beecham Group Limited | Derivatives of thiazolidin-2-ylidene and oxazolidin-2-ylidene with hypoglycaemic acitivity |
-
1980
- 1980-03-27 AT AT80300949T patent/ATE2075T1/de active
- 1980-03-27 DE DE8080300949T patent/DE3061396D1/de not_active Expired
- 1980-03-27 EP EP80300949A patent/EP0018107B1/en not_active Expired
- 1980-04-02 ZA ZA00801970A patent/ZA801970B/xx unknown
- 1980-04-10 IL IL59803A patent/IL59803A0/xx unknown
- 1980-04-11 US US06/139,284 patent/US4409216A/en not_active Expired - Lifetime
- 1980-04-15 GR GR61687A patent/GR67301B/el unknown
- 1980-04-17 ES ES490675A patent/ES8105306A1/es not_active Expired
- 1980-04-18 AU AU57588/80A patent/AU5758880A/en not_active Abandoned
- 1980-04-18 IE IE787/80A patent/IE49697B1/en unknown
- 1980-04-18 NO NO801131A patent/NO801131L/no unknown
- 1980-04-18 DK DK167580A patent/DK167580A/da active IP Right Grant
- 1980-04-18 FI FI801253A patent/FI801253A7/fi not_active Application Discontinuation
- 1980-04-18 JP JP5155880A patent/JPS55141474A/ja active Pending
- 1980-12-09 ES ES497560A patent/ES497560A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| ES8200668A1 (es) | 1981-11-16 |
| ES490675A0 (es) | 1981-05-16 |
| GR67301B (en, 2012) | 1981-06-29 |
| IL59803A0 (en) | 1980-06-30 |
| IE800787L (en) | 1980-10-20 |
| DK167580A (da) | 1980-10-21 |
| AU5758880A (en) | 1980-10-23 |
| ES8105306A1 (es) | 1981-05-16 |
| DE3061396D1 (en) | 1983-01-27 |
| FI801253A7 (fi) | 1981-01-01 |
| ATE2075T1 (de) | 1983-01-15 |
| ZA801970B (en) | 1981-04-29 |
| ES497560A0 (es) | 1981-11-16 |
| NO801131L (no) | 1980-10-21 |
| EP0018107A1 (en) | 1980-10-29 |
| JPS55141474A (en) | 1980-11-05 |
| US4409216A (en) | 1983-10-11 |
| EP0018107B1 (en) | 1982-12-22 |
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