ID30393A - Senyawa tienopirimidina, pembuatan dan penggunaannya - Google Patents

Senyawa tienopirimidina, pembuatan dan penggunaannya

Info

Publication number
ID30393A
ID30393A IDW00200102298A ID20012298A ID30393A ID 30393 A ID30393 A ID 30393A ID W00200102298 A IDW00200102298 A ID W00200102298A ID 20012298 A ID20012298 A ID 20012298A ID 30393 A ID30393 A ID 30393A
Authority
ID
Indonesia
Prior art keywords
tienopirimidina
compounds
making
tienopirimidina compounds
Prior art date
Application number
IDW00200102298A
Other languages
English (en)
Inventor
Shuichi Furuya
Nobuhiro Suzuki
Nobuo Choh
Yoshi Nara
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of ID30393A publication Critical patent/ID30393A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
IDW00200102298A 1999-03-24 2000-03-23 Senyawa tienopirimidina, pembuatan dan penggunaannya ID30393A (id)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP7937199 1999-03-24
JP2000018019 2000-01-25

Publications (1)

Publication Number Publication Date
ID30393A true ID30393A (id) 2001-11-29

Family

ID=26420391

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW00200102298A ID30393A (id) 1999-03-24 2000-03-23 Senyawa tienopirimidina, pembuatan dan penggunaannya

Country Status (28)

Country Link
US (1) US6340686B1 (id)
EP (1) EP1163244B1 (id)
JP (1) JP3240293B2 (id)
KR (2) KR100533483B1 (id)
CN (1) CN1349536A (id)
AR (1) AR023152A1 (id)
AT (1) ATE261449T1 (id)
AU (1) AU764019B2 (id)
BR (1) BR0009297A (id)
CA (1) CA2368108C (id)
CZ (1) CZ294747B6 (id)
DE (1) DE60008862T2 (id)
DK (1) DK1163244T3 (id)
ES (1) ES2212992T3 (id)
HK (1) HK1042495B (id)
HU (1) HUP0200550A3 (id)
ID (1) ID30393A (id)
IL (1) IL145549A (id)
MX (1) MXPA01009566A (id)
MY (1) MY124726A (id)
NO (1) NO20014603L (id)
NZ (1) NZ514737A (id)
OA (1) OA11920A (id)
PL (1) PL351202A1 (id)
PT (1) PT1163244E (id)
SK (1) SK13552001A3 (id)
TW (1) TWI225863B (id)
WO (1) WO2000056739A1 (id)

Families Citing this family (36)

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US6828415B2 (en) * 1993-02-19 2004-12-07 Zentaris Gmbh Oligopeptide lyophilisate, their preparation and use
CN1539836A (zh) * 2000-02-29 2004-10-27 武田药品工业株式会社 制备噻吩并嘧啶衍生物的方法
AU2001248760A1 (en) * 2000-04-13 2001-10-30 Takeda Chemical Industries Ltd. Preventives/remedies for alzheimer's disease
US20040023987A1 (en) * 2000-06-14 2004-02-05 Yoshio Hata Sustained release compositions
EP1319409A4 (en) * 2000-09-22 2006-05-03 Takeda Pharmaceutical SOLID PREPARATIONS
WO2002043766A1 (fr) * 2000-11-29 2002-06-06 Takeda Chemical Industries, Ltd. Compositions medicinales et leur procede de preparation
AU2002221139A1 (en) * 2000-12-15 2002-06-24 Takeda Chemical Industries Ltd. Medicinal compositions of nonpeptidyl gonadotropin-releasing hormone agonist or antagonist, process for producing the same and use thereof
WO2002078669A1 (fr) * 2001-03-30 2002-10-10 Takeda Chemical Industries, Ltd. Solutions medicinales
MXPA04000986A (es) 2001-08-02 2005-02-17 Neurocrine Biosciences Inc 1,2,3-triazin-3,5-dionas sustituidas como antagonistas del receptor de hormona de liberacion de gonadotropina (gnrh).
KR20040030893A (ko) 2001-08-02 2004-04-09 뉴로크린 바이오사이언시즈 인코퍼레이티드 치환된 피리딘-4-온 및 고나도트로핀 분비 호르몬 수용체길항제로서의 이의 용도
AU2002321878A1 (en) 2001-08-02 2003-02-17 Neurocrine Biosciences, Inc. Pyridinone and pyridazinone derivatives as gonadotropin-releasing hormone receptor antagonists
JP2005500356A (ja) * 2001-08-02 2005-01-06 ニューロクライン バイオサイエンシーズ， インコーポレイテッド ゴナドトロピン放出ホルモンレセプターアンタゴニスト
AU2002324586B2 (en) 2001-08-02 2008-04-24 Neurocrine Biosciences, Inc. 1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists
US7569570B2 (en) * 2002-01-30 2009-08-04 Takeda Pharmaceutical Company Limited Thienopyrimidines, process for preparing the same and use thereof
US20050250793A1 (en) * 2002-04-12 2005-11-10 Masami Kusaka Preventives/remedies for hot flash
ATE384066T1 (de) * 2002-08-21 2008-02-15 Astrazeneca Ab Thieno-pyrrole verbindungen als antagonisten der gonadotropin-freisetzenden hormonrezeptoren
CN101153042A (zh) 2003-01-29 2008-04-02 武田药品工业株式会社 噻吩并嘧啶化合物及其用途
GB0307777D0 (en) 2003-04-04 2003-05-07 Medical Res Council Conjugate compounds
WO2006044902A2 (en) * 2004-10-18 2006-04-27 Bwt Property, Inc. A solid-state lighting apparatus for navigational aids
CN101272806A (zh) 2005-07-22 2008-09-24 武田药品工业株式会社 过早排卵抑制剂
EP2329823A4 (en) 2008-09-03 2013-04-03 Takeda Pharmaceutical METHOD FOR IMPROVING CAPACITY OF PREPARATION TO BE ABSORBED AND PREPARATION WHICH CAPACITY TO BE ABSORBED IS IMPROVED
EP2820021B1 (en) * 2012-02-28 2016-11-30 SK Chemicals Co., Ltd. Gonadotropin releasing hormone receptor antagonists, method for the preparation thereof and pharmaceutical composition comprising the same
HUE044048T2 (hu) 2012-09-28 2019-09-30 Takeda Pharmaceuticals Co Eljárás tienopirimidin származék elõállítására
SI3263110T1 (sl) 2015-02-26 2023-09-29 Takeda Pharmaceutical Company Limited Tableta, ki vsebuje derivat metoksisečnine in delce manitola
JP7043503B2 (ja) 2016-09-30 2022-03-29 ミオバント サイエンシズ ゲーエムベーハー 子宮筋腫及び子宮内膜症を治療する方法
JP7062673B2 (ja) 2016-09-30 2022-05-06 ミオバント サイエンシズ ゲーエムベーハー 前立腺がんの治療
KR101973074B1 (ko) * 2018-11-30 2019-04-26 주식회사 티움바이오 퓨로피리미딘 화합물의 염 및 결정형, 및 이를 포함하는 약학적 조성물
WO2021018105A1 (en) * 2019-07-29 2021-02-04 Sunshine Lake Pharma Co., Ltd. Substituted pyrimidinedione compounds and uses thereof
CN111574534B (zh) * 2020-05-25 2021-06-04 东莞市东阳光新药研发有限公司 苯基取代的噻吩并[2,3-d]嘧啶-2,4(1H,3H)-二酮类化合物及其用途
CN111909168B (zh) * 2020-07-31 2022-02-01 广东东阳光药业有限公司 含氮杂环基取代的嘧啶二酮类化合物及其用途
CN111925379B (zh) * 2020-07-31 2022-02-15 广东东阳光药业有限公司 含氮杂芳基取代的嘧啶二酮类化合物及其用途
CN113754679B (zh) * 2020-09-09 2023-04-07 广东东阳光药业有限公司 取代的嘧啶二酮类化合物及其用途
CN112047957B (zh) * 2020-09-09 2022-02-01 广东东阳光药业有限公司 取代的嘧啶二酮类化合物及其用途
CN113563304B (zh) * 2020-12-30 2022-06-28 上海博志研新药物技术有限公司 瑞卢戈利中间体及其制备方法
CN115260211B (zh) * 2021-04-29 2024-02-06 长春金赛药业有限责任公司 含噻吩稠环类衍生物、药物组合物及其制备方法和应用
CN113717149A (zh) * 2021-09-29 2021-11-30 成都伊诺达博医药科技有限公司 一种瑞卢戈利关键中间体及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW449600B (en) * 1994-04-19 2001-08-11 Takeda Chemical Industries Ltd Condensed-ring thiophene derivatives, their production and use
UY23948A1 (es) * 1995-02-08 2001-10-25 Takeda Chemical Industries Ltd Derivados de anillos condensados de tiofeno su producción y uso.
US5627786A (en) * 1995-02-10 1997-05-06 Micron Quantum Devices, Inc. Parallel processing redundancy scheme for faster access times and lower die area
WO1996028405A1 (fr) * 1995-03-10 1996-09-19 Nitto Chemical Industry Co., Ltd. Procede de production de derives de 1,2-ethanediol

Also Published As

Publication number Publication date
CZ294747B6 (cs) 2005-03-16
CA2368108C (en) 2009-12-22
DE60008862T2 (de) 2005-01-27
CA2368108A1 (en) 2000-09-28
OA11920A (en) 2006-04-12
DK1163244T3 (da) 2004-07-12
HUP0200550A2 (en) 2002-06-29
JP3240293B2 (ja) 2001-12-17
MY124726A (en) 2006-06-30
KR100370981B1 (ko) 2003-02-06
SK13552001A3 (sk) 2002-03-05
PT1163244E (pt) 2004-07-30
US6340686B1 (en) 2002-01-22
CN1349536A (zh) 2002-05-15
KR20010015920A (ko) 2001-02-26
CZ20013419A3 (cs) 2002-02-13
AR023152A1 (es) 2002-09-04
NZ514737A (en) 2003-10-31
NO20014603D0 (no) 2001-09-21
PL351202A1 (en) 2003-03-24
MXPA01009566A (es) 2002-05-14
IL145549A (en) 2005-11-20
HK1042495B (zh) 2004-10-08
WO2000056739A1 (en) 2000-09-28
AU764019B2 (en) 2003-08-07
AU3326200A (en) 2000-10-09
BR0009297A (pt) 2001-12-18
IL145549A0 (en) 2002-06-30
JP2001278884A (ja) 2001-10-10
KR100533483B1 (ko) 2005-12-05
ATE261449T1 (de) 2004-03-15
HUP0200550A3 (en) 2004-07-28
KR20010090430A (ko) 2001-10-18
EP1163244A1 (en) 2001-12-19
DE60008862D1 (de) 2004-04-15
TWI225863B (en) 2005-01-01
EP1163244B1 (en) 2004-03-10
HK1042495A1 (en) 2002-08-16
ES2212992T3 (es) 2004-08-16
NO20014603L (no) 2001-11-26

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