ID18770A - Senyawa-senyawa penghambat perpaduan siklik - Google Patents

Senyawa-senyawa penghambat perpaduan siklik

Info

Publication number
ID18770A
ID18770A IDP962581A ID962581A ID18770A ID 18770 A ID18770 A ID 18770A ID P962581 A IDP962581 A ID P962581A ID 962581 A ID962581 A ID 962581A ID 18770 A ID18770 A ID 18770A
Authority
ID
Indonesia
Prior art keywords
commitments
compounding
cycle
cycle commitments
compounding commitments
Prior art date
Application number
IDP962581A
Other languages
English (en)
Indonesian (id)
Inventor
Alfred Dr Jonczyk
Simon Dr Goodman
Beate Dr Diefenbach
Arne Dr Sutter
Gunter Dr Holzemann
Horst Prof Kessler
Michael Dechantsreiter
Original Assignee
Merck Patent Bmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Bmbh filed Critical Merck Patent Bmbh
Publication of ID18770A publication Critical patent/ID18770A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64—Cyclic peptides containing only normal peptide links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Communicable Diseases (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Vascular Medicine (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Toxicology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IDP962581A 1995-09-15 1996-09-12 Senyawa-senyawa penghambat perpaduan siklik ID18770A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19534177A DE19534177A1 (de) 1995-09-15 1995-09-15 Cyclische Adhäsionsinhibitoren

Publications (1)

Publication Number Publication Date
ID18770A true ID18770A (id) 1998-05-07

Family

ID=7772215

Family Applications (1)

Application Number Title Priority Date Filing Date
IDP962581A ID18770A (id) 1995-09-15 1996-09-12 Senyawa-senyawa penghambat perpaduan siklik

Country Status (29)

Country Link
US (1) US6001961A (fr)
EP (1) EP0770622B1 (fr)
JP (3) JP4115550B2 (fr)
KR (1) KR100438244B1 (fr)
CN (1) CN1203090C (fr)
AR (1) AR003574A1 (fr)
AT (1) ATE189461T1 (fr)
AU (1) AU717574B2 (fr)
BR (1) BR9603751A (fr)
CA (1) CA2185489C (fr)
CO (1) CO4750841A1 (fr)
CZ (1) CZ286713B6 (fr)
DE (2) DE19534177A1 (fr)
DK (1) DK0770622T3 (fr)
ES (1) ES2144179T3 (fr)
GR (1) GR3033293T3 (fr)
HU (1) HU224614B1 (fr)
ID (1) ID18770A (fr)
MX (1) MX9604100A (fr)
NO (1) NO316946B1 (fr)
PL (1) PL185125B1 (fr)
PT (1) PT770622E (fr)
RU (1) RU2157379C2 (fr)
SI (1) SI0770622T1 (fr)
SK (1) SK282391B6 (fr)
TR (1) TR199600716A2 (fr)
TW (1) TW517064B (fr)
UA (1) UA49799C2 (fr)
ZA (1) ZA967768B (fr)

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DE19613933A1 (de) * 1996-04-06 1997-10-09 Merck Patent Gmbh Cyclische Adhäsionsinhibitoren
AU733303C (en) 1996-05-31 2002-08-08 Scripps Research Institute, The Methods and compositions useful for inhibition of angiogenesis
PL330240A1 (en) * 1996-05-31 1999-05-10 Scripps Research Inst Methods and compositions useful in inhibiting angiogenesis in which alphavbeta5 acts as intermediary
WO1998037914A1 (fr) * 1997-02-26 1998-09-03 Toray Industries, Inc. Remedes contre l'hepatite
DE19842415A1 (de) * 1998-09-16 2000-03-23 Merck Patent Gmbh Pharmazeutische Zubereitung
WO2000038715A2 (fr) 1998-12-23 2000-07-06 G.D. Searle & Co. Procede d'utilisation d'un antagoniste de l'integrine et radiotherapie en tant que polytherapie dans le traitement des neoplasies
US6521593B1 (en) * 1999-02-01 2003-02-18 Childrens Hospital Los Angeles Methods for inhibiting brain tumor growth
RU2236251C2 (ru) * 1999-02-12 2004-09-20 Дзе Скриппс Рисерч Инститьют Способы лечения опухолей и метастазов с использованием комбинации антиангиогенной терапии и иммунотерапии
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PL316071A1 (en) 1997-03-17
JP4116062B2 (ja) 2008-07-09
DE19534177A1 (de) 1997-03-20
DK0770622T3 (da) 2000-07-03
EP0770622A2 (fr) 1997-05-02
AU6558096A (en) 1997-03-20
ATE189461T1 (de) 2000-02-15
RU2157379C2 (ru) 2000-10-10
DE59604363D1 (de) 2000-03-09
SI0770622T1 (en) 2000-08-31
JP2007186525A (ja) 2007-07-26
BR9603751A (pt) 1998-06-02
US6001961A (en) 1999-12-14
NO963853D0 (no) 1996-09-13
KR100438244B1 (ko) 2004-08-25
NO963853L (no) 1997-03-17
SK282391B6 (sk) 2002-01-07
EP0770622B1 (fr) 2000-02-02
JP2007016042A (ja) 2007-01-25
CA2185489C (fr) 2007-05-08
CZ264396A3 (en) 1997-04-16
AR003574A1 (es) 1998-08-05
CN1149588A (zh) 1997-05-14
KR970015598A (ko) 1997-04-28
ZA967768B (en) 1997-04-07
TR199600716A3 (fr) 1997-04-22
JP4115550B2 (ja) 2008-07-09
TR199600716A2 (tr) 1997-04-22
UA49799C2 (uk) 2002-10-15
NO316946B1 (no) 2004-07-05
PL185125B1 (pl) 2003-02-28
GR3033293T3 (en) 2000-09-29
MX9604100A (es) 1997-08-30
JPH09132593A (ja) 1997-05-20
HU224614B1 (hu) 2005-11-28
HUP9602507A2 (en) 1997-08-28
CN1203090C (zh) 2005-05-25
ES2144179T3 (es) 2000-06-01
HUP9602507A3 (en) 1998-01-28
TW517064B (en) 2003-01-11
CZ286713B6 (en) 2000-06-14
PT770622E (pt) 2000-07-31
HU9602507D0 (en) 1996-11-28
EP0770622A3 (fr) 1997-07-02
SK116796A3 (en) 2001-05-10
CO4750841A1 (es) 1999-03-31
AU717574B2 (en) 2000-03-30
CA2185489A1 (fr) 1997-03-16

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