HUT75114A - 1-oxo-2-(phenylsulfonyl-amino)-pentylpiperidine derivatives, process for producing them and pharmaceutical use of them - Google Patents

1-oxo-2-(phenylsulfonyl-amino)-pentylpiperidine derivatives, process for producing them and pharmaceutical use of them Download PDF

Info

Publication number
HUT75114A
HUT75114A HU9503782A HU9503782A HUT75114A HU T75114 A HUT75114 A HU T75114A HU 9503782 A HU9503782 A HU 9503782A HU 9503782 A HU9503782 A HU 9503782A HU T75114 A HUT75114 A HU T75114A
Authority
HU
Hungary
Prior art keywords
compound
formula
branched
straight
amino
Prior art date
Application number
HU9503782A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9503782D0 (en
Inventor
Jean Michel Altenburger
Gilbert Lassalle
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of HU9503782D0 publication Critical patent/HU9503782D0/hu
Publication of HUT75114A publication Critical patent/HUT75114A/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
HU9503782A 1994-12-23 1995-12-22 1-oxo-2-(phenylsulfonyl-amino)-pentylpiperidine derivatives, process for producing them and pharmaceutical use of them HUT75114A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9415549A FR2728570B1 (fr) 1994-12-23 1994-12-23 Derives de 1-oxo-2-(phenylsulfonylamino)pentylpiperidine, leur preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
HU9503782D0 HU9503782D0 (en) 1996-05-28
HUT75114A true HUT75114A (en) 1997-04-28

Family

ID=9470166

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9503782A HUT75114A (en) 1994-12-23 1995-12-22 1-oxo-2-(phenylsulfonyl-amino)-pentylpiperidine derivatives, process for producing them and pharmaceutical use of them

Country Status (21)

Country Link
US (2) US5602149A (no)
EP (1) EP0718307A2 (no)
JP (1) JPH08239380A (no)
KR (1) KR960022504A (no)
CN (1) CN1131153A (no)
AR (1) AR002259A1 (no)
AU (1) AU4062995A (no)
BR (1) BR9506062A (no)
CA (1) CA2166032A1 (no)
CO (1) CO4700285A1 (no)
CZ (1) CZ346095A3 (no)
FI (1) FI956251A (no)
FR (1) FR2728570B1 (no)
HU (1) HUT75114A (no)
IL (1) IL116532A0 (no)
NO (1) NO955242L (no)
NZ (1) NZ280735A (no)
PL (1) PL312028A1 (no)
SK (1) SK163895A3 (no)
TW (1) TW321647B (no)
ZA (1) ZA9510930B (no)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2728570B1 (fr) * 1994-12-23 1997-04-11 Synthelabo Derives de 1-oxo-2-(phenylsulfonylamino)pentylpiperidine, leur preparation et leur application en therapeutique
FR2749584B1 (fr) * 1996-06-11 1998-07-10 Synthelabo Derives de 1-oxo-2-(1h-imidazol-4-yl)pentylpiperidine, leur preparation et leur application en therapeutique
FR2756285B1 (fr) * 1996-11-22 1998-12-18 Synthelabo Derives de n-(imidazolylbutyle)benzenesulfonamide, leur preparation et leur application en therapeutique
FR2758326B1 (fr) * 1997-01-16 1999-02-12 Synthelabo Derives de pyridone, leur prepaparation et leur utilisation comme intermediaires de synthese
FR2765220B1 (fr) * 1997-06-25 1999-07-30 Synthelabo Derives de 1-oxo-2-(phenylsulfonyl)aminopentyle, leur preparation et leur application en therapeutique
FR2771094B1 (fr) * 1997-11-19 2000-02-04 Synthelabo Derives de piperidine-2-carboxylate, leur preparation et leur application en therapeutique
FR2806722B1 (fr) * 2000-03-23 2002-05-17 Sanofi Synthelabo Derives de n-(heterocyclylbutyl) benzene-ou pyridine sulfonamide, leur preparation et leur application en therapeutique

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1338645C (en) * 1987-01-06 1996-10-15 George R. Pettit Isolation, structural elucidation and synthesis of novel antineoplastic substances denominated "combretastatins"
US5312828A (en) * 1989-06-14 1994-05-17 Finkelstein Joseph A Substituted imidazoles having angiotensin II receptor blocking activity
US5136043A (en) * 1989-06-17 1992-08-04 Hoechst Aktiengesellschaft Process for the preparation of aromatic sulfonyl chlorides
FR2689130B1 (fr) * 1992-03-30 1994-05-27 Synthelabo Derives de 1-[2 (arylsulfonylamino)ethyl-1-oxo] piperidine, leur preparation et leur application en therapeutique.
US5401851A (en) * 1992-06-03 1995-03-28 Eli Lilly And Company Angiotensin II antagonists
US5612360A (en) * 1992-06-03 1997-03-18 Eli Lilly And Company Angiotensin II antagonists
DE4240708A1 (de) * 1992-12-03 1994-06-09 Bayer Ag Verfahren zur Herstellung von Natriumsalzen nitrogruppenhaltiger aromatischer Sulfinsäuren
JP3466614B2 (ja) * 1993-02-12 2003-11-17 コルバス・インターナショナル、インコーポレイテッド 血栓症のインヒビター
FR2710066B1 (fr) 1993-09-14 1995-10-20 Synthelabo Dérivés de 1-[2-amino-5-[1-(triphénylméthyl-1H-imidazol-4-yl]-1-oxopentyl]piperidine, leur préparation et leur utilisation comme intermédiaires de synthèse.
DE69433585D1 (de) * 1993-12-29 2004-04-08 Syngenta Participations Ag Vinylcarboxamid-Derivate als Insectizide und Akarizide
DE4423061C1 (de) * 1994-07-01 1996-01-18 Hoechst Ag Verfahren zur Herstellung von Biphenylen mit Palladacyclen als Katalysatoren
FR2728570B1 (fr) * 1994-12-23 1997-04-11 Synthelabo Derives de 1-oxo-2-(phenylsulfonylamino)pentylpiperidine, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
KR960022504A (ko) 1996-07-18
BR9506062A (pt) 1997-12-23
FR2728570B1 (fr) 1997-04-11
NZ280735A (en) 1997-06-24
US5602149A (en) 1997-02-11
AR002259A1 (es) 1998-03-11
NO955242D0 (no) 1995-12-22
ZA9510930B (en) 1996-06-24
NO955242L (no) 1996-06-24
IL116532A0 (en) 1996-03-31
CO4700285A1 (es) 1998-12-29
AU4062995A (en) 1996-07-04
FI956251A (fi) 1996-06-24
SK163895A3 (en) 1996-09-04
JPH08239380A (ja) 1996-09-17
HU9503782D0 (en) 1996-05-28
CA2166032A1 (fr) 1996-06-24
FR2728570A1 (fr) 1996-06-28
PL312028A1 (en) 1996-06-24
EP0718307A3 (no) 1996-08-07
US5753667A (en) 1998-05-19
EP0718307A2 (fr) 1996-06-26
CN1131153A (zh) 1996-09-18
CZ346095A3 (en) 1996-07-17
FI956251A0 (fi) 1995-12-22
TW321647B (no) 1997-12-01

Similar Documents

Publication Publication Date Title
JP2657760B2 (ja) ４−アミノキナゾリン誘導体およびそれを含有する医薬品
JP2633085B2 (ja) アミド官能基を有するインドリン誘導体、それらの調製、およびそれらが内在する医薬組成物
US4863904A (en) Dipeptides as renin inhibitors
JPH04506222A (ja) Ｎ−置換複素環誘導体およびその製法
EA001280B1 (ru) Замещенные n-[(аминоиминометил или аминометил)фенил] пропиламиды
JP2003040852A (ja) Ｃｏｘ−２阻害薬の合成方法
WO2003002554A1 (fr) Composes de piperazine
JPH06506699A (ja) 抗血栓性ペプチドおよび偽ペプチド
JPH08501099A (ja) 血小板凝集阻害剤
HUT52525A (en) Process for producing retroviral proteaz-inhibitors and pharmaceutical compositions containing them as active components
HUT75114A (en) 1-oxo-2-(phenylsulfonyl-amino)-pentylpiperidine derivatives, process for producing them and pharmaceutical use of them
JP2707936B2 (ja) β−オキソ−β−ベンゼンプロパンチオアミド誘導体
JP2007501267A (ja) 新規イミダゾール誘導体、その製造法及びその医薬としての使用
JP2650117B2 (ja) Ｎ−複素環式アルコール誘導体
JP5103563B2 (ja) ソマトスタチン受容体１及び／又は４選択的アゴニスト及びアンタゴニスト
JPH08508501A (ja) フィブリノーゲンレセプターアンタゴニスト
WO1996015117A1 (fr) Compose optiquement actif
HU211269A9 (en) Piperazinecarboxylic acid its preparation and pharmaceutical compositions containing it
JPH09505040A (ja) アンタゴニストとしての４−（１ｈ−２−メチルイミダゾ４．５−ｃピリジニルメチル）−フェニルスルホンアミドカルボン酸誘導体
FR2781221A1 (fr) Piperazinones substituees en alpha
US6291457B1 (en) Compounds having cytokine inhibitory activity
EP1098888A1 (fr) Derives de piperazinones et leurs applications
FR2781223A1 (fr) Bispiperidines et leurs applications therapeutiques
RU2339634C2 (ru) Кристаллическая форма
HUT54983A (en) Process for producing new thioformamide derivatives and pharmaceutical compositions comprising same

Legal Events

Date Code Title Description
DFC4 Cancellation of temporary protection due to refusal