HUT65694A - Process for producing saccharin derivatives - Google Patents

Process for producing saccharin derivatives Download PDF

Info

Publication number
HUT65694A
HUT65694A HU9203561A HU9203561A HUT65694A HU T65694 A HUT65694 A HU T65694A HU 9203561 A HU9203561 A HU 9203561A HU 9203561 A HU9203561 A HU 9203561A HU T65694 A HUT65694 A HU T65694A
Authority
HU
Hungary
Prior art keywords
formula
lower alkyl
lower alkoxy
compounds
compound
Prior art date
Application number
HU9203561A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9203561D0 (en
Inventor
Dennis John Hlasta
Albert Joseph Mura
Chakrapani Subramanyam
Richard Paul Dunlap
Lee Hamilton Latimer
Ranjit Chimanlal Desai
Original Assignee
Sterling Winthrop Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sterling Winthrop Inc filed Critical Sterling Winthrop Inc
Publication of HU9203561D0 publication Critical patent/HU9203561D0/hu
Publication of HUT65694A publication Critical patent/HUT65694A/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
HU9203561A 1991-11-15 1992-11-13 Process for producing saccharin derivatives HUT65694A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US79303591A 1991-11-15 1991-11-15

Publications (2)

Publication Number Publication Date
HU9203561D0 HU9203561D0 (en) 1993-01-28
HUT65694A true HUT65694A (en) 1994-07-28

Family

ID=25158888

Family Applications (2)

Application Number Title Priority Date Filing Date
HU9203561A HUT65694A (en) 1991-11-15 1992-11-13 Process for producing saccharin derivatives
HU95P/P00612P HU211664A9 (en) 1991-11-15 1995-06-30 Saccharin derivative proteolytic enzime inhibitors

Family Applications After (1)

Application Number Title Priority Date Filing Date
HU95P/P00612P HU211664A9 (en) 1991-11-15 1995-06-30 Saccharin derivative proteolytic enzime inhibitors

Country Status (15)

Country Link
EP (1) EP0542371A1 (US06251921-20010626-C00395.png)
JP (1) JPH06122675A (US06251921-20010626-C00395.png)
KR (1) KR930010016A (US06251921-20010626-C00395.png)
AU (1) AU656027B2 (US06251921-20010626-C00395.png)
CA (1) CA2082774A1 (US06251921-20010626-C00395.png)
CZ (1) CZ338892A3 (US06251921-20010626-C00395.png)
FI (1) FI925166A (US06251921-20010626-C00395.png)
HU (2) HUT65694A (US06251921-20010626-C00395.png)
IL (1) IL103747A (US06251921-20010626-C00395.png)
MX (1) MX9206568A (US06251921-20010626-C00395.png)
NO (1) NO302887B1 (US06251921-20010626-C00395.png)
NZ (1) NZ245126A (US06251921-20010626-C00395.png)
RU (1) RU2114835C1 (US06251921-20010626-C00395.png)
SG (1) SG52778A1 (US06251921-20010626-C00395.png)
TW (1) TW282463B (US06251921-20010626-C00395.png)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5322144A (en) * 1990-07-18 1994-06-21 Otis Elevator Company Active control of elevator platform
US5308938A (en) * 1990-07-18 1994-05-03 Otis Elevator Company Elevator active suspension system
US5294757A (en) * 1990-07-18 1994-03-15 Otis Elevator Company Active vibration control system for an elevator, which reduces horizontal and rotational forces acting on the car
US5321217A (en) * 1990-07-18 1994-06-14 Otis Elevator Company Apparatus and method for controlling an elevator horizontal suspension
US5306818A (en) * 1990-11-01 1994-04-26 Sterling Winthrop Inc. Tetrahydro 2-saccharinylmerthyl aryl carboxylates
US5378720A (en) * 1991-12-19 1995-01-03 Sterling Winthrop Inc. Saccharin derivative proteolytic enzyme inhibitors
AU668694B2 (en) * 1991-12-19 1996-05-16 Sanofi-Synthelabo Saccharin derivative proteolytic enzyme inhibitors
TW226016B (US06251921-20010626-C00395.png) * 1991-12-30 1994-07-01 Sterling Winthrop Inc
DE19533643A1 (de) * 1995-09-12 1997-03-13 Nycomed Arzneimittel Gmbh Neue cyclische Derivate von Benzolsulfonamiden
AU7127100A (en) * 1999-09-10 2001-04-10 Procter & Gamble Company, The Enzyme inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE159720T1 (de) * 1989-05-04 1997-11-15 Sanofi Sa Saccharinderivate zur verwendung als proteolytische enzyminhibitoren sowie verfahren zur herstellung
US5236917A (en) * 1989-05-04 1993-08-17 Sterling Winthrop Inc. Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
DE3917597A1 (de) * 1989-05-26 1990-11-29 Schering Ag Neue leukotrien-b(pfeil abwaerts)4(pfeil abwaerts)-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
AU642537B2 (en) * 1990-11-01 1993-10-21 Sanofi 2-saccharinylmethyl aryl carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof

Also Published As

Publication number Publication date
CZ338892A3 (en) 1993-06-16
KR930010016A (ko) 1993-06-21
SG52778A1 (en) 1998-09-28
FI925166A0 (fi) 1992-11-13
CA2082774A1 (en) 1993-05-16
AU656027B2 (en) 1995-01-19
FI925166A (fi) 1993-05-16
TW282463B (US06251921-20010626-C00395.png) 1996-08-01
IL103747A (en) 1998-06-15
MX9206568A (es) 1993-05-01
RU2114835C1 (ru) 1998-07-10
AU2605792A (en) 1993-05-20
NO924402L (no) 1993-05-18
JPH06122675A (ja) 1994-05-06
IL103747A0 (en) 1993-04-04
NZ245126A (en) 1996-01-26
NO924402D0 (no) 1992-11-13
EP0542371A1 (en) 1993-05-19
HU9203561D0 (en) 1993-01-28
NO302887B1 (no) 1998-05-04
HU211664A9 (en) 1995-12-28

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Legal Events

Date Code Title Description
DGB9 Succession in title of applicant

Owner name: SANOFI, FR

DFC4 Cancellation of temporary protection due to refusal