NO924402L - Sakkarinderivater med proteolytisk enzyminhiberende aktivitet - Google Patents

Sakkarinderivater med proteolytisk enzyminhiberende aktivitet

Info

Publication number
NO924402L
NO924402L NO92924402A NO924402A NO924402L NO 924402 L NO924402 L NO 924402L NO 92924402 A NO92924402 A NO 92924402A NO 924402 A NO924402 A NO 924402A NO 924402 L NO924402 L NO 924402L
Authority
NO
Norway
Prior art keywords
succarine
enzymin
proteolytic
derivatives
inhibitive activity
Prior art date
Application number
NO92924402A
Other languages
English (en)
Other versions
NO302887B1 (no
NO924402D0 (no
Inventor
Richard Paul Dunlap
Albert Joseph Mura
Dennis John Hlasta
Ranjit Chimanlal Desai
Lee Hamilton Latimer
Chakrapani Subramanyam
Original Assignee
Sterling Winthrop Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sterling Winthrop Inc filed Critical Sterling Winthrop Inc
Publication of NO924402D0 publication Critical patent/NO924402D0/no
Publication of NO924402L publication Critical patent/NO924402L/no
Publication of NO302887B1 publication Critical patent/NO302887B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
NO924402A 1991-11-15 1992-11-13 Sakkarinderivater med proteolytisk enzyminhiberende aktivitet, farmasöytisk preparat inneholdende slike derivater samt anvendelse derav NO302887B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US79303591A 1991-11-15 1991-11-15

Publications (3)

Publication Number Publication Date
NO924402D0 NO924402D0 (no) 1992-11-13
NO924402L true NO924402L (no) 1993-05-18
NO302887B1 NO302887B1 (no) 1998-05-04

Family

ID=25158888

Family Applications (1)

Application Number Title Priority Date Filing Date
NO924402A NO302887B1 (no) 1991-11-15 1992-11-13 Sakkarinderivater med proteolytisk enzyminhiberende aktivitet, farmasöytisk preparat inneholdende slike derivater samt anvendelse derav

Country Status (15)

Country Link
EP (1) EP0542371A1 (no)
JP (1) JPH06122675A (no)
KR (1) KR930010016A (no)
AU (1) AU656027B2 (no)
CA (1) CA2082774A1 (no)
CZ (1) CZ338892A3 (no)
FI (1) FI925166A (no)
HU (2) HUT65694A (no)
IL (1) IL103747A (no)
MX (1) MX9206568A (no)
NO (1) NO302887B1 (no)
NZ (1) NZ245126A (no)
RU (1) RU2114835C1 (no)
SG (1) SG52778A1 (no)
TW (1) TW282463B (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5321217A (en) * 1990-07-18 1994-06-14 Otis Elevator Company Apparatus and method for controlling an elevator horizontal suspension
US5294757A (en) * 1990-07-18 1994-03-15 Otis Elevator Company Active vibration control system for an elevator, which reduces horizontal and rotational forces acting on the car
US5308938A (en) * 1990-07-18 1994-05-03 Otis Elevator Company Elevator active suspension system
US5322144A (en) * 1990-07-18 1994-06-21 Otis Elevator Company Active control of elevator platform
US5306818A (en) * 1990-11-01 1994-04-26 Sterling Winthrop Inc. Tetrahydro 2-saccharinylmerthyl aryl carboxylates
US5378720A (en) * 1991-12-19 1995-01-03 Sterling Winthrop Inc. Saccharin derivative proteolytic enzyme inhibitors
AU668694B2 (en) * 1991-12-19 1996-05-16 Sanofi-Synthelabo Saccharin derivative proteolytic enzyme inhibitors
TW226016B (no) * 1991-12-30 1994-07-01 Sterling Winthrop Inc
DE19533643A1 (de) * 1995-09-12 1997-03-13 Nycomed Arzneimittel Gmbh Neue cyclische Derivate von Benzolsulfonamiden
JP2003508480A (ja) * 1999-09-10 2003-03-04 ザ、プロクター、エンド、ギャンブル、カンパニー 酵素インヒビター

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH04507095A (ja) * 1989-05-04 1992-12-10 サノフィ 蛋白分解酵素阻害剤として有用なサッカリン誘導体及びその製造
US5236917A (en) * 1989-05-04 1993-08-17 Sterling Winthrop Inc. Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
DE3917597A1 (de) * 1989-05-26 1990-11-29 Schering Ag Neue leukotrien-b(pfeil abwaerts)4(pfeil abwaerts)-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
AU642537B2 (en) * 1990-11-01 1993-10-21 Sanofi 2-saccharinylmethyl aryl carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof

Also Published As

Publication number Publication date
IL103747A (en) 1998-06-15
HUT65694A (en) 1994-07-28
NO302887B1 (no) 1998-05-04
NO924402D0 (no) 1992-11-13
FI925166A0 (fi) 1992-11-13
KR930010016A (ko) 1993-06-21
EP0542371A1 (en) 1993-05-19
NZ245126A (en) 1996-01-26
AU656027B2 (en) 1995-01-19
JPH06122675A (ja) 1994-05-06
RU2114835C1 (ru) 1998-07-10
CA2082774A1 (en) 1993-05-16
HU9203561D0 (en) 1993-01-28
IL103747A0 (en) 1993-04-04
HU211664A9 (en) 1995-12-28
SG52778A1 (en) 1998-09-28
MX9206568A (es) 1993-05-01
AU2605792A (en) 1993-05-20
CZ338892A3 (en) 1993-06-16
FI925166A (fi) 1993-05-16
TW282463B (no) 1996-08-01

Similar Documents

Publication Publication Date Title
NO924401L (no) 2-substituerte sakkarinderivater med proteolytisk enzym-inhiberende aktivitet
DE69125537T2 (de) Alpha-keto-amidderivate mit Protease inhibierender Aktivität
DE59208263D1 (de) 3-Aryl-4-hydroxy-delta3-dihydrofuranon- und 3-Aryl-4-hydroxy-delta3-dihydrothiophenon-Derivate
DE69208877T2 (de) Chinuclidinderivate
NO922182L (no) Krystallinske oksatiolan-derivater
DE68925161T2 (de) Alkylavermectin-Derivate
DE68927948T2 (de) Trehalosderivate
FI925763A (fi) Fungicida 2-imidazolin-5-on- och 2-imidazolin-5-tionderivat
DK371989A (da) Amidderivater
NO901759D0 (no) Dipeptidderivater med enzym-hemmende virkning.
DE68927657T2 (de) Butynylaminderivate
NO924402L (no) Sakkarinderivater med proteolytisk enzyminhiberende aktivitet
NO922521D0 (no) Piperidinyletanolderivater med terapeutisk virkning
FI925469A (fi) Tiazolylsubstituerade kinolylymetoxifenylaettiksyraderivat
NO894944D0 (no) Dipeptid-derivater med enzym-hemmende virkning.
DK160389A (da) Aryldionderivater
ATA155589A (de) Mitomycinphosphat-derivate
DE69211197T2 (de) 1-Hydroxyvitamin D-Derivate
ITMI912422A0 (it) Derivati ossimici ad attivita' fungicida
KR930702353A (ko) 2- 카르바페넴 유도체
DK93893D0 (da) Svingplov med gribearm
FI37U1 (fi) Tillaegsanordning i samband med personlyftaren
DK124390A (da) Prostaglandinderivater med antitrombotisk virkning
NO920307L (no) Nye dihydro-isokinolinderivater med farmasoeytisk virkning
DE69227554D1 (de) Indolinospirobenzopyran-derivate