HUS1600061I1 - 4[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]-2-pirimidinil]amino]benzonitril - Google Patents

4[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]-2-pirimidinil]amino]benzonitril

Info

Publication number
HUS1600061I1
HUS1600061I1 HUS1600061C HUS1600061C HUS1600061I1 HU S1600061 I1 HUS1600061 I1 HU S1600061I1 HU S1600061 C HUS1600061 C HU S1600061C HU S1600061 C HUS1600061 C HU S1600061C HU S1600061 I1 HUS1600061 I1 HU S1600061I1
Authority
HU
Hungary
Prior art keywords
amino
cyanoethenyl
benzonitrile
dimethylphenyl
pyrimidinyl
Prior art date
Application number
HUS1600061C
Other languages
English (en)
Hungarian (hu)
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38091637&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUS1600061(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from MYPI20043578A external-priority patent/MY169670A/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HUS1600061I1 publication Critical patent/HUS1600061I1/hu

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Hybrid Cells (AREA)
HUS1600061C 2004-09-02 2016-12-20 4[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]-2-pirimidinil]amino]benzonitril HUS1600061I1 (hu)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
MYPI20043578A MY169670A (en) 2003-09-03 2004-09-02 Combinations of a pyrimidine containing nnrti with rt inhibitors
PCT/EP2004/052028 WO2005021001A1 (en) 2003-09-03 2004-09-03 Combinations of a pyrimidine containing nnrti with rt inhibitors
EP05101467 2005-02-25
EP05108086.9A EP1632232B3 (en) 2004-09-02 2005-09-02 Salt of 4[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile

Publications (1)

Publication Number Publication Date
HUS1600061I1 true HUS1600061I1 (hu) 2017-01-30

Family

ID=38091637

Family Applications (2)

Application Number Title Priority Date Filing Date
HUS1600060C HUS1600060I1 (hu) 2004-09-02 2016-12-20 4[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]-2-pirimidinil]amino]benzonitril
HUS1600061C HUS1600061I1 (hu) 2004-09-02 2016-12-20 4[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]-2-pirimidinil]amino]benzonitril

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HUS1600060C HUS1600060I1 (hu) 2004-09-02 2016-12-20 4[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]-2-pirimidinil]amino]benzonitril

Country Status (21)

Country Link
EP (1) EP1632232B3 (enExample)
JP (1) JP4912309B2 (enExample)
CN (1) CN104586850A (enExample)
AT (1) ATE508748T1 (enExample)
BR (1) BRPI0514871A (enExample)
CY (3) CY1112249T1 (enExample)
DK (1) DK1632232T6 (enExample)
EA (1) EA013686B1 (enExample)
ES (1) ES2371442T7 (enExample)
FR (2) FR16C1023I1 (enExample)
HK (1) HK1210029A1 (enExample)
HU (2) HUS1600060I1 (enExample)
IL (1) IL181650A (enExample)
LT (2) LTC1632232I2 (enExample)
ME (1) ME01246B (enExample)
MX (1) MX2007002595A (enExample)
NI (1) NI200700068A (enExample)
NO (3) NO340654B1 (enExample)
PT (1) PT1632232E (enExample)
RS (1) RS51923B2 (enExample)
SI (1) SI1632232T1 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY169670A (en) 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
USRE50189E1 (en) * 2006-01-20 2024-10-29 Janssen Sciences Ireland Unlimited Company Long term treatment of HIV-infection with TMC278
TWI494133B (zh) 2007-03-14 2015-08-01 Tibotec Pharm Ltd 重組用粉末
EA025852B1 (ru) * 2010-11-19 2017-02-28 Джилид Сайэнс, Инк. ТЕРАПЕВТИЧЕСКИЕ КОМПОЗИЦИИ, СОДЕРЖАЩИЕ РИЛПИВИРИН HCl И ТЕНОФОВИРА ДИЗОПРОКСИЛФУМАРАТ
EP2643294B1 (en) * 2011-04-15 2016-08-24 Emcure Pharmaceuticals Limited An improved rilpivirine process
EP2604593A1 (en) 2011-12-14 2013-06-19 Sandoz AG Polymorph of Rilpivirine hydrochloride and its use as antiviral
WO2013087794A1 (en) 2011-12-14 2013-06-20 Sandoz Ag Polymorph of rilpivirine hydrochloride and its use as antiviral
EP2628732A1 (en) 2012-02-20 2013-08-21 Sandoz AG Novel crystalline form of rilpivirine hydrochloride
WO2013153161A2 (en) 2012-04-11 2013-10-17 Sandoz Ag Novel polymorph of rilpivirine hydrochloride
WO2013153162A1 (en) 2012-04-11 2013-10-17 Sandoz Ag Polymorph of rilpivirine hydrochloride
CN103570688B (zh) * 2012-07-19 2016-06-08 中国科学院上海药物研究所 2，5-二氨甲基吡嗪类化合物、其药物组合物、制备方法和用途
GR1008965B (el) * 2015-12-02 2017-02-28 Φαρματεν Ανωνυμος Βιομηχανικη Και Εμπορικη Εταιρεια Φαρμακευτικων Ιατρικων Και Καλλυντικων Προϊοντων Φαρμακευτικο σκευασμα που περιλαμβανει δαρουναβιρη και μεθοδος παρασκευης αυτου
RU2616267C1 (ru) * 2016-01-25 2017-04-13 Закрытое Акционерное Общество "БИОКОМ" Твердая лекарственная форма индинавира немедленного высвобождения и способ ее получения
CA3039562A1 (en) * 2016-10-24 2018-05-03 Janssen Sciences Ireland Unlimited Company Dispersible compositions
JP7287906B2 (ja) * 2017-06-30 2023-06-06 ヴィーブ ヘルスケア カンパニー 組み合わせ並びにその使用及びそれによる治療
CN114392241B (zh) * 2022-01-10 2023-07-25 安徽贝克生物制药有限公司 一种利匹韦林片及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6307543B1 (en) * 1998-09-10 2001-10-23 Silicon Image, Inc. Bi-directional data transfer using two pair of differential lines as a single additional differential pair
JO3429B1 (ar) * 2001-08-13 2019-10-20 Janssen Pharmaceutica Nv مشتقات برميدينات مثبطة فيروس الايدز
MY169670A (en) * 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
CN101481356B (zh) * 2002-08-09 2012-07-11 詹森药业有限公司 制备4-[[4-[[4-(2-氰基乙烯基)-2,6-二甲基苯基]氨基]-2-嘧啶基]氨基]苄腈的方法
AU2002350719A1 (en) * 2002-11-29 2004-06-23 Janssen Pharmaceutica N.V. Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base
US20070021449A1 (en) * 2003-02-07 2007-01-25 Jan Heeres Pyrimidine derivatives for the prevention of hiv infection

Also Published As

Publication number Publication date
ATE508748T1 (de) 2011-05-15
CY2016050I1 (el) 2017-07-12
HK1210029A1 (en) 2016-04-15
NO2017063I1 (no) 2017-11-21
EA200700536A1 (ru) 2007-08-31
JP4912309B2 (ja) 2012-04-11
ES2371442T7 (es) 2022-05-12
JP2008511592A (ja) 2008-04-17
EP1632232A1 (en) 2006-03-08
EP1632232B3 (en) 2022-03-30
RS51923B2 (sr) 2022-05-31
CY2016051I1 (el) 2017-07-12
LTC1632232I2 (lt) 2024-09-10
DK1632232T3 (da) 2011-08-22
DK1632232T6 (da) 2022-04-19
SI1632232T1 (sl) 2011-09-30
FR16C1023I1 (fr) 2017-02-03
IL181650A (en) 2012-08-30
CN104586850A (zh) 2015-05-06
FR16C1025I1 (fr) 2017-02-03
NO2017065I1 (no) 2017-11-21
ES2371442T3 (es) 2012-01-02
IL181650A0 (en) 2007-07-04
ME01246B (me) 2013-06-20
EA013686B1 (ru) 2010-06-30
NO340654B1 (no) 2017-05-22
NI200700068A (es) 2016-09-29
LTPA2016042I1 (lt) 2017-01-10
CY1112249T1 (el) 2015-12-09
MX2007002595A (es) 2007-04-25
EP1632232B1 (en) 2011-05-11
NO20071745L (no) 2007-04-02
HUS1600060I1 (hu) 2017-01-30
LTPA2016043I1 (lt) 2017-01-10
PT1632232E (pt) 2011-08-02
RS51923B (sr) 2012-02-29
FR16C1025I2 (fr) 2025-11-21
BRPI0514871A (pt) 2008-06-24

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HUS1600061I1 (hu) 4[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]-2-pirimidinil]amino]benzonitril
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