HUP1600128A2 - A new process for the preparation of elvitegravir - Google Patents

A new process for the preparation of elvitegravir

Info

Publication number
HUP1600128A2
HUP1600128A2 HU1600128A HUP1600128A HUP1600128A2 HU P1600128 A2 HUP1600128 A2 HU P1600128A2 HU 1600128 A HU1600128 A HU 1600128A HU P1600128 A HUP1600128 A HU P1600128A HU P1600128 A2 HUP1600128 A2 HU P1600128A2
Authority
HU
Hungary
Prior art keywords
elvitegravir
preparation
new process
new
Prior art date
Application number
HU1600128A
Other languages
English (en)
Hungarian (hu)
Inventor
Stanislav Radl
Jan Stach
Original Assignee
Zentiva As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentiva As filed Critical Zentiva As
Publication of HUP1600128A2 publication Critical patent/HUP1600128A2/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
HU1600128A 2013-07-11 2014-07-03 A new process for the preparation of elvitegravir HUP1600128A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CZ2013-544A CZ307255B6 (cs) 2013-07-11 2013-07-11 Nový způsob přípravy elvitegraviru
PCT/CZ2014/000076 WO2015003670A1 (en) 2013-07-11 2014-07-03 A new process for the preparation of elvitegravir

Publications (1)

Publication Number Publication Date
HUP1600128A2 true HUP1600128A2 (en) 2016-07-28

Family

ID=51229772

Family Applications (1)

Application Number Title Priority Date Filing Date
HU1600128A HUP1600128A2 (en) 2013-07-11 2014-07-03 A new process for the preparation of elvitegravir

Country Status (4)

Country Link
CN (1) CN105377818B (zh)
CZ (1) CZ307255B6 (zh)
HU (1) HUP1600128A2 (zh)
WO (1) WO2015003670A1 (zh)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105315203A (zh) * 2014-06-06 2016-02-10 上海迪赛诺化学制药有限公司 一种v型埃替拉韦晶体及其制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200401663T1 (tr) 2002-11-20 2005-04-21 Japan Tobacco Inc. 4-oksokuinolin bileşiği ve bunun HIV integraz inhibitörü olarak kullanımı.
US7531554B2 (en) * 2004-05-20 2009-05-12 Japan Tobacco Inc. 4-oxoquinoline compound and use thereof as HIV integrase inhibitor
CN101437801B (zh) * 2006-03-06 2013-02-06 日本烟草产业株式会社 制备4-氧代喹啉化合物的方法
BRPI0716752A2 (pt) * 2006-09-12 2013-09-17 Gilead Sciences Inc processo e intermediÁrios para preparo de inibidores de intergrase
WO2011004389A2 (en) 2009-06-18 2011-01-13 Matrix Laboratories Ltd An improved process for the preparation of elvitegravir
CZ304983B6 (cs) * 2012-10-12 2015-03-11 Zentiva, K.S. Způsob výroby a nové intermediáty syntézy elvitegraviru
CZ304984B6 (cs) * 2012-10-12 2015-03-11 Zentiva, K.S. Zlepšený způsob výroby a nové intermediáty syntézy elvitegraviru

Also Published As

Publication number Publication date
CN105377818B (zh) 2018-03-30
CZ307255B6 (cs) 2018-05-02
CZ2013544A3 (cs) 2015-01-21
CN105377818A (zh) 2016-03-02
WO2015003670A1 (en) 2015-01-15

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Legal Events

Date Code Title Description
FA9A Lapse of provisional patent protection due to relinquishment or protection considered relinquished