HUP1600128A2 - A new process for the preparation of elvitegravir - Google Patents
A new process for the preparation of elvitegravirInfo
- Publication number
- HUP1600128A2 HUP1600128A2 HU1600128A HUP1600128A HUP1600128A2 HU P1600128 A2 HUP1600128 A2 HU P1600128A2 HU 1600128 A HU1600128 A HU 1600128A HU P1600128 A HUP1600128 A HU P1600128A HU P1600128 A2 HUP1600128 A2 HU P1600128A2
- Authority
- HU
- Hungary
- Prior art keywords
- elvitegravir
- preparation
- new process
- new
- Prior art date
Links
- JUZYLCPPVHEVSV-LJQANCHMSA-N elvitegravir Chemical compound COC1=CC=2N([C@H](CO)C(C)C)C=C(C(O)=O)C(=O)C=2C=C1CC1=CC=CC(Cl)=C1F JUZYLCPPVHEVSV-LJQANCHMSA-N 0.000 title 1
- 229960003586 elvitegravir Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CZ2013-544A CZ307255B6 (en) | 2013-07-11 | 2013-07-11 | A new method of preparing elvitegravir |
| PCT/CZ2014/000076 WO2015003670A1 (en) | 2013-07-11 | 2014-07-03 | A new process for the preparation of elvitegravir |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HUP1600128A2 true HUP1600128A2 (en) | 2016-07-28 |
Family
ID=51229772
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU1600128A HUP1600128A2 (en) | 2013-07-11 | 2014-07-03 | A new process for the preparation of elvitegravir |
Country Status (4)
| Country | Link |
|---|---|
| CN (1) | CN105377818B (en) |
| CZ (1) | CZ307255B6 (en) |
| HU (1) | HUP1600128A2 (en) |
| WO (1) | WO2015003670A1 (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105315203A (en) * | 2014-06-06 | 2016-02-10 | 上海迪赛诺化学制药有限公司 | V-type elvitegravir crystal and preparation method thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0306214B1 (en) | 2002-11-20 | 2017-08-08 | Japan Tobacco Inc. | 4-OXOQUINOLINE COMPOUND AND USE OF THIS AS HIV INTEGRASE INHIBITOR |
| WO2005113509A1 (en) * | 2004-05-20 | 2005-12-01 | Japan Tobacco Inc. | Novel 4-oxoquinoline compound and use thereof as hiv integrase inhibitor |
| US8420821B2 (en) * | 2006-03-06 | 2013-04-16 | Japan Tobacco Inc. | Process for production of 4-oxoquinoline compound |
| PT2069280E (en) | 2006-09-12 | 2015-06-08 | Gilead Sciences Inc | Process and intermediates for preparing hiv integrase inhibitors |
| WO2011004389A2 (en) * | 2009-06-18 | 2011-01-13 | Matrix Laboratories Ltd | An improved process for the preparation of elvitegravir |
| CZ304984B6 (en) * | 2012-10-12 | 2015-03-11 | Zentiva, K.S. | Enhanced process for preparing and novel intermediates of elvitegravir synthesis |
| CZ304983B6 (en) * | 2012-10-12 | 2015-03-11 | Zentiva, K.S. | Preparation process and novel intermediates of elvitegravir synthesis |
-
2013
- 2013-07-11 CZ CZ2013-544A patent/CZ307255B6/en not_active IP Right Cessation
-
2014
- 2014-07-03 HU HU1600128A patent/HUP1600128A2/en unknown
- 2014-07-03 CN CN201480038026.3A patent/CN105377818B/en not_active Expired - Fee Related
- 2014-07-03 WO PCT/CZ2014/000076 patent/WO2015003670A1/en active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| CZ307255B6 (en) | 2018-05-02 |
| WO2015003670A1 (en) | 2015-01-15 |
| CZ2013544A3 (en) | 2015-01-21 |
| CN105377818A (en) | 2016-03-02 |
| CN105377818B (en) | 2018-03-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA9A | Lapse of provisional patent protection due to relinquishment or protection considered relinquished |