HUP0900417A3 - Polymorphs of donepezil hydrochloride and process for production and pharmaceutical compositions containing them - Google Patents
Polymorphs of donepezil hydrochloride and process for production and pharmaceutical compositions containing themInfo
- Publication number
- HUP0900417A3 HUP0900417A3 HU0900417A HUP0900417A HUP0900417A3 HU P0900417 A3 HUP0900417 A3 HU P0900417A3 HU 0900417 A HU0900417 A HU 0900417A HU P0900417 A HUP0900417 A HU P0900417A HU P0900417 A3 HUP0900417 A3 HU P0900417A3
- Authority
- HU
- Hungary
- Prior art keywords
- polymorphs
- production
- pharmaceutical compositions
- compositions containing
- donepezil hydrochloride
- Prior art date
Links
- 229960003135 donepezil hydrochloride Drugs 0.000 title 1
- XWAIAVWHZJNZQQ-UHFFFAOYSA-N donepezil hydrochloride Chemical compound [H+].[Cl-].O=C1C=2C=C(OC)C(OC)=CC=2CC1CC(CC1)CCN1CC1=CC=CC=C1 XWAIAVWHZJNZQQ-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Investigating Or Analysing Materials By Optical Means (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP14629396 | 1996-06-07 | ||
PCT/JP1997/001932 WO1997046527A1 (en) | 1996-06-07 | 1997-06-06 | Polymorphs of donepezil hydrochloride and process for production |
Publications (2)
Publication Number | Publication Date |
---|---|
HU0900417D0 HU0900417D0 (en) | 2009-08-28 |
HUP0900417A3 true HUP0900417A3 (en) | 2012-12-28 |
Family
ID=15404413
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0900417A HUP0900417A3 (en) | 1996-06-07 | 1997-06-06 | Polymorphs of donepezil hydrochloride and process for production and pharmaceutical compositions containing them |
Country Status (17)
Country | Link |
---|---|
US (1) | US6140321A (hu) |
JP (2) | JP2005015486A (hu) |
KR (1) | KR100545851B1 (hu) |
CN (1) | CN1312129C (hu) |
AT (1) | ATE445603T1 (hu) |
AU (1) | AU1153097A (hu) |
CA (1) | CA2516108C (hu) |
DE (1) | DE69739622D1 (hu) |
DK (1) | DK1211243T3 (hu) |
ES (1) | ES2330997T3 (hu) |
HK (1) | HK1080078A1 (hu) |
HU (1) | HUP0900417A3 (hu) |
PT (1) | PT1211243E (hu) |
SI (1) | SI22888B (hu) |
UA (1) | UA60307C2 (hu) |
WO (1) | WO1997046526A1 (hu) |
ZA (1) | ZA975064B (hu) |
Families Citing this family (92)
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JP2001517617A (ja) | 1997-09-24 | 2001-10-09 | ノヴァ モレキュラー インク. | 神経変性疾患の治療を目的としてapoeレベルを増加させる方法 |
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KR20040075371A (ko) * | 2002-02-07 | 2004-08-27 | 에-자이가부시기가이샤 | 발모 촉진제, 경피 적용 제제 및 발모 촉진 방법 |
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Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FI95572C (fi) * | 1987-06-22 | 1996-02-26 | Eisai Co Ltd | Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi |
-
1996
- 1996-12-27 WO PCT/JP1996/003881 patent/WO1997046526A1/en active Application Filing
- 1996-12-27 AU AU11530/97A patent/AU1153097A/en not_active Abandoned
- 1996-12-30 US US08/774,802 patent/US6140321A/en not_active Expired - Fee Related
-
1997
- 1997-06-06 ES ES02005248T patent/ES2330997T3/es not_active Expired - Lifetime
- 1997-06-06 HU HU0900417A patent/HUP0900417A3/hu unknown
- 1997-06-06 CN CNB200510075915XA patent/CN1312129C/zh not_active Expired - Fee Related
- 1997-06-06 PT PT02005248T patent/PT1211243E/pt unknown
- 1997-06-06 DE DE69739622T patent/DE69739622D1/de not_active Expired - Lifetime
- 1997-06-06 AT AT02005248T patent/ATE445603T1/de active
- 1997-06-06 UA UA99010107A patent/UA60307C2/uk unknown
- 1997-06-06 SI SI9720102A patent/SI22888B/sl not_active IP Right Cessation
- 1997-06-06 DK DK02005248.6T patent/DK1211243T3/da active
- 1997-06-06 CA CA002516108A patent/CA2516108C/en not_active Expired - Fee Related
- 1997-06-06 KR KR1020047017860A patent/KR100545851B1/ko not_active IP Right Cessation
- 1997-06-09 ZA ZA9705064A patent/ZA975064B/xx unknown
-
2004
- 2004-07-12 JP JP2004205012A patent/JP2005015486A/ja active Pending
-
2006
- 2006-01-04 HK HK06100124A patent/HK1080078A1/xx not_active IP Right Cessation
-
2008
- 2008-08-04 JP JP2008201060A patent/JP2009040783A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
DK1211243T3 (da) | 2010-02-08 |
KR20040104707A (ko) | 2004-12-10 |
ATE445603T1 (de) | 2009-10-15 |
HK1080078A1 (en) | 2006-04-21 |
PT1211243E (pt) | 2009-11-06 |
US6140321A (en) | 2000-10-31 |
ES2330997T3 (es) | 2009-12-18 |
JP2005015486A (ja) | 2005-01-20 |
SI22888B (sl) | 2010-06-30 |
CN1312129C (zh) | 2007-04-25 |
UA60307C2 (uk) | 2003-10-15 |
HU0900417D0 (en) | 2009-08-28 |
ZA975064B (en) | 1998-04-01 |
CA2516108A1 (en) | 1997-12-11 |
CA2516108C (en) | 2008-12-02 |
WO1997046526A1 (en) | 1997-12-11 |
CN1699343A (zh) | 2005-11-23 |
AU1153097A (en) | 1998-01-05 |
SI22888A (sl) | 2010-04-30 |
JP2009040783A (ja) | 2009-02-26 |
KR100545851B1 (ko) | 2006-01-24 |
DE69739622D1 (de) | 2009-11-26 |
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Legal Events
Date | Code | Title | Description |
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FD9A | Lapse of provisional protection due to non-payment of fees |