HUP0201673A3 - Process for the preparation of 4-[1-hydroxy-4-[4-(hydroxydiphenylmethyl)-1-piperidinyl]-butyl]-alpha, alpha-dimethylbenzeneacetic acid - Google Patents
Process for the preparation of 4-[1-hydroxy-4-[4-(hydroxydiphenylmethyl)-1-piperidinyl]-butyl]-alpha, alpha-dimethylbenzeneacetic acidInfo
- Publication number
- HUP0201673A3 HUP0201673A3 HU0201673A HUP0201673A HUP0201673A3 HU P0201673 A3 HUP0201673 A3 HU P0201673A3 HU 0201673 A HU0201673 A HU 0201673A HU P0201673 A HUP0201673 A HU P0201673A HU P0201673 A3 HUP0201673 A3 HU P0201673A3
- Authority
- HU
- Hungary
- Prior art keywords
- alpha
- hydroxydiphenylmethyl
- piperidinyl
- hydroxy
- butyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2001RM000260A ITRM20010260A1 (it) | 2001-05-17 | 2001-05-17 | Processo per la preparazione della fexofenadina o acido 4 1-idrossi-4-4- (idrossidifenilmetil)-1-piperidinil|-butil|-alfa,alfa-dimetilbenz |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| HU0201673D0 HU0201673D0 (https=) | 2002-07-29 |
| HUP0201673A2 HUP0201673A2 (hu) | 2003-02-28 |
| HUP0201673A3 true HUP0201673A3 (en) | 2004-07-28 |
Family
ID=11455529
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0201673A HUP0201673A3 (en) | 2001-05-17 | 2002-05-16 | Process for the preparation of 4-[1-hydroxy-4-[4-(hydroxydiphenylmethyl)-1-piperidinyl]-butyl]-alpha, alpha-dimethylbenzeneacetic acid |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US6815549B2 (https=) |
| EP (1) | EP1260505B1 (https=) |
| JP (1) | JP2003026658A (https=) |
| AT (1) | ATE290528T1 (https=) |
| CA (1) | CA2386452A1 (https=) |
| CZ (1) | CZ295949B6 (https=) |
| DE (1) | DE60203142T2 (https=) |
| ES (1) | ES2237631T3 (https=) |
| HU (1) | HUP0201673A3 (https=) |
| IT (1) | ITRM20010260A1 (https=) |
| PL (1) | PL353977A1 (https=) |
| PT (1) | PT1260505E (https=) |
| SI (1) | SI1260505T1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2239554T1 (es) * | 2002-06-10 | 2005-10-01 | Teva Pharmaceutical Industries Ltd. | Forma xvi polimorfica de hidrocloruro de fexofenadina. |
| EP1616861A3 (en) * | 2004-06-15 | 2006-02-08 | Dipharma S.p.A. | A process for the preparation of keto compounds |
| ITMI20041568A1 (it) * | 2004-07-30 | 2004-10-30 | Dipharma Spa | "polimorfi di fexofenadina base" |
| ITMI20061492A1 (it) * | 2006-07-27 | 2008-01-28 | Archimica Srl | Processo per la preparazione di fexofenadina. |
| ITMI20070987A1 (it) | 2007-05-16 | 2008-11-17 | Dipharma Francis Srl | Procedimento per la preparazione di composti chetonici |
| IT1395337B1 (it) * | 2009-03-04 | 2012-09-14 | Dipharma Francis Srl | Procedimento per la preparazione di intermedi chetonici |
| WO2011158262A1 (en) * | 2010-06-15 | 2011-12-22 | Chemelectiva S.R.L. | Polymorphic form of fexofenadine hydrochloride, intermediates and process for its preparation |
| CN102079708B (zh) * | 2011-02-11 | 2013-10-02 | 浙江启明药业有限公司 | 4-(4-卤丁酰基)-α,α-二甲基苯乙酸酯的合成方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2176201T3 (es) | 1992-04-10 | 2002-12-01 | Merrell Pharma Inc | Derivados de 4-difenilmetil piperidina y procedimiento de preparacion. |
| US6147216A (en) * | 1993-06-25 | 2000-11-14 | Merrell Pharmaceuticals Inc. | Intermediates useful for the preparation of antihistaminic piperidine derivatives |
| US6153754A (en) * | 1995-12-21 | 2000-11-28 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
| US6201124B1 (en) | 1995-12-21 | 2001-03-13 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
-
2001
- 2001-05-17 IT IT2001RM000260A patent/ITRM20010260A1/it unknown
-
2002
- 2002-05-15 CA CA002386452A patent/CA2386452A1/en not_active Abandoned
- 2002-05-16 PT PT02010234T patent/PT1260505E/pt unknown
- 2002-05-16 AT AT02010234T patent/ATE290528T1/de not_active IP Right Cessation
- 2002-05-16 US US10/145,765 patent/US6815549B2/en not_active Expired - Fee Related
- 2002-05-16 SI SI200230095T patent/SI1260505T1/xx unknown
- 2002-05-16 ES ES02010234T patent/ES2237631T3/es not_active Expired - Lifetime
- 2002-05-16 EP EP02010234A patent/EP1260505B1/en not_active Expired - Lifetime
- 2002-05-16 DE DE60203142T patent/DE60203142T2/de not_active Expired - Fee Related
- 2002-05-16 HU HU0201673A patent/HUP0201673A3/hu unknown
- 2002-05-17 PL PL02353977A patent/PL353977A1/xx not_active Application Discontinuation
- 2002-05-17 JP JP2002143142A patent/JP2003026658A/ja not_active Ceased
- 2002-05-17 CZ CZ20021726A patent/CZ295949B6/cs not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ITRM20010260A0 (it) | 2001-05-17 |
| EP1260505A1 (en) | 2002-11-27 |
| HUP0201673A2 (hu) | 2003-02-28 |
| SI1260505T1 (en) | 2005-06-30 |
| US20020198233A1 (en) | 2002-12-26 |
| DE60203142D1 (de) | 2005-04-14 |
| CA2386452A1 (en) | 2002-11-17 |
| ATE290528T1 (de) | 2005-03-15 |
| CZ20021726A3 (cs) | 2003-01-15 |
| ITRM20010260A1 (it) | 2002-11-18 |
| DE60203142T2 (de) | 2006-04-13 |
| PT1260505E (pt) | 2005-05-31 |
| PL353977A1 (en) | 2002-11-18 |
| EP1260505B1 (en) | 2005-03-09 |
| ES2237631T3 (es) | 2005-08-01 |
| HU0201673D0 (https=) | 2002-07-29 |
| US6815549B2 (en) | 2004-11-09 |
| JP2003026658A (ja) | 2003-01-29 |
| CZ295949B6 (cs) | 2005-12-14 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL160060A0 (en) | Piperidine derivatives useful as ccr5 antagonists | |
| PL348417A1 (en) | 4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders | |
| IL157551A0 (en) | Ccr5 antagonists useful for treating aids | |
| HUP0201673A3 (en) | Process for the preparation of 4-[1-hydroxy-4-[4-(hydroxydiphenylmethyl)-1-piperidinyl]-butyl]-alpha, alpha-dimethylbenzeneacetic acid | |
| IL189986A0 (en) | Process for producing 1-benzyl-4-[(5,6-dimethoxy-1-indanon)-2-yl]methylpiperidine or hydrochloride thereof | |
| PL1761492T3 (pl) | Szczawian 1-benzylo-4-[(5,6-dimetoksy-1-indanon)-2-ylo]metylopiperydyny (szczawian donepezilu) i jego polimorfy | |
| WO2001094313A3 (en) | Crystal modification of fexofenadine | |
| AU2001247848A1 (en) | Process for the preparation of 1,5-dideoxy-1,5-imino hexitols from oximes or imines | |
| ZA200309557B (en) | Novel crystalline forms of 4-[4-[4-(hydroxydiphenylmethy)-1-piperindinyl]-1-hydroxybutyl]-alpha, alpha-dimethylbenzene acetic acid and its hydrochloride. | |
| NO20035572D0 (no) | Fremgangsmåte til fremstilling av piperidinderivatet fexofenadin | |
| IL157709A0 (en) | Process for the preparation of 1,2-benzisoxazole-3-acetic acid | |
| HU9800511D0 (en) | Process for producing 4-{4-[4-(hydroxy-diphenyl)-1-piperidinyl]-1-hydroxy-butyl}-alpha-alpha-dimethyl-phenyl-acetic.acid and phosphorylized derivatives thereof | |
| IL188916A0 (en) | Process for producing 1-benzyl-4-[(5,6-dimethoxy-1-indanone)-2-ylidene]methylpiperidine | |
| IL178766A0 (en) | Processes for producing 1 - benzyl - 4 - [(5, 6 - dimethoxy - 1indanon) - 2 - yl] methylpiperidine and hydrochloride thereof | |
| IL152570A0 (en) | A process for the preparation of 4-[1-hydroxy-4-[4-(hydroxydiphenylmethyl)-1-piperidinyl]-alpha, alpha-di methylbenzeneacetic acid | |
| EP1616861A3 (en) | A process for the preparation of keto compounds | |
| EP1316549A4 (en) | 1-BENZYL-4 - [(5,6-DIMETHOXY-2-FLUORO-1-INDANONE) -2-YL] METHYLPIPERIDIN | |
| SE0102809D0 (sv) | Novel compounds | |
| AU3818900A (en) | Process for the preparation of substituted piperidines | |
| WO2007049303A3 (en) | An improved process for the preparation of highly pure fexofenadine | |
| ITMI20011772A0 (it) | Processo per la preparazione della 2,5-bis-(2,2,2-trifluoroetossi)-n-(2-piperidilmetil)-benzamide(flecainide) | |
| HUP0402390A3 (en) | Process for the preparation of 4-(8-chloro-5,6-dihydro-11h-benzo(5,6)-cyclohepta-(1,2-b)-pyridin-11-ylidene)-1-piperidinecarboxylic acid ethyl ester (loratadine) and the intermediates | |
| HUP0302866A3 (en) | 3-(3-amidinophenyl)-5-[({[1-(1-iminoethyl)-4-piperidyl}amino)methyl]benzoic acid dihydrochloride and process for preparing the same | |
| EP1841739B8 (en) | Process for producing 1-benzyl-4-[(5,6-dimethoxy-1-indanon-2-yl)methyl] piperidine or salt thereof via novel intermediate | |
| AU2002223617A1 (en) | Novel neurokinin antagonists, method for the production thereof and pharmaceutical compositions containing said compounds |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD9A | Lapse of provisional protection due to non-payment of fees |