HUP0005004A2 - Eljárás szulfonil-amino-karbonil-triazolinon-sók előállítására - Google Patents

Eljárás szulfonil-amino-karbonil-triazolinon-sók előállítására

Info

Publication number
HUP0005004A2
HUP0005004A2 HU0005004A HUP0005004A HUP0005004A2 HU P0005004 A2 HUP0005004 A2 HU P0005004A2 HU 0005004 A HU0005004 A HU 0005004A HU P0005004 A HUP0005004 A HU P0005004A HU P0005004 A2 HUP0005004 A2 HU P0005004A2
Authority
HU
Hungary
Prior art keywords
alkyl
aryl
formula
salts
substituted
Prior art date
Application number
HU0005004A
Other languages
English (en)
Inventor
Vijay C. Desai
Klaus Jelich
Shekhar V. Kulkarni
Vidyanatha A. Prasad
Eric Rivadeneira
Original Assignee
Bayer Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/472,335 external-priority patent/US6147221A/en
Priority claimed from US09/472,672 external-priority patent/US6147222A/en
Application filed by Bayer Corporation filed Critical Bayer Corporation
Publication of HU0005004D0 publication Critical patent/HU0005004D0/hu
Publication of HUP0005004A2 publication Critical patent/HUP0005004A2/hu
Publication of HUP0005004A3 publication Critical patent/HUP0005004A3/hu
Publication of HU229877B1 publication Critical patent/HU229877B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/12—Oxygen or sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

A találmány tárgya eljárás szulfonil-amino-karbonil-triazolinon-sókelőállítására oly módon, hogy a) egy (I) általános képletűszubsztituált triazolinon vegyületet - a képletben R1 és R2mindegyikének jelentése szubsztituált vagy szubsztituálatlan alkil-,alkenil-, alkinil-, cikloalkil-, cikloalkil-alkil-, aril- vagy aril-alkil-csoport - reagáltatnak egy (II) általános képletű szulfonil-izocianáttal - a képletben R3 jelentése szubsztituálatlan vagyszubsztituált alkil-, aril-, aril-alkil- vagy heteroarilcsoport - , b)a kapott szulfonil-amino-karbonil-triazolinin intermedier egyegyedényes eljárásban (az intermedier termék izolálása vagyelválasztása nélkül) egy bázissal reagáltatják, így nyerik a (IV)általános képletű sót - a képletben R1, R2 és R3 jelentése a fenti ésM jelentése egy alkáli- vagy alkáliföldfém vagy egy protonált ammónia-származék. Ó
HU0005004A 1999-12-27 2000-12-22 Process for the manufacture of the salts of sulfonylaminocarbonyl triazolinone compounds HU229877B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/472,335 US6147221A (en) 1999-12-27 1999-12-27 Process for the manufacture of sulfonylaminocarbonyl triazolinones and salts thereof
US09/472,672 US6147222A (en) 1999-12-27 1999-12-27 Process for the manufacture of sulfonylaminocarbonyl triazolinones and salts thereof under pH controlled conditions

Publications (4)

Publication Number Publication Date
HU0005004D0 HU0005004D0 (en) 2001-03-28
HUP0005004A2 true HUP0005004A2 (hu) 2001-11-28
HUP0005004A3 HUP0005004A3 (en) 2002-12-28
HU229877B1 HU229877B1 (en) 2014-11-28

Family

ID=27043734

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0005004A HU229877B1 (en) 1999-12-27 2000-12-22 Process for the manufacture of the salts of sulfonylaminocarbonyl triazolinone compounds

Country Status (15)

Country Link
EP (1) EP1113009B1 (hu)
JP (1) JP4846092B2 (hu)
KR (1) KR100704718B1 (hu)
CN (1) CN1179953C (hu)
AR (1) AR027120A1 (hu)
AT (1) ATE292122T1 (hu)
BR (1) BR0006287B1 (hu)
DE (1) DE60019075T2 (hu)
DK (1) DK1113009T3 (hu)
ES (1) ES2238964T3 (hu)
HK (1) HK1038015A1 (hu)
HU (1) HU229877B1 (hu)
IL (1) IL140521A (hu)
IN (1) IN189996B (hu)
TW (1) TWI280243B (hu)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR037097A1 (es) 2001-10-05 2004-10-20 Novartis Ag Compuestos acilsulfonamidas, composiciones farmaceuticas y el uso de dichos compuestos para la preparacion de un medicamento
CN103265499B (zh) * 2013-06-04 2014-10-22 江苏省农用激素工程技术研究中心有限公司 5-甲氧基-4-甲基-2,4-二氢-3h-1,2,4-三唑-3-酮的精制方法
CN103936684B (zh) * 2014-04-30 2016-10-05 江苏省农用激素工程技术研究中心有限公司 磺酰胺基羰基三唑啉酮化合物及其制备方法和应用
US10238112B1 (en) * 2018-01-24 2019-03-26 Arysta Lifescience Inc. Flucarbazone sodium hemihydrate method and composition
CN114929677A (zh) * 2019-12-30 2022-08-19 江苏龙灯化学有限公司 氟酮磺隆钠新晶型

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3934081A1 (de) * 1989-10-12 1991-04-18 Bayer Ag Sulfonylaminocarbonyltriazolinone
US5599944A (en) * 1987-03-24 1997-02-04 Bayer Aktiengesellschaft Intermediates for herbicidal sulphonylaminocarbonyltriazolinones having substituents which are bonded via sulphur
DE4110795A1 (de) * 1991-04-04 1992-10-08 Bayer Ag Sulfonylaminocarbonyltriazolinone mit ueber sauerstoff gebundenen substituenten
US5241074A (en) * 1988-05-09 1993-08-31 Bayer Aktiengesellschaft Sulphonylaminocarbonyltriazolinones
US5534486A (en) * 1991-04-04 1996-07-09 Bayer Aktiengesellschaft Herbicidal sulphonylaminocarbonyl triazolinones having substituents bonded via oxygen
US6147221A (en) * 1999-12-27 2000-11-14 Bayer Corporation Process for the manufacture of sulfonylaminocarbonyl triazolinones and salts thereof
US6147222A (en) * 1999-12-27 2000-11-14 Bayer Corporation Process for the manufacture of sulfonylaminocarbonyl triazolinones and salts thereof under pH controlled conditions
US6160125A (en) * 1999-12-27 2000-12-12 Bayer Corporation Process for the manufacture of sulfonylaminocarbonyl triazolinones in the presence of xylene as solvent

Also Published As

Publication number Publication date
ATE292122T1 (de) 2005-04-15
HU229877B1 (en) 2014-11-28
CN1179953C (zh) 2004-12-15
DK1113009T3 (da) 2005-06-27
KR100704718B1 (ko) 2007-04-09
IL140521A (en) 2005-12-18
IN189996B (hu) 2003-05-31
HU0005004D0 (en) 2001-03-28
IL140521A0 (en) 2002-02-10
CN1301696A (zh) 2001-07-04
JP4846092B2 (ja) 2011-12-28
BR0006287A (pt) 2002-01-02
DE60019075T2 (de) 2006-04-27
EP1113009B1 (en) 2005-03-30
HUP0005004A3 (en) 2002-12-28
EP1113009A1 (en) 2001-07-04
DE60019075D1 (de) 2005-05-04
AR027120A1 (es) 2003-03-12
BR0006287B1 (pt) 2010-11-30
HK1038015A1 (en) 2002-03-01
ES2238964T3 (es) 2005-09-16
KR20010062193A (ko) 2001-07-07
JP2001206878A (ja) 2001-07-31
TWI280243B (en) 2007-05-01

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