HRP20190728T1 - Derivati aminobenzamida kao učinkovita sredstva za kontrolu životinjskih parazita - Google Patents

Derivati aminobenzamida kao učinkovita sredstva za kontrolu životinjskih parazita Download PDF

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HRP20190728T1
HRP20190728T1 HRP20190728TT HRP20190728T HRP20190728T1 HR P20190728 T1 HRP20190728 T1 HR P20190728T1 HR P20190728T T HRP20190728T T HR P20190728TT HR P20190728 T HRP20190728 T HR P20190728T HR P20190728 T1 HRP20190728 T1 HR P20190728T1
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haloalkyl
alkoxy
haloalkylthio
alkylthio
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HRP20190728TT
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Ulrich Görgens
Akihiko Yanagi
Katsuaki Wada
Tetsuya Murata
Yukiyoshi Watanabe
Jun Mihara
Koichi Araki
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Bayer Cropscience Ag
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Claims (3)

1. Derivat aminobenzamida formule (I-1), ili njegova sol pri čemu X predstavlja vodikov atom, halogeni atom, hidroksi skupinu, skupinu C1-C6 alkil ili skupinu trifluorometil; R1 predstavlja vodikov atom, C1-C6 alkil skupinu C1-C6 haloalkil skupinu, C1-C6 alkoksi skupinu, C1-C6 haloalkoksi skupinu, C1-C6 alkiltio skupinu, C1-C6 haloalkiltio skupinu, C1-C6 alkilkarbonil skupinu, C1-C6 haloalkilkarbonil skupinu ili predstavlja fenil ili benzil po izboru supstituiran s najmanje jednom skupinom odabranom iz skupine koja sadrži C1-C6 alkil, C1-C6 alkoksi, C1-C6 alkiltio, C1-C6 alkilsulfinil, C1-C6 alkilsulfonil, C1-C6 haloalkil, C1-C6 haloalkoksi, C1-C6 haloalkiltio, C1-C6 haloalkilsulfinil, C1-C6 haloalkilsulfonil, nitro, hidroksi, i halogen; ili piridil, pirazolil, tienil, furil, izoksazolil, tiadiazolil ili piridilmetil, pirazolilmetil, tienilmetil, furilmetil, izoksazolilmetil, ili tiadiazolilmetil po izboru supstituiranu s najmanje jednom skupinom odabranom iz skupine koja sadrži C1-C6 alkil, C1-C6 alkoksi, C1-C6 alkiltio, C1-C6 alkilsulfinil, C1-C6 alkilsulfonil, C1-C6 haloalkil, C1-C6 haloalkoksi, C1-C6 haloalkiltio, C1-C6 haloalkilsulfinil, C1-C6 haloalkilsulfonil, nitro, hidroksi, i halogen R3 i R5 predstavljaju međusobno neovisno halogeni atom, skupinu C1-C4 alkil, skupinu C1-C4 haloalkil, skupinu C1-C4 alkoksi, skupinu C1-C4 haloalkoksi, skupinu C1-C3 alkiltio, skupinu C1-C3 haloalkiltio, skupinu C1-C3 alkilsulfinil, skupinu C1-C3 haloalkilsulfinil, skupinu C1-C3 alkilsulfonil, skupinu C1-C3 haloalkilsulfonil ili cijano skupinu; R4 predstavlja skupinu C1-C4 alkil, skupinu C1-C4 haloalkil, skupinu C1-C4 haloalkil C1-C4 alkoksi, skupinu C1-C4 haloalkil C1-C4 haloalkoksi, skupinu C1-C4 alkoksi, skupinu C1-C4 haloalkoksi, skupinu C1-C3 alkiltio, skupinu C1-C3 haloalkiltio, skupinu C1-C3 alkilsulfinil, skupinu C1-C3 haloalkilsulfinil, skupinu C1-C3 alkilsulfonil, skupinu C1-C3 haloalkilsulfonil ili skupinu SF5; L predstavlja fenilnu skupinu, ili supstituiranu fenilnu skupinu koja ima jedan ili više supstituenata koji mogu biti isti ili različiti i koji su odabrani iz niza koji sadrži halogeni atom, skupinu C1-C4 alkil, skupinu C1-C4 haloalkil, skupinu C2-C4 alkenil, skupinu C2-C4 haloalkenil, skupinu C2-C4 alkinil, skupinu C2-C4 haloalkinil, skupinu C3-C6 cikloalkil, skupinu C3-C6 halocikloalkil, skupinu C1-C3 alkoksi, skupinu C1-C3 haloalkoksi, skupinu C1-C3 alkiltio, skupinu C1-C3 haloalkiltio, skupinu C1-C3 alkilsulfinil, skupinu C1-C3 haloalkilsulfinil, skupinu C1-C3 alkilsulfonil, skupinu C1-C3 haloalkilsulfonil, skupinu C1-C4 alkilamino, skupinu di- C1-C4 alkilamino, cijano skupinu, nitro skupinu, hidroksi skupinu, C1-C4 alkilkarbonil skupinu, skupinu C1-C4 alkilkarboniloksi, skupinu C1-C4 alkoksikarbonil, acetilamino skupinu i fenilnu skupinu; ili piridil skupinu; ili piridil skupinu koja ima jedan ili više supstituenata koji mogu biti isti ili različiti i koji su odabrani iz niza koji sadrži halogeni atom, skupinu C1-C4 alkil, skupinu C1-C4 haloalkil, skupinu C2-C4 alkenil, skupinu C2-C4 haloalkenil, skupinu C2-C4 alkinil, skupinu C2-C4 haloalkinil, skupinu C3-C6 cikloalkil, skupinu C3-C6 halocikloalkil, skupinu C1-C3 alkoksi, skupinu C1-C3 haloalkoksi, skupinu C1-C3 alkiltio, skupinu C1-C3 haloalkiltio, skupinu C1-C3 alkilsulfinil, skupinu C1-C3 haloalkilsulfinil, skupinu C1-C3 alkilsulfonil, skupinu C1-C3 haloalkilsulfonil, skupinu C1-C4 alkilamino, skupinu di-C1-C4 alkilamino, cijano skupinu, nitro skupinu, hidroksi skupinu, skupinu C1-C4 alkilkarbonil, skupinu C1-C4 alkilkarboniloksi, skupinu C1-C4 alkoksikarbonil, acetilamino skupinu i fenilnu skupinu; ili vodik, skupinu C1-C4 alkil, skupinu C1-C4 haloalkil, skupinu C2-C4 alkenil, skupinu C2-C4 haloalkenil, skupinu C2-C4 alkinil, skupinu C2-C4 haloalkinil, skupinu C3-C6 cikloalkil, skupinu C3-C6 halocikloalkil, skupinu C1-C3 alkoksi, skupinu C1-C3 haloalkoksi, skupinu C1-C3 alkiltio, skupinu C1-C3 haloalkiltio, skupinu C1-C3 alkilsulfinil, skupinu C1-C3 haloalkilsulfinil, skupinu C1-C3 alkilsulfonil i skupinu C1-C3 haloalkilsulfonil; ili skupinu C1-C4 alkil, skupinu C1-C4 haloalkil, skupinu C2-C4 alkenil, skupinu C2-C4 haloalkenil, skupinu C2-C4 alkinil, skupinu C2-C4 haloalkinil, skupinu C3-C6 cikloalkil, skupinu C3-C6 halocikloalkil, skupinu C1-C3 alkoksi, skupinu C1-C3 haloalkoksi, skupinu C1-C3 alkiltio, skupinu C1-C3 haloalkiltio, skupinu C1-C3 alkilsulfinil, skupinu C1-C3 haloalkilsulfinil, skupinu C1-C3 alkilsulfonil i skupinu C1-C3 haloalkilsulfonil, svaku supstituiranu s fenilnom skupinom koja ima jedan ili više supstituenata koji mogu biti isti ili različiti i koji su odabrani iz niza koji sadrži halogeni atom, skupinu C1-C4 alkil, skupinu C1-C4 haloalkil, skupinu C2-C4 alkenil, skupinu C2-C4 haloalkenil, skupinu C2-C4 alkinil, skupinu C2-C4 haloalkinil, skupinu C3-C6 cikloalkil, skupinu C3-C6 halocikloalkil, skupinu C1-C3 alkoksi, skupinu C1-C3 haloalkoksi, skupinu C1-C3 alkiltio, skupinu C1-C3 haloalkiltio, skupinu C1-C3 alkilsulfinil, skupinu C1-C3 haloalkilsulfinil, skupinu C1-C3 alkilsulfonil, skupinu C1-C3 haloalkilsulfonil, skupinu C1-C4 alkilamino, skupinu di-C1-C4 alkilamino, cijano skupinu, nitro skupinu, hidroksi skupinu, skupinu C1-C4 alkilkarbonil, skupinu C1-C4 alkilkarboniloksi, skupinu C1-C4 alkoksikarbonil, acetilamino skupinu i fenilnu skupinu; ili piridil skupinu; naznačen time što se upotrebljava za kontrolu krpelja odabranih iz skupine koja sadrži Amblyomma americanum, Dermacentor variabilis, Dermacentor reticulatus, i Rhipicephalus sanguineus.
2. Farmaceutski pripravak koji sadrži najmanje jedan derivat aminobenzamida prema zahtjevu 1 naznačen time što se upotrebljava za sprječavanje infekcije s bolestima koje se prenose parazitima.
3. Derivat aminobenzamida prema zahtjevu 1 naznačen time što se koristi za sprječavanje infekcije s bolestima koje se prenose putem krpelja odabranih iz skupine koju čine Amblyomma americanum, Dermacentor variabilis, Dermacentor reticulatus, i Rhipicephalus sanguineus.
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