AR069764A1 - Derivados de aminobenzamida como agentes utiles para controlar parasitos animales - Google Patents

Derivados de aminobenzamida como agentes utiles para controlar parasitos animales

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Publication number
AR069764A1
AR069764A1 ARP080105445A ARP080105445A AR069764A1 AR 069764 A1 AR069764 A1 AR 069764A1 AR P080105445 A ARP080105445 A AR P080105445A AR P080105445 A ARP080105445 A AR P080105445A AR 069764 A1 AR069764 A1 AR 069764A1
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Argentina
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group
alkyl
halo
thio
haloalkyl
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ARP080105445A
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Bayer Cropscience Ag
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    • C07C237/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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    • C07C271/06—Esters of carbamic acids
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    • C07C271/26—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring
    • C07C271/28—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring to a carbon atom of a non-condensed six-membered aromatic ring
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Abstract

Composiciones farmacéuticas veterinarias que comprenden al menos una aminobenzamida de formula (1) para prevenir la infeccion con enfermedades transmitidas a través de parásitos, a su uso para la preparacion de una composicion farmacéutica veterinaria para controlar parásitos animales y a un procedimiento para prevenir la infeccion con enfermedades transmitidas a través de parásitos. Reivindicacion 1: Derivado de aminobenzamida de formula (1), o una de sus sales en la que A1, A2, A3 y A4 representan cada uno independientemente uno del otro C-X, N o N=O; X representa independientemente uno del otro un átomo de hidrogeno, un átomo de halogeno, un grupo hidroxi, un grupo alquilo C1-6 o un grupo trifluorometilo; B1 y B2 representan cada uno independientemente uno del otro un átomo de oxigeno o un átomo de azufre; R1 y R2 respectivamente representan independientemente uno del otro un átomo de hidrogeno, un grupo alquilo C1-6 , un grupo haloalquilo C1-6 , un grupo alcoxi C1-6 , un grupo haloalcoxi C1-6 , un grupo (alquil C1-6)tio, un grupo halo(alquil C1-6)tio, un grupo (alquil C1-6)carbonilo, un grupo halo(alquil C1-6)carbonilo; o representa un grupo fenilo o un grupo bencilo opcionalmente sustituido con al menos un grupo seleccionado del grupo constituido por alquilo C1-6, alcoxi C1-6, (alquil C1-6)tio, (alquil C1-6)sulfinilo, (alquil C1-6)sulfonilo, haloalquilo C1-6, haloalcoxi C1-6, halo(alquil C1-6)tio, halo(alquil C1-6)sulfinilo, halo(alquil C1-6)sulfonilo, nitro, hidroxi, y halogeno; o piridilo, pirazolilo, tienilo, furilo, isoxazolilo, tiadiazolilo o piridilmetilo, pirazolilmetilo, tienilmetilo, furilmetilo, isoxazolilmetiIo, o tiadiazolilmetilo opcionalmente sustituido con al menos un grupo seleccionado del grupo constituido por alquilo C1-6, alcoxi C1-6, (alquil C1-6)tio, (alquil C1-6)sulfinilo, (alquil C1-6)sulfonilo, haloalquilo C1-6, haloalcoxi C1-6, halo(alquil C1-6)tio, halo(alquil C1-6)sulfinilo, halo(alquil C1-6)sulfonilo, nitro, hidroxi, y halogeno; Q representa L o Y-R6 con Y representando oxígeno, azufre, amino, aminoalquilo C1-4; y R6 representando un grupo alquilo C1-6, un grupo haloalquilo C1-6, un grupo alquenilo C2-6, un grupo haloalquenilo C2-6, un grupo alquinilo C2-6, un grupo haloalquinilo C2-6, un grupo cicloalquilo C3-8 o un grupo halocicloalquilo C3-8; o -E1-Z1-R7 (donde E1 representa un grupo alquileno C1-4, un grupo alquenileno C2-4, un grupo alquinileno C3-4, un grupo haloalquileno C1-4, un grupo haloalquenileno C2-4 o un grupo haloalquinileno C3-4, R7 representa un átomo de hidrogeno, un grupo alquilo C1-6, un grupo alquenilo C2-6, un grupo alquinilo C2-6, un grupo haloalquilo C1-6, un grupo haloalquenilo C2-6 o un grupo haloalquinilo C2-6, y Z1 representa -O-, -S-, -SO-, -SO2, -C(=O)-, -C(=O)O-, -OC(=O)-, -N(R8)-, -C(=O)N(R8)- o - N(R8)C(=O)-); o -E2-R9 (donde E2 representa un grupo alquileno C1-4, un grupo alquenileno C2-4, un grupo alquinileno C3-4, un grupo haloalquileno C1-4, un grupo haloalquenileno C2-4 o un grupo haloalquinileno C3-4 y R9 representa un grupo cicloalquilo C3-8, un grupo halocicloalquilo C3-8, un grupo ciano, un grupo nitro, un grupo hidroxi, un grupo fenilo, o un grupo fenilo sustituido que tiene uno o más sustituyentes que pueden ser iguales o distintos y que se seleccionan de un átomo de halogeno, un grupo alquilo C1-6, un grupo haloalquilo C1-6, un grupo alcoxi C1-6, un grupo haloalcoxi C1-6, un grupo (alquil C1-6)tio, un grupo halo(alquil C1-6)tio, un grupo (alquil C1-6)sulfinilo, un grupo halo(alquil C1-6)sulfinilo, un grupo (alquil C1-6)sulfonilo, un grupo halo(alquil C1-6)sulfonilo, un grupo ciano, un grupo nitro, un grupo hidroxi, un grupo (alquil C1-4)carbonilo, un grupo halo(alquil C1-4)carbonilo, un grupo (alquil C1-4)carboniloxi y un grupo (alcoxi C1-4)carbonilo, o un grupo piridilo, o un grupo piridilo sustituido que tiene uno o más sustituyentes que se seleccionan de un átomo de halogeno, un grupo haloalquilo C1-6 y un grupo haloalcoxi C1-6, un grupo tienilo o un grupo tetrahidrofurano); L representa un grupo fenilo; o un grupo heterociclilo; o hidrogeno, un grupo alquilo C1-6, un grupo alquenilo C2-6, un grupo alquinilo C2-6, un grupo cicloalquilo C3-8, un grupo cicloalquenilo C3-8, un grupo aldehído C1-6 , un grupo iminoaldehído C1-6, un grupo alcoxiiminoaldehído C1-6, un grupo alcoxiimino C1-6-alquilo C1-6, un grupo alcoxi C1-6, un grupo (alquil C1-6)tio, un grupo halo(alquil C1-6)tio, un grupo (alquil C1-6)sulfinilo, y un grupo (alquil C1-6)sulfonilo; donde cada uno de los restos anteriormente citados está opcionalmente sustituido con un átomo de halogeno, un grupo alquilo C1-4, un grupo haloalquilo C1-4, un grupo alquenilo C2-4, un grupo haloalquenilo C2-4, un grupo alquinilo C2-4, un grupo haloalquinilo C2-4, un grupo cicloalquilo C3-6, un grupo halocicloalquilo C3-6, un grupo alcoxi C1-3, un grupo haloalcoxi C1-3, un grupo (alquil C1-3)tio, un grupo halo(alquil C1-3)tio, un grupo (alquil C1-3)sulfinilo, un grupo halo(alquil C1-3)sulfinilo, un grupo (alquil C1-3)sulfonilo, un grupo halo(alquil C1-3)sulfonilo, un grupo (alquil C1-4)amino, un grupo di(alquil C1-4)amino, un grupo ciano, un grupo nitro, un grupo hidroxi, un grupo (alquil C1-4)carbonilo, un grupo (alquil C1-4)carboniloxi, un grupo (alcoxi C1-4)carbonilo, un grupo acetilamino, un grupo fenilo, y un grupo piridilo; W representa un grupo fenilo, o un grupo fenilo sustituido que tiene uno o más sustituyentes que pueden ser iguales o distintos y que se seleccionan de un átomo de halogeno, un grupo alquilo C1-4, un grupo haloalquilo C1-4, grupo haloalquilo C1-4-alcoxi C1-4, grupo haloalquilo C1-4-haloalcoxi C1-4, un grupo alcoxi C1-4, un grupo haloalcoxi C1-4, un grupo (alquil C1-3)tio, un grupo halo(alquil C1-3)tio, un grupo (alquil C1-3)sulfinilo, un grupo halo(alquil C1-3)sulfinilo, un grupo (alquil C1-3)sulfonilo, un grupo halo(alquil C1-3)sulfonilo, un grupo ciano, un grupo carbonilalquilo C1-4, un grupo carboni-haloalquilo C1-4: o un grupo SF5 para prevenir la infeccion con enfermedades transmitidas a través de parásitos.
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