HRP20120138T1 - Energetski dodatak prehrani za skeletne mišiće i za zaštitu kardiovaskularnog sustava - Google Patents

Energetski dodatak prehrani za skeletne mišiće i za zaštitu kardiovaskularnog sustava Download PDF

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HRP20120138T1
HRP20120138T1 HRP20120138TT HRP20120138T HRP20120138T1 HR P20120138 T1 HRP20120138 T1 HR P20120138T1 HR P20120138T T HRP20120138T T HR P20120138TT HR P20120138 T HRP20120138 T HR P20120138T HR P20120138 T1 HRP20120138 T1 HR P20120138T1
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carnitine
dietary supplement
acid
group
mixtures
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HRP20120138TT
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Gaetani Franco
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Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.
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Publication of HRP20120138T1 publication Critical patent/HRP20120138T1/hr

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/525Isoalloxazines, e.g. riboflavins, vitamin B2
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23LFOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L33/00Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
    • A23L33/10Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23LFOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L33/00Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
    • A23L33/10Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
    • A23L33/15Vitamins
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23LFOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L33/00Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
    • A23L33/10Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
    • A23L33/17Amino acids, peptides or proteins
    • A23L33/175Amino acids
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23PSHAPING OR WORKING OF FOODSTUFFS, NOT FULLY COVERED BY A SINGLE OTHER SUBCLASS
    • A23P10/00Shaping or working of foodstuffs characterised by the products
    • A23P10/40Shaping or working of foodstuffs characterised by the products free-flowing powder or instant powder, i.e. powder which is reconstituted rapidly when liquid is added
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/205Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23VINDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
    • A23V2002/00Food compositions, function of food ingredients or processes for food or foodstuffs

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Polymers & Plastics (AREA)
  • Food Science & Technology (AREA)
  • Epidemiology (AREA)
  • Nutrition Science (AREA)
  • Mycology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Dodatak prehrani, naznačen time što sadrži:- kao aktivne sastojke, kombinaciju pomiješanih ili odvojeno pakiranih: a) propionil-1-karnitina ili njegove farmakološki prihvatljive soli i izborno karnitin, kojeg se bira iz skupine koju čine L-karnitin, acetil-1-karnitin, valeril-1-karnitin, izovaleril-1-karnitin i butiril-1-karnitin, ili njihove farmakološki prihvatljive soli ili njihove smjese; b) koenzim Q10;c) riboflavin; d) pantotenska kiselina; i- slijedeće izborne komponente: f) aminokiselina, koju se bira iz skupine koju čine valin, leucin, izoleucin ili njihove smjese; g) kreatin, kojeg se bira iz skupine koju čine kreatin i fosfokreatin ili njihove smjese; ih) mineralna sol. Patent sadrži još 8 patentnih zahtjeva.

Claims (9)

1. Dodatak prehrani, naznačen time što sadrži: – kao aktivne sastojke, kombinaciju pomiješanih ili odvojeno pakiranih: a) propionil-1-karnitina ili njegove farmakološki prihvatljive soli i izborno karnitin, kojeg se bira iz skupine koju čine l-karnitin, acetil-1-karnitin, valeril-1-karnitin, izovaleril-1-karnitin i butiril-1-karnitin, ili njihove farmakološki prihvatljive soli ili njihove smjese; b) koenzim Q10; c) riboflavin; d) pantotenska kiselina; i – slijedeće izborne komponente: f) aminokiselina, koju se bira iz skupine koju čine valin, leucin, izoleucin ili njihove smjese; g) kreatin, kojeg se bira iz skupine koju čine kreatin i fosfokreatin ili njihove smjese; i h) mineralna sol.
2. Dodatak prehrani u skladu s patentnim zahtjevom 1, naznačen time što se farmakološki prihvatljivu sol bira iz skupine koju čine: klorid; bromid; jodid; aspartat, kiseli aspartat; citrat, kiseli citrat; fosfat, kiseli fosfat; fumarat, kiseli fumarat; glicerofosfat; glukozni fosfat; laktat; maleat, kiseli maleat; mukat; orotat; oksalat; kiseli oksalat; sulfat, kiseli sulfat; tartarat; trikloracetat; trifluoracetat i metansulfonat.
3. Dodatak prehrani u skladu s patentnim zahtjevom 1, naznačen time što se mineralnu sol (h) bira iz skupine koju čine: dinatrijev citrat, monokalijev fosfat, kalcijev laktat i magnezijev taurat.
4. Dodatak prehrani u skladu s patentnim zahtjevom 1, naznačen time što se težinski omjer (a):(b):(c):(d) kreće od 10:0,04:0,08:0,4 to 1:4:4:20.
5. Dodatak prehrani u skladu s patentnim zahtjevom 4, naznačen time što se težinski omjer (a):(b):(c):(d) kreće od 10:2:2:2 do 1:1:1:5.
6. Dodatak prehrani u skladu s patentnim zahtjevom 1, naznačen time što je u obliku tableta, lozengeta, pilula, kapsula i granulata.
7. Dodatak prehrani u skladu s patentnim zahtjevom 6, koji je u obliku jedinice doziranja, naznačen time što sadrži: propionil-1-karnitin 50 mg do 2.000 mg koenzim Q10 5 mg do 200 mg riboflavin 5 mg do 200 mg pantotenska kiselina 10 mg do 1.000 mg.
8. Postupak povećavanja sposobnosti skeletnih mišića da održavaju dulje periode intenzivne fizičke aktivnosti, naznačen time što se sastoji u primjeni dodatka prehrani u skladu s bilo kojim od patentnih zahtjeva 1 do 7.
9. Postupak osiguravanja energije i jačanja skeletnih mišića, naznačen time što se sastoji u primjeni dodatka prehrani u skladu s bilo kojim od patentnih zahtjeva 1 do 7.
HRP20120138TT 2005-10-20 2012-02-10 Energetski dodatak prehrani za skeletne mišiće i za zaštitu kardiovaskularnog sustava HRP20120138T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11/253,806 US8252309B2 (en) 2000-04-04 2005-10-20 Dietary supplement energy-providing to skeletal muscles
PCT/EP2006/066538 WO2007045533A1 (en) 2005-10-20 2006-09-20 Dietary supplement energy-providing to skeletal muscles and protecting the cardio vascular tract

Publications (1)

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HRP20120138T1 true HRP20120138T1 (hr) 2012-05-31

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HRP20120138TT HRP20120138T1 (hr) 2005-10-20 2012-02-10 Energetski dodatak prehrani za skeletne mišiće i za zaštitu kardiovaskularnog sustava

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US (2) US8252309B2 (hr)
EP (1) EP1940251B1 (hr)
JP (1) JP2009512430A (hr)
CN (1) CN101291599A (hr)
AR (1) AR056129A1 (hr)
AT (1) ATE535159T1 (hr)
AU (1) AU2006303417A1 (hr)
BR (1) BRPI0617487A2 (hr)
CA (1) CA2622555A1 (hr)
CY (1) CY1112660T1 (hr)
DK (1) DK1940251T3 (hr)
ES (1) ES2378655T3 (hr)
HR (1) HRP20120138T1 (hr)
PL (1) PL1940251T3 (hr)
PT (1) PT1940251E (hr)
RS (1) RS52129B (hr)
SI (1) SI1940251T1 (hr)
TW (1) TW200803761A (hr)
WO (1) WO2007045533A1 (hr)

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CA2622555A1 (en) 2007-04-26
CY1112660T1 (el) 2016-02-10
RS52129B (en) 2012-08-31
AU2006303417A1 (en) 2007-04-26
JP2009512430A (ja) 2009-03-26
WO2007045533A1 (en) 2007-04-26
ES2378655T3 (es) 2012-04-16
CN101291599A (zh) 2008-10-22
ATE535159T1 (de) 2011-12-15
US8252309B2 (en) 2012-08-28
SI1940251T1 (sl) 2012-03-30
PT1940251E (pt) 2012-03-16
DK1940251T3 (da) 2012-03-19
US20060057188A1 (en) 2006-03-16
AR056129A1 (es) 2007-09-19
BRPI0617487A2 (pt) 2011-07-26
PL1940251T3 (pl) 2012-05-31
EP1940251B1 (en) 2011-11-30
TW200803761A (en) 2008-01-16
US20090257996A1 (en) 2009-10-15
EP1940251A1 (en) 2008-07-09

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