HRP20090592T1 - Izoksazolni derivat za ublažavanje neuropatskih bolova - Google Patents

Izoksazolni derivat za ublažavanje neuropatskih bolova Download PDF

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Publication number
HRP20090592T1
HRP20090592T1 HR20090592T HRP20090592T HRP20090592T1 HR P20090592 T1 HRP20090592 T1 HR P20090592T1 HR 20090592 T HR20090592 T HR 20090592T HR P20090592 T HRP20090592 T HR P20090592T HR P20090592 T1 HRP20090592 T1 HR P20090592T1
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HR
Croatia
Prior art keywords
neuropathic pain
pharmaceutically acceptable
treatment
formula
composition
Prior art date
Application number
HR20090592T
Other languages
English (en)
Inventor
Napoletano Mauro
Moriggi Ermanno
Original Assignee
Zambon S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon S.P.A. filed Critical Zambon S.P.A.
Publication of HRP20090592T1 publication Critical patent/HRP20090592T1/hr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Izoksazolni derivat formule (I) ili njegova farmaceutski prihvatljiva sol, naznačeni time, što se koriste za primjenu u liječenju neuropatskih bolova. Patent sadrži još 5 patentnih zahtjeva.

Claims (6)

1. Izoksazolni derivat formule (I) [image] ili njegova farmaceutski prihvatljiva sol, naznačeni time, što se koriste za primjenu u liječenju neuropatskih bolova.
2. Kompozicija za primjenu u liječenju neuropatskih bolova, naznačena time što kompozicija sadrži, kao aktivni spoj, spoj formule (I) prema patentnom zahtjevu 1 ili njegovu farmaceutski prihvatljivu sol i najmanje farmaceutski prihvatljiv inertni punitelj.
3. Primjena izoksazolnog derivata formule (I) [image] ili njegove farmaceutski prihvatljive soli, naznačena time, što se koristi u proizvodnji lijeka za liječenje neuropatskih bolova.
4. Primjena kompozicije u proizvodnji lijeka za liječenje neuropatskih bolova, naznačena time što kompozicija sadrži, kao aktivni spoj, spoj formule (I) prema patentnom zahtjevu 1 ili njegovu farmaceutski prihvatljivu sol i najmanje farmaceutski prihvatljiv inertni punitelj.
5. Jedinica pakovanja naznačena time što sadrži farmaceutsku kompoziciju prema patentnom zahtjevu 2, zajedno sa uputstvima za uporabu navedene kompozicije u liječenju neuropatskih bolova.
6. Farmaceutske kompozicije naznačene time što sadrže, kao aktivno sredstvo, spoj formule (I) prema patentnom zahtjevu 1 ili njegovu farmaceutski prihvatljivu sol u kombinaciji sa najmanje drugim spojem efikasnim u liječenju neuropatskih bolova i farmaceutski prihvatljivim inertnim puniteljem.
HR20090592T 2004-11-16 2009-11-04 Izoksazolni derivat za ublažavanje neuropatskih bolova HRP20090592T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT002187A ITMI20042187A1 (it) 2004-11-16 2004-11-16 Derivati isossazolici per allievare il dolore neiropatico
PCT/EP2005/055940 WO2006053860A1 (en) 2004-11-16 2005-11-14 Isoxazolic derivative to relieve neuropathic pain

Publications (1)

Publication Number Publication Date
HRP20090592T1 true HRP20090592T1 (hr) 2009-12-31

Family

ID=35840677

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20090592T HRP20090592T1 (hr) 2004-11-16 2009-11-04 Izoksazolni derivat za ublažavanje neuropatskih bolova

Country Status (16)

Country Link
US (1) US7834040B2 (hr)
EP (1) EP1817029B1 (hr)
AT (1) ATE442848T1 (hr)
CA (1) CA2586664C (hr)
CY (1) CY1110563T1 (hr)
DE (1) DE602005016711D1 (hr)
DK (1) DK1817029T3 (hr)
EA (1) EA013905B1 (hr)
ES (1) ES2331921T3 (hr)
HR (1) HRP20090592T1 (hr)
IT (1) ITMI20042187A1 (hr)
PL (1) PL1817029T3 (hr)
PT (1) PT1817029E (hr)
RS (1) RS51020B (hr)
SI (1) SI1817029T1 (hr)
WO (1) WO2006053860A1 (hr)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02500365A (ja) * 1987-05-20 1990-02-08 ザムボン グループ エス.ピー.エー. 認識補助作用を持つ化合物

Also Published As

Publication number Publication date
US20080108679A1 (en) 2008-05-08
CY1110563T1 (el) 2015-04-29
PT1817029E (pt) 2009-11-20
ATE442848T1 (de) 2009-10-15
RS51020B (sr) 2010-10-31
ITMI20042187A1 (it) 2005-02-16
WO2006053860A1 (en) 2006-05-26
EA200701086A1 (ru) 2007-12-28
ES2331921T3 (es) 2010-01-20
EP1817029B1 (en) 2009-09-16
CA2586664A1 (en) 2006-05-26
SI1817029T1 (sl) 2010-01-29
EP1817029A1 (en) 2007-08-15
DK1817029T3 (da) 2009-12-14
CA2586664C (en) 2012-09-18
US7834040B2 (en) 2010-11-16
DE602005016711D1 (de) 2009-10-29
PL1817029T3 (pl) 2010-02-26
EA013905B1 (ru) 2010-08-30

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