HRP20090592T1 - Izoksazolni derivat za ublažavanje neuropatskih bolova - Google Patents
Izoksazolni derivat za ublažavanje neuropatskih bolova Download PDFInfo
- Publication number
- HRP20090592T1 HRP20090592T1 HR20090592T HRP20090592T HRP20090592T1 HR P20090592 T1 HRP20090592 T1 HR P20090592T1 HR 20090592 T HR20090592 T HR 20090592T HR P20090592 T HRP20090592 T HR P20090592T HR P20090592 T1 HRP20090592 T1 HR P20090592T1
- Authority
- HR
- Croatia
- Prior art keywords
- neuropathic pain
- pharmaceutically acceptable
- treatment
- formula
- composition
- Prior art date
Links
- 208000004296 neuralgia Diseases 0.000 title claims abstract 8
- 208000021722 neuropathic pain Diseases 0.000 title claims abstract 8
- 150000003839 salts Chemical class 0.000 claims abstract 6
- 239000003814 drug Substances 0.000 claims abstract 3
- 150000001875 compounds Chemical class 0.000 claims 6
- 239000000203 mixture Substances 0.000 claims 5
- 239000000945 filler Substances 0.000 claims 3
- 229940079593 drug Drugs 0.000 claims 2
- 150000002545 isoxazoles Chemical class 0.000 claims 2
- 239000008194 pharmaceutical composition Substances 0.000 claims 2
- 239000013543 active substance Substances 0.000 claims 1
- 238000004806 packaging method and process Methods 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Izoksazolni derivat formule (I) ili njegova farmaceutski prihvatljiva sol, naznačeni time, što se koriste za primjenu u liječenju neuropatskih bolova. Patent sadrži još 5 patentnih zahtjeva.
Claims (6)
1. Izoksazolni derivat formule (I)
[image]
ili njegova farmaceutski prihvatljiva sol, naznačeni time, što se koriste za primjenu u liječenju neuropatskih bolova.
2. Kompozicija za primjenu u liječenju neuropatskih bolova, naznačena time što kompozicija sadrži, kao aktivni spoj, spoj formule (I) prema patentnom zahtjevu 1 ili njegovu farmaceutski prihvatljivu sol i najmanje farmaceutski prihvatljiv inertni punitelj.
3. Primjena izoksazolnog derivata formule (I)
[image]
ili njegove farmaceutski prihvatljive soli, naznačena time, što se koristi u proizvodnji lijeka za liječenje neuropatskih bolova.
4. Primjena kompozicije u proizvodnji lijeka za liječenje neuropatskih bolova, naznačena time što kompozicija sadrži, kao aktivni spoj, spoj formule (I) prema patentnom zahtjevu 1 ili njegovu farmaceutski prihvatljivu sol i najmanje farmaceutski prihvatljiv inertni punitelj.
5. Jedinica pakovanja naznačena time što sadrži farmaceutsku kompoziciju prema patentnom zahtjevu 2, zajedno sa uputstvima za uporabu navedene kompozicije u liječenju neuropatskih bolova.
6. Farmaceutske kompozicije naznačene time što sadrže, kao aktivno sredstvo, spoj formule (I) prema patentnom zahtjevu 1 ili njegovu farmaceutski prihvatljivu sol u kombinaciji sa najmanje drugim spojem efikasnim u liječenju neuropatskih bolova i farmaceutski prihvatljivim inertnim puniteljem.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT002187A ITMI20042187A1 (it) | 2004-11-16 | 2004-11-16 | Derivati isossazolici per allievare il dolore neiropatico |
PCT/EP2005/055940 WO2006053860A1 (en) | 2004-11-16 | 2005-11-14 | Isoxazolic derivative to relieve neuropathic pain |
Publications (1)
Publication Number | Publication Date |
---|---|
HRP20090592T1 true HRP20090592T1 (hr) | 2009-12-31 |
Family
ID=35840677
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HR20090592T HRP20090592T1 (hr) | 2004-11-16 | 2009-11-04 | Izoksazolni derivat za ublažavanje neuropatskih bolova |
Country Status (16)
Country | Link |
---|---|
US (1) | US7834040B2 (hr) |
EP (1) | EP1817029B1 (hr) |
AT (1) | ATE442848T1 (hr) |
CA (1) | CA2586664C (hr) |
CY (1) | CY1110563T1 (hr) |
DE (1) | DE602005016711D1 (hr) |
DK (1) | DK1817029T3 (hr) |
EA (1) | EA013905B1 (hr) |
ES (1) | ES2331921T3 (hr) |
HR (1) | HRP20090592T1 (hr) |
IT (1) | ITMI20042187A1 (hr) |
PL (1) | PL1817029T3 (hr) |
PT (1) | PT1817029E (hr) |
RS (1) | RS51020B (hr) |
SI (1) | SI1817029T1 (hr) |
WO (1) | WO2006053860A1 (hr) |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH02500365A (ja) * | 1987-05-20 | 1990-02-08 | ザムボン グループ エス.ピー.エー. | 認識補助作用を持つ化合物 |
-
2004
- 2004-11-16 IT IT002187A patent/ITMI20042187A1/it unknown
-
2005
- 2005-11-14 EP EP05815995A patent/EP1817029B1/en active Active
- 2005-11-14 SI SI200530813T patent/SI1817029T1/sl unknown
- 2005-11-14 DK DK05815995T patent/DK1817029T3/da active
- 2005-11-14 DE DE602005016711T patent/DE602005016711D1/de active Active
- 2005-11-14 RS RSP-2009/0477A patent/RS51020B/sr unknown
- 2005-11-14 AT AT05815995T patent/ATE442848T1/de active
- 2005-11-14 PT PT05815995T patent/PT1817029E/pt unknown
- 2005-11-14 US US11/718,935 patent/US7834040B2/en not_active Expired - Fee Related
- 2005-11-14 WO PCT/EP2005/055940 patent/WO2006053860A1/en active Application Filing
- 2005-11-14 EA EA200701086A patent/EA013905B1/ru not_active IP Right Cessation
- 2005-11-14 ES ES05815995T patent/ES2331921T3/es active Active
- 2005-11-14 CA CA2586664A patent/CA2586664C/en not_active Expired - Fee Related
- 2005-11-14 PL PL05815995T patent/PL1817029T3/pl unknown
-
2009
- 2009-11-04 HR HR20090592T patent/HRP20090592T1/hr unknown
- 2009-12-01 CY CY20091101263T patent/CY1110563T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
US20080108679A1 (en) | 2008-05-08 |
CY1110563T1 (el) | 2015-04-29 |
PT1817029E (pt) | 2009-11-20 |
ATE442848T1 (de) | 2009-10-15 |
RS51020B (sr) | 2010-10-31 |
ITMI20042187A1 (it) | 2005-02-16 |
WO2006053860A1 (en) | 2006-05-26 |
EA200701086A1 (ru) | 2007-12-28 |
ES2331921T3 (es) | 2010-01-20 |
EP1817029B1 (en) | 2009-09-16 |
CA2586664A1 (en) | 2006-05-26 |
SI1817029T1 (sl) | 2010-01-29 |
EP1817029A1 (en) | 2007-08-15 |
DK1817029T3 (da) | 2009-12-14 |
CA2586664C (en) | 2012-09-18 |
US7834040B2 (en) | 2010-11-16 |
DE602005016711D1 (de) | 2009-10-29 |
PL1817029T3 (pl) | 2010-02-26 |
EA013905B1 (ru) | 2010-08-30 |
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