HN2012001262A - Nuevos derivados de 8heterociclo-piperidina condensada)-( piperazinil)-1-alcanona o de (heterociclo-pirrolidina condensada)-(piperazinil)-1-alcanona y su utilizacion como inhibidores de p75 - Google Patents

Nuevos derivados de 8heterociclo-piperidina condensada)-( piperazinil)-1-alcanona o de (heterociclo-pirrolidina condensada)-(piperazinil)-1-alcanona y su utilizacion como inhibidores de p75

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HN2012001262A
HN2012001262A HN2012001262A HN2012001262A HN2012001262A HN 2012001262 A HN2012001262 A HN 2012001262A HN 2012001262 A HN2012001262 A HN 2012001262A HN 2012001262 A HN2012001262 A HN 2012001262A HN 2012001262 A HN2012001262 A HN 2012001262A
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Honduras
Prior art keywords
alcanone
piperazinil
heteroycycle
pirrolidine
concensed
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HN2012001262A
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English (en)
Inventor
Marco Baroni
Francoise Bono
Sandrine Delbary-Gossart
Valentina Vercesi
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Sanofi Sa
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Publication of HN2012001262A publication Critical patent/HN2012001262A/es

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Abstract

LA INVENCION SE REFIERE A DERIVADOS DE (HETEROCICLO-PIPERIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA Y A (HETEROCICLO-PIRROLIDINA CONDENSADAS)-(PIPERAZINIL)-1-ALCANONA DE FORMULA GENERAL (1) EN LA QUE A,W,N Y R2 SON TALES COMO SE DEFINEN EN LA REIVINDICACION 1, ASI COMO SU PROCEDIMIENTO DE PREPARACION Y SU APLICACION EN TERAPEUTICA.
HN2012001262A 2009-12-14 2012-06-13 Nuevos derivados de 8heterociclo-piperidina condensada)-( piperazinil)-1-alcanona o de (heterociclo-pirrolidina condensada)-(piperazinil)-1-alcanona y su utilizacion como inhibidores de p75 HN2012001262A (es)

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Application Number Priority Date Filing Date Title
FR0906023A FR2953839A1 (fr) 2009-12-14 2009-12-14 Nouveaux derives d'(heterocycle-piperidine condensee)-(piperazinyl)-1alcanone ou d'(heterocycle-pyrrolidine condensee)-(piperazinyl)-1alcanone et leur utilisation comme inhibiteurs de p75

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HN2012001262A true HN2012001262A (es) 2015-07-13

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FR2932481B1 (fr) 2008-06-13 2010-10-08 Sanofi Aventis Derives de 4-{2-°4-phenyl-3,6-dihydro-2h-pyridin-1-yl!-2- oxo-alkyl}-1-piperazin-2-one, leur preparation et leur application en therapeutique.
FR2932482B1 (fr) * 2008-06-13 2010-10-08 Sanofi Aventis Nouveaux derives de (phenyl-3,6-dihydro-2h-pyridinyl)- (piperazinyl ponte)-1-alcanone et leur utilisation comme inhibiteurs de p75
FR2953836B1 (fr) * 2009-12-14 2012-03-16 Sanofi Aventis Nouveaux derives (heterocycle-tetrahydro-pyridine)-(piperazinyl)-1-alcanone et (heterocycle-dihydro-pyrrolidine)-(piperazinyl)-1-alcanone et leur utilisation comme inhibiteurs de p75
FR2953839A1 (fr) * 2009-12-14 2011-06-17 Sanofi Aventis Nouveaux derives d'(heterocycle-piperidine condensee)-(piperazinyl)-1alcanone ou d'(heterocycle-pyrrolidine condensee)-(piperazinyl)-1alcanone et leur utilisation comme inhibiteurs de p75

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JP5735979B2 (ja) 2015-06-17
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FR2953839A1 (fr) 2011-06-17
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