HK1206358A1 - Process for the preparation of pyrazole carboxylic acid derivatives - Google Patents

Process for the preparation of pyrazole carboxylic acid derivatives

Info

Publication number
HK1206358A1
HK1206358A1 HK15107082.7A HK15107082A HK1206358A1 HK 1206358 A1 HK1206358 A1 HK 1206358A1 HK 15107082 A HK15107082 A HK 15107082A HK 1206358 A1 HK1206358 A1 HK 1206358A1
Authority
HK
Hong Kong
Prior art keywords
preparation
carboxylic acid
acid derivatives
pyrazole carboxylic
pyrazole
Prior art date
Application number
HK15107082.7A
Other languages
English (en)
Chinese (zh)
Inventor
比約恩.巴特爾斯
弗里茨.布利斯
卡特里.格勒布科茨賓登
馬蒂亞斯.克爾納
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HK1206358A1 publication Critical patent/HK1206358A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/16Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions not involving the amino or carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/04Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/12Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C281/00Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
    • C07C281/02Compounds containing any of the groups, e.g. carbazates
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C281/00Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
    • C07C281/02Compounds containing any of the groups, e.g. carbazates
    • C07C281/04Compounds containing any of the groups, e.g. carbazates the other nitrogen atom being further doubly-bound to a carbon atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HK15107082.7A 2012-08-17 2015-07-24 Process for the preparation of pyrazole carboxylic acid derivatives HK1206358A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12180802 2012-08-17
PCT/EP2013/066953 WO2014027009A1 (fr) 2012-08-17 2013-08-14 Procédé de préparation de dérivés d'acide pyrazole carboxylique

Publications (1)

Publication Number Publication Date
HK1206358A1 true HK1206358A1 (en) 2016-01-08

Family

ID=46851296

Family Applications (1)

Application Number Title Priority Date Filing Date
HK15107082.7A HK1206358A1 (en) 2012-08-17 2015-07-24 Process for the preparation of pyrazole carboxylic acid derivatives

Country Status (12)

Country Link
US (1) US9346763B2 (fr)
EP (1) EP2885276B1 (fr)
JP (1) JP6122118B2 (fr)
KR (1) KR20150042847A (fr)
CN (1) CN104540807B (fr)
BR (1) BR112015002779A2 (fr)
CA (1) CA2880846A1 (fr)
ES (1) ES2588056T3 (fr)
HK (1) HK1206358A1 (fr)
MX (1) MX348635B (fr)
RU (1) RU2638112C2 (fr)
WO (1) WO2014027009A1 (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ726432A (en) 2014-04-25 2022-07-01 Bayer Healthcare Llc Syringe with rolling diaphragm
ES2566228B1 (es) * 2014-09-11 2017-02-08 Consejo Superior De Investigaciones Cientificas Uso de ésteres derivados de pirazol protón-ionizables y sus correspondientes sales para el tratamiento de la enfermedad de Chagas y la leishmaniasis
CN104529899A (zh) * 2014-12-19 2015-04-22 浙江泰达作物科技有限公司 高区域选择性制备1-烷基-3-卤代烷基吡唑衍生物的方法
WO2016172467A1 (fr) 2015-04-24 2016-10-27 Bayer Healthcare Llc Seringue avec diaphragme roulant
AR109649A1 (es) 2016-09-16 2019-01-09 Bayer Healthcare Llc Camisa de presión con elemento de retención de jeringa
WO2018075386A1 (fr) 2016-10-17 2018-04-26 Bayer Healthcare Llc Injecteur de fluide avec mécanisme de mise en prise de seringue
CA3040480C (fr) 2016-10-17 2024-01-23 Bayer Healthcare Llc Injecteur de fluide avec mecanisme de mise en prise de seringue
WO2019055497A1 (fr) 2017-09-13 2019-03-21 Bayer Healthcare Llc Capuchon coulissant de seringue pour remplissage et distribution séparés
JP7440521B2 (ja) 2018-09-11 2024-02-28 バイエル・ヘルスケア・エルエルシー 液注入器システム用シリンジ保持特徴部
AU2020345829A1 (en) 2019-09-10 2022-03-17 Bayer Healthcare Llc Pressure jackets and syringe retention features for angiography fluid injectors
CN115151298A (zh) 2020-02-21 2022-10-04 拜耳医药保健有限责任公司 用于医疗流体递送的流体路径连接器
AU2021227677A1 (en) 2020-02-28 2022-09-15 Bayer Healthcare Llc Fluid mixing set
MX2022016123A (es) 2020-06-18 2023-02-09 Bayer Healthcare Llc Aparato de suspension de burbujas de aire en linea para trayectorias de fluidos de inyectores de angiografia.
CA3191167A1 (fr) 2020-08-11 2022-02-17 Bayer Healthcare Llc Caracteristiques pour une seringue d'angiographie
MX2023006363A (es) 2020-12-01 2023-06-13 Bayer Healthcare Llc Casete para la retencion de componentes de la trayectoria de un fluido para sistema inyector de fluido.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009116435A1 (fr) * 2008-03-18 2009-09-24 三井化学アグロ株式会社 Procédé de fabrication d'un dérivé d'acide acylacétique contenant du fluor, procédé de fabrication d'un dérivé d'ester d'acide carboxylique pyrazole contenant du fluor et procédé de fabrication d'un dérivé d'acide carboxylique pyrazole contenant du fluor
US8410117B2 (en) * 2010-03-26 2013-04-02 Hoffmann-La Roche Inc. Imidazopyrimidine derivatives

Also Published As

Publication number Publication date
CN104540807B (zh) 2016-09-14
EP2885276A1 (fr) 2015-06-24
MX348635B (es) 2017-06-22
WO2014027009A1 (fr) 2014-02-20
BR112015002779A2 (pt) 2019-10-15
CA2880846A1 (fr) 2014-02-20
JP2015530371A (ja) 2015-10-15
JP6122118B2 (ja) 2017-04-26
RU2015106856A (ru) 2016-10-10
RU2638112C2 (ru) 2017-12-15
ES2588056T3 (es) 2016-10-28
US20150158818A1 (en) 2015-06-11
EP2885276B1 (fr) 2016-06-01
CN104540807A (zh) 2015-04-22
KR20150042847A (ko) 2015-04-21
US9346763B2 (en) 2016-05-24
MX2015001023A (es) 2015-04-08
BR112015002779A8 (pt) 2017-12-19

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