BR112015002779A8 - processo para a preparação de derivados de ácido carboxílico de pirazol - Google Patents

processo para a preparação de derivados de ácido carboxílico de pirazol

Info

Publication number
BR112015002779A8
BR112015002779A8 BR112015002779A BR112015002779A BR112015002779A8 BR 112015002779 A8 BR112015002779 A8 BR 112015002779A8 BR 112015002779 A BR112015002779 A BR 112015002779A BR 112015002779 A BR112015002779 A BR 112015002779A BR 112015002779 A8 BR112015002779 A8 BR 112015002779A8
Authority
BR
Brazil
Prior art keywords
preparation
carboxylic acid
acid derivatives
pyrazole carboxylic
pyrazole
Prior art date
Application number
BR112015002779A
Other languages
English (en)
Other versions
BR112015002779A2 (pt
Inventor
Bartels Bjoern
Bliss Friitz
Groebke Zbinden Katrin
Koerner Matthias
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR112015002779A8 publication Critical patent/BR112015002779A8/pt
Publication of BR112015002779A2 publication Critical patent/BR112015002779A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/16Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions not involving the amino or carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/04Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/12Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C281/00Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
    • C07C281/02Compounds containing any of the groups, e.g. carbazates
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C281/00Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
    • C07C281/02Compounds containing any of the groups, e.g. carbazates
    • C07C281/04Compounds containing any of the groups, e.g. carbazates the other nitrogen atom being further doubly-bound to a carbon atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
BR112015002779A 2012-08-17 2013-08-14 processo para a preparação de derivados de ácido carboxílico de pirazol BR112015002779A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12180802 2012-08-17
PCT/EP2013/066953 WO2014027009A1 (en) 2012-08-17 2013-08-14 Process for the preparation of pyrazole carboxylic acid derivatives

Publications (2)

Publication Number Publication Date
BR112015002779A8 true BR112015002779A8 (pt) 2017-12-19
BR112015002779A2 BR112015002779A2 (pt) 2019-10-15

Family

ID=46851296

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015002779A BR112015002779A2 (pt) 2012-08-17 2013-08-14 processo para a preparação de derivados de ácido carboxílico de pirazol

Country Status (12)

Country Link
US (1) US9346763B2 (pt)
EP (1) EP2885276B1 (pt)
JP (1) JP6122118B2 (pt)
KR (1) KR20150042847A (pt)
CN (1) CN104540807B (pt)
BR (1) BR112015002779A2 (pt)
CA (1) CA2880846A1 (pt)
ES (1) ES2588056T3 (pt)
HK (1) HK1206358A1 (pt)
MX (1) MX348635B (pt)
RU (1) RU2638112C2 (pt)
WO (1) WO2014027009A1 (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2946838C (en) 2014-04-25 2023-04-04 Bayer Healthcare Llc Syringe with rolling diaphragm
ES2566228B1 (es) * 2014-09-11 2017-02-08 Consejo Superior De Investigaciones Cientificas Uso de ésteres derivados de pirazol protón-ionizables y sus correspondientes sales para el tratamiento de la enfermedad de Chagas y la leishmaniasis
CN104529899A (zh) * 2014-12-19 2015-04-22 浙江泰达作物科技有限公司 高区域选择性制备1-烷基-3-卤代烷基吡唑衍生物的方法
WO2016172467A1 (en) 2015-04-24 2016-10-27 Bayer Healthcare Llc Syringe with rolling diaphragm
CN109689129B (zh) 2016-09-16 2022-04-19 拜耳医药保健有限公司 具有针筒保持元件的压力护套
EP3525839B1 (en) 2016-10-17 2021-12-29 Bayer Healthcare LLC Fluid injector with syringe engagement mechanism
JP7023947B2 (ja) 2016-10-17 2022-02-22 バイエル・ヘルスケア・エルエルシー シリンジ係合機構を備える流体インジェクタ
ES2904369T3 (es) 2017-09-13 2022-04-04 Bayer Healthcare Llc Capuchón de jeringa deslizante para llenado y distribución por separado
EP4028077A1 (en) 2019-09-10 2022-07-20 Bayer HealthCare LLC Pressure jackets and syringe retention features for angiography fluid injectors
CN115151298A (zh) 2020-02-21 2022-10-04 拜耳医药保健有限责任公司 用于医疗流体递送的流体路径连接器
CN115697435A (zh) 2020-06-18 2023-02-03 拜耳医药保健有限责任公司 用于血管造影注入器流体路径的在线气泡悬浮装置

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8344156B2 (en) * 2008-03-18 2013-01-01 Mitsui Chemicals Agro, Inc. Method for producing fluorine-containing acylacetic acid derivative, method for producing fluorine-containing pyrazolecarboxylic acid ester derivative, and method for producing fluorine-containing pyrazolecarboxylic acid derivative
US8410117B2 (en) * 2010-03-26 2013-04-02 Hoffmann-La Roche Inc. Imidazopyrimidine derivatives

Also Published As

Publication number Publication date
JP2015530371A (ja) 2015-10-15
WO2014027009A1 (en) 2014-02-20
EP2885276A1 (en) 2015-06-24
HK1206358A1 (en) 2016-01-08
KR20150042847A (ko) 2015-04-21
US9346763B2 (en) 2016-05-24
RU2638112C2 (ru) 2017-12-15
BR112015002779A2 (pt) 2019-10-15
ES2588056T3 (es) 2016-10-28
MX348635B (es) 2017-06-22
MX2015001023A (es) 2015-04-08
JP6122118B2 (ja) 2017-04-26
RU2015106856A (ru) 2016-10-10
CN104540807A (zh) 2015-04-22
US20150158818A1 (en) 2015-06-11
EP2885276B1 (en) 2016-06-01
CN104540807B (zh) 2016-09-14
CA2880846A1 (en) 2014-02-20

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2595 DE 29-09-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]