HK1186732A1 - -芳基咪唑並 噠嗪、 -苯基咪唑並 吡啶、和 -苯基咪唑並 吡嗪衍生物 - Google Patents
-芳基咪唑並 噠嗪、 -苯基咪唑並 吡啶、和 -苯基咪唑並 吡嗪衍生物Info
- Publication number
- HK1186732A1 HK1186732A1 HK13114185.1A HK13114185A HK1186732A1 HK 1186732 A1 HK1186732 A1 HK 1186732A1 HK 13114185 A HK13114185 A HK 13114185A HK 1186732 A1 HK1186732 A1 HK 1186732A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- phenylimidazo
- arylimidazo
- pyridazine
- pyridine
- pyrazine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201061426216P | 2010-12-22 | 2010-12-22 | |
US201161514833P | 2011-08-03 | 2011-08-03 | |
US201161523688P | 2011-08-15 | 2011-08-15 | |
PCT/US2011/066837 WO2012088411A1 (en) | 2010-12-22 | 2011-12-22 | 2-arylimidazo[1,2-b]pyridazine, 2-phenylimidazo[1,2-a]pyridine, and 2-phenylimidazo[1,2-a]pyrazine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1186732A1 true HK1186732A1 (zh) | 2014-03-21 |
Family
ID=45478596
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK13114185.1A HK1186732A1 (zh) | 2010-12-22 | 2013-12-23 | -芳基咪唑並 噠嗪、 -苯基咪唑並 吡啶、和 -苯基咪唑並 吡嗪衍生物 |
Country Status (13)
Country | Link |
---|---|
US (1) | US8871767B2 (zh) |
EP (1) | EP2635578B1 (zh) |
JP (1) | JP6088980B2 (zh) |
KR (1) | KR101959726B1 (zh) |
CN (1) | CN103261198B (zh) |
AU (1) | AU2011348143B2 (zh) |
BR (1) | BR112013015959A2 (zh) |
CA (1) | CA2821546C (zh) |
HK (1) | HK1186732A1 (zh) |
MX (1) | MX2013007148A (zh) |
RU (1) | RU2598385C2 (zh) |
TW (1) | TWI617559B (zh) |
WO (1) | WO2012088411A1 (zh) |
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SI3083627T1 (sl) | 2013-12-19 | 2019-01-31 | Novartis Ag | Derivati (1,2,4)triazolo(1,5-a)pirimidina kot inhibitorji protozoan proteasoma za zdravljenje parazitskih bolezni, kot je lišmanioza |
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US20130131057A1 (en) | 2010-05-13 | 2013-05-23 | Centro Nacional De Investigaciones Oncologicas (Cnio | New bicyclic compounds as pi3-k and mtor inhibitors |
EP2444084A1 (en) | 2010-10-21 | 2012-04-25 | Centro Nacional de Investigaciones Oncológicas (CNIO) | Use of PI3K inibitors for the treatment of obesity |
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2011
- 2011-12-21 TW TW100147653A patent/TWI617559B/zh not_active IP Right Cessation
- 2011-12-22 CA CA2821546A patent/CA2821546C/en not_active Expired - Fee Related
- 2011-12-22 US US13/335,072 patent/US8871767B2/en not_active Expired - Fee Related
- 2011-12-22 BR BR112013015959A patent/BR112013015959A2/pt not_active Application Discontinuation
- 2011-12-22 RU RU2013133881/04A patent/RU2598385C2/ru not_active IP Right Cessation
- 2011-12-22 WO PCT/US2011/066837 patent/WO2012088411A1/en active Application Filing
- 2011-12-22 CN CN201180059833.XA patent/CN103261198B/zh active Active
- 2011-12-22 MX MX2013007148A patent/MX2013007148A/es active IP Right Grant
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- 2011-12-22 KR KR1020137018166A patent/KR101959726B1/ko active IP Right Grant
- 2011-12-22 EP EP11808541.4A patent/EP2635578B1/en active Active
- 2011-12-22 AU AU2011348143A patent/AU2011348143B2/en not_active Ceased
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Also Published As
Publication number | Publication date |
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KR20140019311A (ko) | 2014-02-14 |
US20120178751A1 (en) | 2012-07-12 |
CA2821546C (en) | 2019-03-05 |
MX2013007148A (es) | 2013-11-01 |
CN103261198B (zh) | 2016-06-08 |
US8871767B2 (en) | 2014-10-28 |
AU2011348143A1 (en) | 2013-06-20 |
JP2014500331A (ja) | 2014-01-09 |
TWI617559B (zh) | 2018-03-11 |
WO2012088411A1 (en) | 2012-06-28 |
RU2598385C2 (ru) | 2016-09-27 |
BR112013015959A2 (pt) | 2018-07-10 |
CN103261198A (zh) | 2013-08-21 |
CA2821546A1 (en) | 2012-06-28 |
JP6088980B2 (ja) | 2017-03-01 |
TW201307342A (zh) | 2013-02-16 |
EP2635578B1 (en) | 2015-12-16 |
RU2013133881A (ru) | 2015-01-27 |
AU2011348143B2 (en) | 2016-09-08 |
KR101959726B1 (ko) | 2019-03-19 |
EP2635578A1 (en) | 2013-09-11 |
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