HK1176548A1 - Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg - Google Patents

Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg

Info

Publication number
HK1176548A1
HK1176548A1 HK13103363.8A HK13103363A HK1176548A1 HK 1176548 A1 HK1176548 A1 HK 1176548A1 HK 13103363 A HK13103363 A HK 13103363A HK 1176548 A1 HK1176548 A1 HK 1176548A1
Authority
HK
Hong Kong
Prior art keywords
mgbg
pharmaceutical
methods
oral delivery
treating disease
Prior art date
Application number
HK13103363.8A
Other languages
English (en)
Chinese (zh)
Inventor
．麥基爾恩
．布利策
Original Assignee
帕薩羅杰卡有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 帕薩羅杰卡有限公司 filed Critical 帕薩羅杰卡有限公司
Publication of HK1176548A1 publication Critical patent/HK1176548A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
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    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Biophysics (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Biotechnology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
HK13103363.8A 2009-07-16 2013-03-18 Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg HK1176548A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22606009P 2009-07-16 2009-07-16
US29009509P 2009-12-24 2009-12-24
PCT/US2010/042253 WO2011009039A2 (en) 2009-07-16 2010-07-16 Pharmaceutical for oral delivery comprising mgbg and methods of treating disease

Publications (1)

Publication Number Publication Date
HK1176548A1 true HK1176548A1 (en) 2013-08-02

Family

ID=43450234

Family Applications (1)

Application Number Title Priority Date Filing Date
HK13103363.8A HK1176548A1 (en) 2009-07-16 2013-03-18 Pharmaceutical for oral delivery comprising mgbg and methods of treating disease mgbg

Country Status (12)

Country Link
US (4) US8258186B2 (de)
EP (2) EP3473247A1 (de)
JP (4) JP6112449B2 (de)
CN (2) CN104997762B (de)
AU (2) AU2010273277B2 (de)
BR (1) BR112012000862A8 (de)
CA (1) CA2768018C (de)
DK (1) DK2453886T3 (de)
ES (1) ES2715173T3 (de)
HK (1) HK1176548A1 (de)
NZ (3) NZ715686A (de)
WO (1) WO2011009039A2 (de)

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NZ715686A (en) 2009-07-16 2017-08-25 Pathologica Llc Pharmaceutical for oral delivery comprising mgbg and methods of treating disease
US9675566B2 (en) * 2009-07-16 2017-06-13 Pathologica Llc Method of treatment with anti-inflammatory and analgesic compounds which are GI-, renal-, and platelet-sparing
PT2665471T (pt) 2011-01-19 2018-03-21 Pathologica Llc Formas de dosagem farmacêutica orais de libertação controlada que compreendem mgbg
WO2013083813A2 (en) * 2011-12-07 2013-06-13 Universität Zürich Modulators of spermine/spermidine n'-acetyltransferase (ssat) and ssat associated proteins for use in prevention or treatment of rheumatoid arthritis
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BR112012000862A8 (pt) 2018-01-09
EP2453886A4 (de) 2012-12-05
US20110112199A1 (en) 2011-05-12
US20170290788A1 (en) 2017-10-12
CN104997762B (zh) 2019-03-08
CA2768018A1 (en) 2011-01-20
JP2020063258A (ja) 2020-04-23
US8609734B2 (en) 2013-12-17
NZ597488A (en) 2014-10-31
AU2010273277A1 (en) 2012-02-02
CA2768018C (en) 2019-08-27
JP2018127460A (ja) 2018-08-16
DK2453886T3 (en) 2019-03-25
EP3473247A1 (de) 2019-04-24
JP2016065045A (ja) 2016-04-28
EP2453886B1 (de) 2018-12-12
EP2453886A2 (de) 2012-05-23
AU2016266049B2 (en) 2018-10-18
JP6112449B2 (ja) 2017-04-12
CN102686222A (zh) 2012-09-19
CN104997762A (zh) 2015-10-28
US8258186B2 (en) 2012-09-04
AU2010273277B2 (en) 2016-12-22
NZ715686A (en) 2017-08-25
BR112012000862A2 (pt) 2017-10-31
AU2016266049A1 (en) 2016-12-22
JP2012533565A (ja) 2012-12-27
US20140051765A1 (en) 2014-02-20
US9616035B2 (en) 2017-04-11
WO2011009039A2 (en) 2011-01-20
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JP6883930B2 (ja) 2021-06-09
ES2715173T3 (es) 2019-06-03

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