HK1088327A1 - Thiadiazine derivatives and use thereof as positive ampa receptor modulator - Google Patents

Thiadiazine derivatives and use thereof as positive ampa receptor modulator

Info

Publication number
HK1088327A1
HK1088327A1 HK06108870A HK06108870A HK1088327A1 HK 1088327 A1 HK1088327 A1 HK 1088327A1 HK 06108870 A HK06108870 A HK 06108870A HK 06108870 A HK06108870 A HK 06108870A HK 1088327 A1 HK1088327 A1 HK 1088327A1
Authority
HK
Hong Kong
Prior art keywords
receptor modulator
ampa receptor
thiadiazine derivatives
positive ampa
positive
Prior art date
Application number
HK06108870A
Other languages
English (en)
Inventor
Graindorge Emmanuel
Francotte Pierre
Boverie Stephane
De Tullio Pascal
Pirotte Bernard
Lestage Pierre
Danober Laurence
Renard Pierre
Caignard Daniel-Henri
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of HK1088327A1 publication Critical patent/HK1088327A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
HK06108870A 2003-05-05 2006-08-10 Thiadiazine derivatives and use thereof as positive ampa receptor modulator HK1088327A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0305448A FR2854634B1 (fr) 2003-05-05 2003-05-05 Nouveaux derives de thiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
PCT/FR2004/001070 WO2004099217A1 (fr) 2003-05-05 2004-05-04 Derives de thiadiazine et leur utilisation comme modulateurs positifs des recepteurs ampa

Publications (1)

Publication Number Publication Date
HK1088327A1 true HK1088327A1 (en) 2006-11-03

Family

ID=33306157

Family Applications (1)

Application Number Title Priority Date Filing Date
HK06108870A HK1088327A1 (en) 2003-05-05 2006-08-10 Thiadiazine derivatives and use thereof as positive ampa receptor modulator

Country Status (21)

Country Link
US (1) US7476668B2 (ru)
EP (1) EP1620441A1 (ru)
JP (1) JP4461139B2 (ru)
KR (1) KR100741235B1 (ru)
CN (1) CN100363368C (ru)
AR (1) AR044245A1 (ru)
AU (1) AU2004236005B2 (ru)
BR (1) BRPI0410002A (ru)
CA (1) CA2524377C (ru)
EA (1) EA009240B1 (ru)
FR (1) FR2854634B1 (ru)
GE (1) GEP20084318B (ru)
HK (1) HK1088327A1 (ru)
MA (1) MA27732A1 (ru)
MX (1) MXPA05011823A (ru)
MY (1) MY136694A (ru)
NO (1) NO20055695L (ru)
NZ (1) NZ543214A (ru)
UA (1) UA80046C2 (ru)
WO (1) WO2004099217A1 (ru)
ZA (1) ZA200508660B (ru)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2005280058B2 (en) 2004-08-25 2010-09-02 Essentialis, Inc. Pharmaceutical formulations of potassium ATP channel openers and uses thereof
US7799777B2 (en) 2006-01-05 2010-09-21 Essentialis, Inc. Salts of potassium ATP channel openers and uses thereof
US20110218190A1 (en) * 2008-11-10 2011-09-08 The Regents Of The University Of California Therapeutic uses of ampa receptor modulators for treatment of motor dysfunction
HUE049460T2 (hu) 2010-08-10 2020-09-28 Takeda Pharmaceuticals Co Heterociklusos vegyület és annak alkalmazása ampa receptor pozitív allosztérikus modulátorként
JP5901365B2 (ja) * 2012-03-12 2016-04-06 株式会社トクヤマ イミダート化合物の製造方法
EP3311842A1 (en) 2013-06-13 2018-04-25 VeroScience LLC Compositions and methods for treating metabolic disorders
CA2991400C (en) 2015-07-06 2020-05-12 Public University Corporation Yokohama City University Phenylsulphonamide derivatives useful as ampa receptor imaging agents
JP6241974B1 (ja) 2017-01-11 2017-12-06 公立大学法人横浜市立大学 霊長類生体の脳内ａｍｐａ受容体のイメージング方法、プログラム、及びスクリーニング方法
US10680583B1 (en) * 2019-02-26 2020-06-09 Xilinx, Inc. Control circuit for and method of controlling an operation of an integrated circuit device

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3733409A (en) * 1969-05-20 1973-05-15 Schering Corp Method of treating hypertension using thieno (1,2,4) thiadiazines
AU4345297A (en) * 1996-09-17 1998-04-14 Regents Of The University Of California, The Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor
KR20010021936A (ko) * 1997-07-16 2001-03-15 한센 핀 베네드, 안네 제헤르, 웨이콥 마리안느 융합된 1,2,4-티아디아진 유도체, 그의 제조와 사용
CA2320354A1 (en) * 1998-02-18 1999-08-26 Neurosearch A/S Novel compounds and their use as positive ampa receptor modulators
FR2801587B1 (fr) * 1999-11-30 2002-01-11 Adir Nouveaux derives de benzothiadiazines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
CN100363368C (zh) 2008-01-23
MXPA05011823A (es) 2006-05-25
JP4461139B2 (ja) 2010-05-12
FR2854634A1 (fr) 2004-11-12
WO2004099217A1 (fr) 2004-11-18
CA2524377C (fr) 2010-08-24
BRPI0410002A (pt) 2006-04-25
CA2524377A1 (fr) 2004-11-18
NZ543214A (en) 2009-02-28
CN1798750A (zh) 2006-07-05
AU2004236005B2 (en) 2010-01-21
UA80046C2 (en) 2007-08-10
US7476668B2 (en) 2009-01-13
MY136694A (en) 2008-11-28
AU2004236005A1 (en) 2004-11-18
JP2006525292A (ja) 2006-11-09
GEP20084318B (en) 2008-03-10
KR20060006830A (ko) 2006-01-19
US20070004709A1 (en) 2007-01-04
ZA200508660B (en) 2007-01-31
EA200501696A1 (ru) 2006-06-30
EP1620441A1 (fr) 2006-02-01
EA009240B1 (ru) 2007-12-28
MA27732A1 (fr) 2006-01-02
NO20055695L (no) 2005-12-01
KR100741235B1 (ko) 2007-07-19
AR044245A1 (es) 2005-09-07
FR2854634B1 (fr) 2005-07-08

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20120504