HK1064950A1 - Methods for treating or preventing vascular inflammation using sterol absorption inhibitor(s) - Google Patents
Methods for treating or preventing vascular inflammation using sterol absorption inhibitor(s)Info
- Publication number
- HK1064950A1 HK1064950A1 HK04107816.3A HK04107816A HK1064950A1 HK 1064950 A1 HK1064950 A1 HK 1064950A1 HK 04107816 A HK04107816 A HK 04107816A HK 1064950 A1 HK1064950 A1 HK 1064950A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- absorption inhibitor
- treating
- methods
- vascular inflammation
- preventing vascular
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US32393701P | 2001-09-21 | 2001-09-21 | |
PCT/US2002/029756 WO2003026644A1 (en) | 2001-09-21 | 2002-09-19 | Methods for treating or preventing vascular inflammation using sterol absorption inhibitor(s) |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1064950A1 true HK1064950A1 (en) | 2005-02-08 |
Family
ID=23261347
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK04107816.3A HK1064950A1 (en) | 2001-09-21 | 2004-10-11 | Methods for treating or preventing vascular inflammation using sterol absorption inhibitor(s) |
Country Status (21)
Country | Link |
---|---|
US (1) | US20030119757A1 (zh) |
EP (1) | EP1427409B1 (zh) |
JP (2) | JP4395370B2 (zh) |
CN (2) | CN1556700A (zh) |
AT (1) | ATE411018T1 (zh) |
AU (2) | AU2002335770B2 (zh) |
BR (1) | BR0212907A (zh) |
CA (1) | CA2460344A1 (zh) |
CY (1) | CY1110894T1 (zh) |
DE (1) | DE60229406D1 (zh) |
DK (1) | DK1427409T3 (zh) |
ES (1) | ES2312624T3 (zh) |
HK (1) | HK1064950A1 (zh) |
HU (1) | HUP0401501A3 (zh) |
MX (1) | MXPA04002572A (zh) |
NO (1) | NO333968B1 (zh) |
NZ (1) | NZ531060A (zh) |
PT (1) | PT1427409E (zh) |
SI (1) | SI1427409T1 (zh) |
WO (1) | WO2003026644A1 (zh) |
ZA (1) | ZA200402104B (zh) |
Families Citing this family (25)
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JP2005504091A (ja) * | 2001-09-21 | 2005-02-10 | シェーリング コーポレイション | ステロール吸収阻害剤としてアゼチジノンを用いる黄色腫の処置 |
GB0215579D0 (en) | 2002-07-05 | 2002-08-14 | Astrazeneca Ab | Chemical compounds |
NZ539624A (en) * | 2002-09-27 | 2008-08-29 | Martek Biosciences Corp | Prophylactic docosahexaenoic acid therapy for patients with subclinical inflammation |
US7208486B2 (en) | 2003-03-07 | 2007-04-24 | Schering Corporation | Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof |
WO2004081002A1 (en) | 2003-03-07 | 2004-09-23 | Schering Corporation | Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia |
US20070003600A1 (en) * | 2003-06-11 | 2007-01-04 | Carolyn Moore | Methods for reducing c-reactive protein |
EP1680189A2 (en) * | 2003-11-05 | 2006-07-19 | Schering Corporation | Combinations of lipid modulating agents and substituted azetidinones and treatments for vascular conditions |
PL380414A1 (pl) * | 2003-11-10 | 2007-01-22 | Microbia, Inc. | 4-Diarylo-1- fenyloazetydyn-2-ony |
GB0329778D0 (en) * | 2003-12-23 | 2004-01-28 | Astrazeneca Ab | Chemical compounds |
WO2005061452A1 (en) | 2003-12-23 | 2005-07-07 | Astrazeneca Ab | Diphenylazetidinone derivates possessing cholesterol absorption inhibitory activity |
US7803838B2 (en) * | 2004-06-04 | 2010-09-28 | Forest Laboratories Holdings Limited | Compositions comprising nebivolol |
US7838552B2 (en) | 2004-06-04 | 2010-11-23 | Forest Laboratories Holdings Limited | Compositions comprising nebivolol |
CN101035520A (zh) * | 2004-08-09 | 2007-09-12 | 武田药品工业株式会社 | Crp降低剂 |
UY29607A1 (es) * | 2005-06-20 | 2007-01-31 | Astrazeneca Ab | Compuestos quimicos |
AR057072A1 (es) * | 2005-06-22 | 2007-11-14 | Astrazeneca Ab | Compuestos quimicos derivados de 2-azetidinona, formulacion farmaceutica y un proceso de preparacion del compuesto |
AR054482A1 (es) * | 2005-06-22 | 2007-06-27 | Astrazeneca Ab | Derivados de azetidinona para el tratamiento de hiperlipidemias |
AR057383A1 (es) * | 2005-06-22 | 2007-12-05 | Astrazeneca Ab | Compuestos quimicos derivados de 2-azetidinona, formulacion farmaceutica y un proceso de preparacion del compuesto |
SA06270191B1 (ar) | 2005-06-22 | 2010-03-29 | استرازينيكا ايه بي | مشتقات من 2- أزيتيدينون جديدة باعتبارها مثبطات لامتصاص الكوليسترول لعلاج حالات فرط نسبة الدهون في الدم |
AR057380A1 (es) * | 2005-06-22 | 2007-11-28 | Astrazeneca Ab | Compuestos quimicos derivados de 2-azetidinona y uso terapeutico de los mismos |
JP2009529055A (ja) * | 2006-03-06 | 2009-08-13 | テバ ファーマシューティカル インダストリーズ リミティド | エゼチミベ組成物 |
AR060623A1 (es) * | 2006-04-27 | 2008-07-02 | Astrazeneca Ab | Compuestos derivados de 2-azetidinona y un metodo de preparacion |
JP4740938B2 (ja) | 2007-12-27 | 2011-08-03 | ダイセル化学工業株式会社 | 6位高アセチル化セルロースジアセテート及びその製造方法 |
CA2757722C (en) | 2009-04-01 | 2018-05-22 | Matrix Laboratories Ltd. | Enzymatic process for the preparation of (s)-5-(4-fluoro-phenyl)-5-hydroxy- 1morpholin-4-yl-pentan-1-one, an intermediate of ezetimibe and further conversion to ezetimibe |
CN103755617A (zh) * | 2013-12-31 | 2014-04-30 | 北京万全德众医药生物技术有限公司 | 一种制备依折麦布关键杂质的方法 |
CN103755616A (zh) * | 2013-12-31 | 2014-04-30 | 北京万全德众医药生物技术有限公司 | 一种制备依泽替米贝异构体的方法 |
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-
2002
- 2002-09-19 HU HU0401501A patent/HUP0401501A3/hu unknown
- 2002-09-19 DK DK02770534T patent/DK1427409T3/da active
- 2002-09-19 SI SI200230758T patent/SI1427409T1/sl unknown
- 2002-09-19 EP EP02770534A patent/EP1427409B1/en not_active Expired - Lifetime
- 2002-09-19 MX MXPA04002572A patent/MXPA04002572A/es active IP Right Grant
- 2002-09-19 ES ES02770534T patent/ES2312624T3/es not_active Expired - Lifetime
- 2002-09-19 PT PT02770534T patent/PT1427409E/pt unknown
- 2002-09-19 BR BR0212907-8A patent/BR0212907A/pt not_active Application Discontinuation
- 2002-09-19 AT AT02770534T patent/ATE411018T1/de active
- 2002-09-19 AU AU2002335770A patent/AU2002335770B2/en not_active Ceased
- 2002-09-19 US US10/247,032 patent/US20030119757A1/en not_active Abandoned
- 2002-09-19 CN CNA028184343A patent/CN1556700A/zh active Pending
- 2002-09-19 CN CN200910261594A patent/CN101785772A/zh active Pending
- 2002-09-19 CA CA002460344A patent/CA2460344A1/en not_active Abandoned
- 2002-09-19 DE DE60229406T patent/DE60229406D1/de not_active Expired - Lifetime
- 2002-09-19 JP JP2003530281A patent/JP4395370B2/ja not_active Expired - Fee Related
- 2002-09-19 WO PCT/US2002/029756 patent/WO2003026644A1/en active IP Right Grant
- 2002-09-19 NZ NZ531060A patent/NZ531060A/en not_active IP Right Cessation
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2004
- 2004-03-16 ZA ZA2004/02104A patent/ZA200402104B/en unknown
- 2004-04-20 NO NO20041598A patent/NO333968B1/no not_active IP Right Cessation
- 2004-10-11 HK HK04107816.3A patent/HK1064950A1/xx not_active IP Right Cessation
-
2005
- 2005-11-18 AU AU2005234666A patent/AU2005234666B2/en not_active Ceased
-
2008
- 2008-12-08 CY CY20081101419T patent/CY1110894T1/el unknown
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2009
- 2009-09-11 JP JP2009211106A patent/JP2009286801A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
HUP0401501A2 (hu) | 2004-12-28 |
US20030119757A1 (en) | 2003-06-26 |
WO2003026644A1 (en) | 2003-04-03 |
DK1427409T3 (da) | 2009-01-12 |
EP1427409B1 (en) | 2008-10-15 |
ZA200402104B (en) | 2005-06-29 |
NO333968B1 (no) | 2013-11-04 |
ES2312624T3 (es) | 2009-03-01 |
NZ531060A (en) | 2006-06-30 |
EP1427409A1 (en) | 2004-06-16 |
MXPA04002572A (es) | 2004-05-31 |
JP2009286801A (ja) | 2009-12-10 |
CN101785772A (zh) | 2010-07-28 |
HUP0401501A3 (en) | 2012-02-28 |
ATE411018T1 (de) | 2008-10-15 |
CN1556700A (zh) | 2004-12-22 |
BR0212907A (pt) | 2004-10-13 |
NO20041598L (no) | 2004-06-17 |
JP2005504092A (ja) | 2005-02-10 |
CA2460344A1 (en) | 2003-04-03 |
DE60229406D1 (de) | 2008-11-27 |
JP4395370B2 (ja) | 2010-01-06 |
AU2002335770B2 (en) | 2005-08-18 |
CY1110894T1 (el) | 2015-06-10 |
AU2005234666A1 (en) | 2005-12-08 |
PT1427409E (pt) | 2008-11-27 |
SI1427409T1 (sl) | 2009-02-28 |
AU2005234666B2 (en) | 2006-09-21 |
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