BR0212907A - Métodos para tratamento ou prevenção de inflamação vascular usando inibidor(es) da absorção de esteróis - Google Patents

Métodos para tratamento ou prevenção de inflamação vascular usando inibidor(es) da absorção de esteróis

Info

Publication number
BR0212907A
BR0212907A BR0212907-8A BR0212907A BR0212907A BR 0212907 A BR0212907 A BR 0212907A BR 0212907 A BR0212907 A BR 0212907A BR 0212907 A BR0212907 A BR 0212907A
Authority
BR
Brazil
Prior art keywords
methods
treating
vascular inflammation
absorption inhibitor
sterol absorption
Prior art date
Application number
BR0212907-8A
Other languages
English (en)
Inventor
Harry R Davis
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23261347&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR0212907(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of BR0212907A publication Critical patent/BR0212907A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)

Abstract

"MéTODOS PARA TRATAMENTO OU PREVENçãO DE INFLAMAçãO VASCULAR USANDO INIBIDOR(ES) DA ABSORçãO DE ESTERóIS". A presente invenção refere-se a métodos para tratar ou prevenir inflamação vascular ou para reduzir os níveis sang³íneos de proteína c-reativa por administração de pelo menos um inibidor da absorção de esterol e/ou pelo menos um inibidor da absorção de 5<244>-estanol.
BR0212907-8A 2001-09-21 2002-09-19 Métodos para tratamento ou prevenção de inflamação vascular usando inibidor(es) da absorção de esteróis BR0212907A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32393701P 2001-09-21 2001-09-21
PCT/US2002/029756 WO2003026644A1 (en) 2001-09-21 2002-09-19 Methods for treating or preventing vascular inflammation using sterol absorption inhibitor(s)

Publications (1)

Publication Number Publication Date
BR0212907A true BR0212907A (pt) 2004-10-13

Family

ID=23261347

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0212907-8A BR0212907A (pt) 2001-09-21 2002-09-19 Métodos para tratamento ou prevenção de inflamação vascular usando inibidor(es) da absorção de esteróis

Country Status (21)

Country Link
US (1) US20030119757A1 (pt)
EP (1) EP1427409B1 (pt)
JP (2) JP4395370B2 (pt)
CN (2) CN101785772A (pt)
AT (1) ATE411018T1 (pt)
AU (2) AU2002335770B2 (pt)
BR (1) BR0212907A (pt)
CA (1) CA2460344A1 (pt)
CY (1) CY1110894T1 (pt)
DE (1) DE60229406D1 (pt)
DK (1) DK1427409T3 (pt)
ES (1) ES2312624T3 (pt)
HK (1) HK1064950A1 (pt)
HU (1) HUP0401501A3 (pt)
MX (1) MXPA04002572A (pt)
NO (1) NO333968B1 (pt)
NZ (1) NZ531060A (pt)
PT (1) PT1427409E (pt)
SI (1) SI1427409T1 (pt)
WO (1) WO2003026644A1 (pt)
ZA (1) ZA200402104B (pt)

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AR057383A1 (es) * 2005-06-22 2007-12-05 Astrazeneca Ab Compuestos quimicos derivados de 2-azetidinona, formulacion farmaceutica y un proceso de preparacion del compuesto
AR057380A1 (es) * 2005-06-22 2007-11-28 Astrazeneca Ab Compuestos quimicos derivados de 2-azetidinona y uso terapeutico de los mismos
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JP4395370B2 (ja) 2010-01-06
DE60229406D1 (de) 2008-11-27
AU2005234666A1 (en) 2005-12-08
MXPA04002572A (es) 2004-05-31
NO333968B1 (no) 2013-11-04
PT1427409E (pt) 2008-11-27
NO20041598L (no) 2004-06-17
NZ531060A (en) 2006-06-30
JP2005504092A (ja) 2005-02-10
CA2460344A1 (en) 2003-04-03
JP2009286801A (ja) 2009-12-10
AU2002335770B2 (en) 2005-08-18
AU2005234666B2 (en) 2006-09-21
ES2312624T3 (es) 2009-03-01
SI1427409T1 (sl) 2009-02-28
EP1427409A1 (en) 2004-06-16
HUP0401501A2 (hu) 2004-12-28
CY1110894T1 (el) 2015-06-10
HK1064950A1 (en) 2005-02-08
WO2003026644A1 (en) 2003-04-03
DK1427409T3 (da) 2009-01-12
EP1427409B1 (en) 2008-10-15
CN1556700A (zh) 2004-12-22
CN101785772A (zh) 2010-07-28
US20030119757A1 (en) 2003-06-26
ATE411018T1 (de) 2008-10-15
HUP0401501A3 (en) 2012-02-28

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