CY1106791T1 - Συνδυασμοι αναστολεα (-ων) απορροφησης στερολης με καρδιαγγειακο παραγοντα (-ες) για τη θεραπεια αγγειακων καταστασεων - Google Patents
Συνδυασμοι αναστολεα (-ων) απορροφησης στερολης με καρδιαγγειακο παραγοντα (-ες) για τη θεραπεια αγγειακων καταστασεωνInfo
- Publication number
- CY1106791T1 CY1106791T1 CY20071101045T CY071101045T CY1106791T1 CY 1106791 T1 CY1106791 T1 CY 1106791T1 CY 20071101045 T CY20071101045 T CY 20071101045T CY 071101045 T CY071101045 T CY 071101045T CY 1106791 T1 CY1106791 T1 CY 1106791T1
- Authority
- CY
- Cyprus
- Prior art keywords
- absorption inhibitor
- combinations
- sterol absorption
- treatment
- vascular conditions
- Prior art date
Links
- 229930182558 Sterol Natural products 0.000 title abstract 4
- 150000003432 sterols Chemical class 0.000 title abstract 4
- 235000003702 sterols Nutrition 0.000 title abstract 4
- 238000010521 absorption reaction Methods 0.000 title abstract 3
- 239000003112 inhibitor Substances 0.000 title abstract 3
- 230000002792 vascular Effects 0.000 title abstract 2
- 239000002371 cardiac agent Substances 0.000 title 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 229940125692 cardiovascular agent Drugs 0.000 abstract 1
- 239000002327 cardiovascular agent Substances 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/74—Synthetic polymeric materials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/455—Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Abstract
Η παρούσα εφεύρεση παρέχει συνθέσεις, θεραπευτικούς συνδυασμούς και μεθόδους που συμπεριλαμβάνουν: (α) τουλάχιστον έναν αναστολέα απορρόφησης στερόλης και (β) τουλάχιστον έναν καρδιαγγειακό παράγοντα διαφορετικό από τον αναστολέα απορρόφησης στερόλης, που μπορεί να είναι χρήσιμοι για θεραπεία αγγειακών καταστάσεων, παχυσαρκίας, διαβήτη και μείωσης επιπέδων στερολών στο πλάσμα.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US26427501P | 2001-01-26 | 2001-01-26 | |
US26439601P | 2001-01-26 | 2001-01-26 | |
US26460001P | 2001-01-26 | 2001-01-26 | |
US32384201P | 2001-09-21 | 2001-09-21 | |
PCT/US2002/001196 WO2002058731A2 (en) | 2001-01-26 | 2002-01-25 | Combinations of sterol absorption inhibitor(s) with cardiovascular agent(s) for the treatment of vascular conditions |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1106791T1 true CY1106791T1 (el) | 2012-05-23 |
Family
ID=27500817
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20071101045T CY1106791T1 (el) | 2001-01-26 | 2007-08-07 | Συνδυασμοι αναστολεα (-ων) απορροφησης στερολης με καρδιαγγειακο παραγοντα (-ες) για τη θεραπεια αγγειακων καταστασεων |
Country Status (28)
Country | Link |
---|---|
US (1) | US20030069221A1 (el) |
EP (3) | EP1541175A3 (el) |
JP (1) | JP2004517919A (el) |
KR (2) | KR20080077033A (el) |
CN (1) | CN1582168A (el) |
AR (2) | AR032643A1 (el) |
AT (1) | ATE362757T1 (el) |
AU (1) | AU2002241903B2 (el) |
BR (1) | BR0206644A (el) |
CA (1) | CA2434436A1 (el) |
CY (1) | CY1106791T1 (el) |
CZ (1) | CZ20032031A3 (el) |
DE (1) | DE60220269T2 (el) |
DK (1) | DK1385548T3 (el) |
EC (1) | ECSP074704A (el) |
ES (1) | ES2286233T3 (el) |
HK (1) | HK1060854A1 (el) |
HU (1) | HUP0303923A2 (el) |
IL (2) | IL156585A0 (el) |
MX (1) | MXPA03006724A (el) |
NO (1) | NO20033358L (el) |
NZ (1) | NZ545332A (el) |
PL (1) | PL369033A1 (el) |
PT (1) | PT1385548E (el) |
RU (1) | RU2003126186A (el) |
SI (1) | SI1385548T1 (el) |
SK (1) | SK9492003A3 (el) |
WO (1) | WO2002058731A2 (el) |
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