HK1055749A1 - Process for the synthesis of an lhrh peptide - Google Patents

Process for the synthesis of an lhrh peptide

Info

Publication number
HK1055749A1
HK1055749A1 HK03107934A HK03107934A HK1055749A1 HK 1055749 A1 HK1055749 A1 HK 1055749A1 HK 03107934 A HK03107934 A HK 03107934A HK 03107934 A HK03107934 A HK 03107934A HK 1055749 A1 HK1055749 A1 HK 1055749A1
Authority
HK
Hong Kong
Prior art keywords
peptide
synthesis
lhrh peptide
protecting group
residue
Prior art date
Application number
HK03107934A
Other languages
English (en)
Inventor
Steven Allen Jackson
Original Assignee
Ipsen Mfg Ireland Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ipsen Mfg Ireland Ltd filed Critical Ipsen Mfg Ireland Ltd
Publication of HK1055749A1 publication Critical patent/HK1055749A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • C07K1/068General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for heterocyclic side chains
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/23Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Analytical Chemistry (AREA)
  • Endocrinology (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HK03107934A 2000-12-22 2003-11-04 Process for the synthesis of an lhrh peptide HK1055749A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IE20001079 2000-12-22
PCT/IE2001/000159 WO2002051861A2 (en) 2000-12-22 2001-12-19 Process for the synthesis of a peptide having a tryptophan residue

Publications (1)

Publication Number Publication Date
HK1055749A1 true HK1055749A1 (en) 2004-01-21

Family

ID=11042704

Family Applications (1)

Application Number Title Priority Date Filing Date
HK03107934A HK1055749A1 (en) 2000-12-22 2003-11-04 Process for the synthesis of an lhrh peptide

Country Status (25)

Country Link
US (1) US7122628B2 (cs)
EP (1) EP1343808B1 (cs)
JP (1) JP4064817B2 (cs)
KR (1) KR100591832B1 (cs)
CN (2) CN101003563A (cs)
AT (1) ATE339442T1 (cs)
AU (1) AU2002222439C1 (cs)
BR (1) BR0116447B1 (cs)
CA (1) CA2432708C (cs)
CZ (1) CZ299141B6 (cs)
DE (1) DE60123115T2 (cs)
DK (1) DK1343808T3 (cs)
ES (1) ES2266104T3 (cs)
HK (1) HK1055749A1 (cs)
HU (2) HU230601B1 (cs)
IE (1) IES20011090A2 (cs)
IL (2) IL156258A0 (cs)
MX (1) MXPA03005678A (cs)
NO (1) NO325038B1 (cs)
NZ (1) NZ526990A (cs)
PL (1) PL205949B1 (cs)
PT (1) PT1343808E (cs)
RU (1) RU2276156C2 (cs)
WO (1) WO2002051861A2 (cs)
ZA (1) ZA200304809B (cs)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7091311B2 (en) 1996-06-07 2006-08-15 Smithkline Beecham Corporation Peptides and compounds that bind to a receptor
BR0314591A (pt) 2002-09-18 2005-08-09 Ortho Mcneil Pharm Inc Métodos de aumento de plaquetas e produção de célula tronco hematopoiética
DK1675606T3 (en) * 2003-08-28 2017-06-19 Janssen Pharmaceuticals Inc Peptides and compound that bind to thrombopoietin receptors
EP1968995A1 (en) * 2005-12-30 2008-09-17 F. Hoffmann-la Roche AG Methods for the synthesis of arginine-containing peptides
WO2014047822A1 (zh) * 2012-09-27 2014-04-03 深圳翰宇药业股份有限公司 一种制备布舍瑞林的方法
US10308677B2 (en) 2014-12-19 2019-06-04 Cem Corporation Coupling method for peptide synthesis at elevated temperatures
US9969769B2 (en) 2014-12-19 2018-05-15 Cem Corporation Coupling method for peptide synthesis at elevated temperatures

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4211693A (en) 1977-09-20 1980-07-08 The Salk Institute For Biological Studies Peptides with para-substituted phenylalanine
US4569927A (en) * 1984-02-23 1986-02-11 The Salk Institute For Biological Studies GnRH Antagonists IV
IL74827A (en) 1984-05-21 1989-06-30 Salk Inst For Biological Studi Peptides active as gnrh antagonists and pharmaceutical compositions containing them
IT1203600B (it) * 1985-12-06 1989-02-15 Phidea Srl Metodo per preparare il (d-trp6)-lhrh
US5175254A (en) * 1988-09-24 1992-12-29 Societe D'expansion Scientifque Expansia Solid phase peptide synthesis using a polyacrylic support in aqueous solution
GB8822502D0 (en) * 1988-09-24 1988-10-26 Expansia Sa New peptide synthesis method
JPH05331188A (ja) 1992-05-28 1993-12-14 Nippon Chemiphar Co Ltd トリペプチド、その製造方法及びエンドセリン拮抗剤

Also Published As

Publication number Publication date
PT1343808E (pt) 2007-01-31
CA2432708A1 (en) 2002-07-04
HUP0302633A2 (hu) 2003-12-29
PL205949B1 (pl) 2010-06-30
EP1343808B1 (en) 2006-09-13
IES20011090A2 (en) 2002-12-30
HUP0302633A3 (en) 2008-04-28
MXPA03005678A (es) 2003-10-06
CZ299141B6 (cs) 2008-04-30
EP1343808A2 (en) 2003-09-17
NO325038B1 (no) 2008-01-21
ES2266104T3 (es) 2007-03-01
KR100591832B1 (ko) 2006-06-20
KR20030081355A (ko) 2003-10-17
AU2002222439C1 (en) 2005-10-27
BR0116447B1 (pt) 2014-04-29
WO2002051861A3 (en) 2002-10-10
NO20032852L (no) 2003-08-22
CN101003563A (zh) 2007-07-25
ZA200304809B (en) 2004-04-20
JP4064817B2 (ja) 2008-03-19
IL156258A (en) 2008-06-05
BR0116447A (pt) 2003-10-07
WO2002051861A2 (en) 2002-07-04
NO20032852D0 (no) 2003-06-20
HUP1400157A2 (en) 2003-12-29
DK1343808T3 (da) 2006-12-11
CA2432708C (en) 2011-07-12
RU2003122779A (ru) 2005-02-20
JP2004516330A (ja) 2004-06-03
PL361993A1 (en) 2004-10-18
NZ526990A (en) 2005-04-29
AU2002222439B2 (en) 2005-04-07
DE60123115T2 (de) 2007-03-29
US7122628B2 (en) 2006-10-17
CN1481389A (zh) 2004-03-10
DE60123115D1 (de) 2006-10-26
IL156258A0 (en) 2004-01-04
HU230601B1 (hu) 2017-02-28
HU229701B1 (en) 2014-05-28
ATE339442T1 (de) 2006-10-15
CZ20031634A3 (cs) 2003-09-17
US20040077827A1 (en) 2004-04-22
RU2276156C2 (ru) 2006-05-10

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Legal Events

Date Code Title Description
CHPA Change of a particular in the register (except of change of ownership)
PE Patent expired

Effective date: 20211218