HK1039317A1 - 半胱氨酸蛋白酶ice/ced-3家族的(取代)的酰基二肽抑 - Google Patents

半胱氨酸蛋白酶ice/ced-3家族的(取代)的酰基二肽抑

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Publication number
HK1039317A1
HK1039317A1 HK02100909.8A HK02100909A HK1039317A1 HK 1039317 A1 HK1039317 A1 HK 1039317A1 HK 02100909 A HK02100909 A HK 02100909A HK 1039317 A1 HK1039317 A1 HK 1039317A1
Authority
HK
Hong Kong
Prior art keywords
ced
ice
family
substituted
cysteine proteases
Prior art date
Application number
HK02100909.8A
Other languages
English (en)
Inventor
S Karanewsky Donald
J Kalish Vincent
D Robinson Edward
R Ullman Brett
Original Assignee
Idun Pharmaceuticals Inc
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Filing date
Publication date
Application filed by Idun Pharmaceuticals Inc filed Critical Idun Pharmaceuticals Inc
Publication of HK1039317A1 publication Critical patent/HK1039317A1/zh

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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07K5/08—Tripeptides
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    • C07C2601/14—The ring being saturated
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    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline
    • C—CHEMISTRY; METALLURGY
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    • C07C2603/58—Ring systems containing bridged rings containing three rings
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HK02100909.8A 1998-10-22 2002-02-06 半胱氨酸蛋白酶ice/ced-3家族的(取代)的酰基二肽抑 HK1039317A1 (zh)

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WO2000023421A1 (en) 2000-04-27
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