HK1009273A1 - Sertindole prodrugs - Google Patents

Sertindole prodrugs

Info

Publication number
HK1009273A1
HK1009273A1 HK98110040A HK98110040A HK1009273A1 HK 1009273 A1 HK1009273 A1 HK 1009273A1 HK 98110040 A HK98110040 A HK 98110040A HK 98110040 A HK98110040 A HK 98110040A HK 1009273 A1 HK1009273 A1 HK 1009273A1
Authority
HK
Hong Kong
Prior art keywords
sertindole
group
prodrugs
iii
optionally substituted
Prior art date
Application number
HK98110040A
Other languages
English (en)
Inventor
Jens Kristian Perregaard
Henrik Perdersen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of HK1009273A1 publication Critical patent/HK1009273A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Curing Cements, Concrete, And Artificial Stone (AREA)
  • Pyrane Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Inorganic Compounds Of Heavy Metals (AREA)
  • Indole Compounds (AREA)
HK98110040A 1990-10-03 1998-08-20 Sertindole prodrugs HK1009273A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK238190A DK238190D0 (da) 1990-10-03 1990-10-03 Depotderivater
PCT/DK1991/000291 WO1992006089A1 (en) 1990-10-03 1991-09-27 Sertindole prodrugs

Publications (1)

Publication Number Publication Date
HK1009273A1 true HK1009273A1 (en) 1999-05-28

Family

ID=8111993

Family Applications (1)

Application Number Title Priority Date Filing Date
HK98110040A HK1009273A1 (en) 1990-10-03 1998-08-20 Sertindole prodrugs

Country Status (21)

Country Link
US (1) US5428036A (ko)
EP (1) EP0592433B1 (ko)
JP (1) JP3100980B2 (ko)
KR (1) KR100212430B1 (ko)
AT (1) ATE175964T1 (ko)
AU (1) AU652783B2 (ko)
CA (1) CA2093433C (ko)
DE (1) DE69130803T2 (ko)
DK (2) DK238190D0 (ko)
ES (1) ES2125870T3 (ko)
FI (1) FI102679B (ko)
GR (1) GR3029399T3 (ko)
HK (1) HK1009273A1 (ko)
IE (1) IE913384A1 (ko)
IL (1) IL99652A (ko)
NO (1) NO301475B1 (ko)
NZ (1) NZ240051A (ko)
PH (1) PH30129A (ko)
PT (1) PT99142B (ko)
WO (1) WO1992006089A1 (ko)
ZA (1) ZA917881B (ko)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5776963A (en) 1989-05-19 1998-07-07 Hoechst Marion Roussel, Inc. 3-(heteroaryl)-1- (2,3-dihydro-1h-isoindol-2-yl)alkyl!pyrrolidines and 3-(heteroaryl)-1- (2,3-dihydro-1h-indol-1-yl)alkyl!pyrrolidines and related compounds and their therapeutic untility
US5643784A (en) * 1990-12-04 1997-07-01 H, Lundbeck A/S Indan derivatives
NZ243065A (en) * 1991-06-13 1995-07-26 Lundbeck & Co As H Piperidine derivatives and pharmaceutical compositions
DK206591D0 (da) * 1991-12-23 1991-12-23 Lundbeck & Co As H Behandling af psykoser
JPH0625964U (ja) * 1992-05-25 1994-04-08 ミクロン機器株式会社 通信機能付きコインカウンタ及び有料装置
US6489341B1 (en) * 1999-06-02 2002-12-03 Sepracor Inc. Methods for the treatment of neuroleptic and related disorders using sertindole derivatives
WO2002076404A2 (en) 2001-03-23 2002-10-03 Protarga, Inc. Fatty alcohol drug conjugates
AU2002303164A1 (en) 2001-03-23 2002-10-08 Protarga, Inc. Fatty amine drug conjugates
US20100168197A1 (en) * 2007-02-28 2010-07-01 Naresh Kumar Muscarinic receptor antagonists
HRP20171415T4 (hr) 2009-06-25 2023-03-03 Alkermes Pharma Ireland Limited Heterociklični spojevi za liječenje neuroloških i psiholoških poremećaja
WO2010151711A1 (en) 2009-06-25 2010-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds
WO2011163594A2 (en) * 2010-06-24 2011-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
CN112423754A (zh) 2018-03-05 2021-02-26 奥克梅斯制药爱尔兰有限公司 阿立哌唑的给药策略

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3408356A (en) * 1965-08-31 1968-10-29 Squibb & Sons Inc Long chain esters of 4'-fluoro-4-[4-hydroxy-4-(alpha, alpha, alpha-trifluorotolyl)piperi-dino]butyrophenone and the like
US4038305A (en) * 1972-03-20 1977-07-26 Aktieselskabet Grindstedvaerket Cyclopentenone derivatives
GB1469108A (en) * 1973-06-25 1977-03-30 Kefalas As Thiaxanthene derivative
JPS568318A (en) * 1979-06-28 1981-01-28 Janssen Pharmaceutica Nv Non oral long acting composition of haloperidol and bromperidol derivative
IT1199116B (it) * 1984-07-03 1988-12-30 Fidia Farmaceutici Derivati di gangliosidi
IE58370B1 (en) * 1985-04-10 1993-09-08 Lundbeck & Co As H Indole derivatives
GB8621892D0 (en) * 1986-09-11 1986-10-15 Lundbeck & Co As H Organic compound
GB8908085D0 (en) * 1989-04-11 1989-05-24 Lundbeck & Co As H New therapeutic use
DE3921886A1 (de) * 1989-07-04 1991-01-17 Wolfgang Mohr Vorrichtung zum schneiden von gestapeltem, blattfoermigen gut

Also Published As

Publication number Publication date
DK238190D0 (da) 1990-10-03
NO931219L (no) 1993-04-01
ZA917881B (en) 1992-07-29
CA2093433C (en) 2000-11-21
IE913384A1 (en) 1992-04-08
PT99142A (pt) 1994-02-28
FI931472A (fi) 1993-04-01
CA2093433A1 (en) 1992-04-04
IL99652A (en) 1997-04-15
NO931219D0 (no) 1993-03-31
ATE175964T1 (de) 1999-02-15
EP0592433A1 (en) 1994-04-20
WO1992006089A1 (en) 1992-04-16
GR3029399T3 (en) 1999-05-28
FI102679B1 (fi) 1999-01-29
DE69130803D1 (de) 1999-03-04
US5428036A (en) 1995-06-27
KR100212430B1 (ko) 1999-08-02
FI102679B (fi) 1999-01-29
AU652783B2 (en) 1994-09-08
DE69130803T2 (de) 1999-08-19
NZ240051A (en) 1993-05-26
PT99142B (pt) 1999-04-30
IL99652A0 (en) 1992-08-18
KR930702335A (ko) 1993-09-08
PH30129A (en) 1997-01-21
FI931472A0 (fi) 1993-04-01
AU8710491A (en) 1992-04-28
EP0592433B1 (en) 1999-01-20
ES2125870T3 (es) 1999-03-16
JPH06501939A (ja) 1994-03-03
NO301475B1 (no) 1997-11-03
DK0592433T3 (da) 1999-09-13
JP3100980B2 (ja) 2000-10-23

Similar Documents

Publication Publication Date Title
ZA917881B (en) Sertindole prodrugs
IL104305A0 (en) Piperazine derivatives,their preparation and pharmaceutical compositions containing them
ES8305356A1 (es) Un procedimiento para la produccion de un derivado de carbostirilo
KR850003719A (ko) 시아노피라졸 제초제에 대한 개량
SG76479A1 (en) Pleuromutilin derivatives
TW238304B (en) A process for the preparation of 1-substituted-5(4H)-tetrazolinones
ES475588A1 (es) Procedimiento para la obtencion de derivados del acido inde-no -2,1-b- tiofen-2-oxamico
ATE70531T1 (de) Carbacyclinester, verfahren zu ihrer herstellung und ihre verwendung in der medizin.
GR3032285T3 (en) Process and intermediates for bis-aza-bicyclic anxiolytic agents.
ATE19879T1 (de) Furyloxazolylessigsaeure-derivate, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzungen.
ATE36520T1 (de) Polyprenylverbindung, ihre herstellung und pharmazeutische verwendung.
DE69327092D1 (de) Optisch aktives 1-phenylpyrrolidonderivat und dessen herstellung
HUT53638A (en) Process for producing 15-amino-substituted 20,21-dinoreburnamenie derivatives and pharmaceutical compositions containing them
ES8200112A1 (es) Un procedimiento para la preparacion de un derivado del aci do clavulanico.

Legal Events

Date Code Title Description
PF Patent in force
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20080927